Topic leaderboard
Therapeutic activity of chemical compounds
Ranked by the PatentIndex Score — a 1–99 percentile within A61P · public-visibility date · generated 2026-07-19
top 25 per window · public-visibility date
Rising· last 2 yrs
Inventors whose newest A61P patents became public in the last 2 years — the current frontier
- 199Svetlana O. Doronina29 patents · 3,971 citations
- 296Drew Weissman23 patents · 1,412 citations
- 392Jason Mccartney72 patents · 4,104 citations
- 488Thomas J. Magliery18 patents · 1,517 citations
- 583Fei Ran12 patents · 2,383 citations
- 679Sara S. Hadida Ruah84 patents · 4,044 citations
- 775Serengulam V. Govindan82 patents · 2,118 citations
- 871Stacey Shepard58 patents · 2,323 citations
- 967Haiyong Hugh Huang63 patents · 1,552 citations
- 1063Richard O. Mannion42 patents · 1,176 citations
- 1158Edward P. O'Donnell41 patents · 1,166 citations
- 1254William H. Mckenna41 patents · 1,166 citations
- 1350Samuel Davis46 patents · 1,582 citations
- 1446Ketan Mehta31 patents · 1,964 citations
- 1542Yu-Hsing Tu34 patents · 1,736 citations
- 1638Stacey R. Dillon40 patents · 706 citations
- 1733Daniel Dix38 patents · 1,668 citations
- 1829Herriot Tabuteau197 patents · 9,344 citations
- 1925Kelly Frye24 patents · 1,347 citations
- 2021Kenneth S. Graham22 patents · 942 citations
- 2117Wei Dang25 patents · 1,541 citations
- 2213Giuseppe Ciaramella53 patents · 1,656 citations
- 238John Spencer Emtage12 patents · 3,803 citations
- 244James P. Rizzi38 patents · 2,054 citations
- 251Jiazhong Zhang53 patents · 2,179 citations
Active· last 5 yrs
Sustained A61P output across the last 5 years
- 199Louis Fries10 patents · 3,343 citations
- 296Mauricio R. Alvira35 patents · 2,978 citations
- 392Svetlana O. Doronina29 patents · 3,971 citations
- 488Michael C. Milone36 patents · 3,207 citations
- 583Michael D. Kalos22 patents · 3,096 citations
- 679Bruce L. Levine32 patents · 3,087 citations
- 775David L. Porter17 patents · 3,065 citations
- 871Brian Mcguinness20 patents · 3,034 citations
- 967Roland A. Newman24 patents · 4,038 citations
- 1063Gerald Mcmahon38 patents · 2,990 citations
- 1158Somasekhar Bhamidipati140 patents · 3,661 citations
- 1254Jeffrey Clough86 patents · 3,429 citations
- 1350Holger Keim61 patents · 3,198 citations
- 1446Sacha Holland84 patents · 2,331 citations
- 1542Sue Fletcher40 patents · 2,334 citations
- 1638Graham Mcclorey32 patents · 2,030 citations
- 1733Lloyd Jeffs12 patents · 1,782 citations
- 1829Stephane Bancel14 patents · 1,595 citations
- 1925Christopher Breder54 patents · 1,438 citations
- 2021Tirtha Chakraborty27 patents · 1,681 citations
- 2117Lik Hon15 patents · 1,710 citations
- 2213Jesper Wengel18 patents · 3,039 citations
- 238Roger Shen-Chu Chen54 patents · 2,695 citations
- 244Francis Burrows13 patents · 2,429 citations
- 251Katalin Kariko14 patents · 1,413 citations
All-time canon
Career PatentIndex Score in A61P
- 199Cary L. Queen12 patents · 26,158 citations
- 296Harold E. Selick7 patents · 25,683 citations
- 392Sharon Kaye Spratt8 patents · 3,914 citations
- 488Geoffrey Walter Grigg10 patents · 4,903 citations
- 583John B. Ridgway7 patents · 5,694 citations
- 679Benjamin Oshlack128 patents · 11,069 citations
- 775Mark Chasin53 patents · 8,550 citations
- 871Philip Ross Hamann13 patents · 5,036 citations
- 967Irwin Hollander5 patents · 4,871 citations
- 1063Woonza M. Rhee11 patents · 4,847 citations
- 1158Frank Delustro10 patents · 4,810 citations
- 1254Robert F. Kaiko24 patents · 5,159 citations
- 1350Louis Fries10 patents · 3,343 citations
- 1446Paul Sakorafas18 patents · 3,719 citations
- 1542Hua-Pin Huang50 patents · 3,712 citations
- 1638Mauricio R. Alvira35 patents · 2,978 citations
- 1733Hanne Bentz10 patents · 3,671 citations
- 1829Ramon A. Burns, Jr.7 patents · 3,045 citations
- 1925Svetlana O. Doronina29 patents · 3,971 citations
- 2021Brian E. Toki16 patents · 3,412 citations
- 2117Michael C. Milone36 patents · 3,207 citations
- 2213Michael D. Kalos22 patents · 3,096 citations
- 238Bruce L. Levine32 patents · 3,087 citations
- 244David L. Porter17 patents · 3,065 citations
- 251Robert Hudziak13 patents · 3,557 citations
Rising· last 2 yrs
The top-scoring A61P patents made public in the last 2 years
- 199US11883373B1✦ AITreatment of depression in certain patient populations30 cites · 202472% earned
- 296US11925636B2✦ AIBupropion dosage forms with reduced food and alcohol dosing effects28 cites · 202475% earned
- 392US12097263B2✦ AIMuscle targeting complexes and uses thereof for treating myotonic dystrophy18 cites · 202481% earned
- 488US12005124B2Muscle targeting complexes and uses thereof for treating dystrophinopathies23 cites · 202473% earned
- 583US12018087B2Muscle-targeting complexes comprising an anti-transferrin receptor antibody linked to an o23 cites · 202477% earned
- 679US12156914B2Pharmaceutical compositions comprising bupropion and cysteine23 cites · 202477% earned
- 775US12012460B2Muscle-targeting complexes comprising an anti-transferrin receptor antibody linked to an o22 cites · 202471% earned
- 871US11986444B2Treatment of poor metabolizers of dextromethorphan with a combination of bupropion and dex22 cites · 202480% earned
- 967US12491184B2Compositions and methods of use for modified release minoxidil7 cites · 202554% earned
- 1063US12144868B2Muscle targeting complexes and uses thereof for treating dystrophinopathies14 cites · 202475% earned
- 1158US11999947B2Adenosine nucleobase editors and uses thereof18 cites · 202477% earned
- 1254US12128109B2Muscle targeting complexes and formulations for treating dystrophinopathies17 cites · 202484% earned
- 1350US12268693B2Pharmaceutical compositions comprising a tolfenamic acid11 cites · 202478% earned
- 1446US12070459B2Pharmaceutical capsule compositions comprising lumateperone mono-tosylate16 cites · 202472% earned
- 1542US12138260B2Compounds and combinations thereof for treating neurological and psychiatric conditions16 cites · 202478% earned
- 1638US12128052B2Pharmaceutical compositions comprising meloxicam13 cites · 202470% earned
- 1733US12090155B2Methods13 cites · 202479% earned
- 1829US12005118B2Pharmaceutical compositions comprising meloxicam13 cites · 202483% earned
- 1925US12318397B1Methods and compositions for testosterone production4 cites · 202562% earned
- 2021US12329825B1Muscle targeting complexes comprising an anti-transferrin receptor antibody linked to an o4 cites · 202570% earned
- 2117US12447148B2Methods of improving lung function4 cites · 202582% earned
- 2213US12115142B2Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics10 cites · 202465% earned
- 238US12246023B2Use of reboxetine to treat narcolepsy10 cites · 202470% earned
- 244US12097175B2Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics9 cites · 202466% earned
- 251US12365669B2THRβ receptor agonist compound and preparation method and use thereof3 cites · 202559% earned
Active· last 5 yrs
The top-scoring A61P patents of the last 5 years
- 199US10953089B1✦ AICoronavirus vaccine formulations99 cites · 202183% earned
- 296US11147808B2✦ AIMethod of decreasing the fluctuation index of dextromethorphan82 cites · 202193% earned
- 392US11191739B2✦ AIBupropion as a modulator of drug activity82 cites · 202193% earned
- 488US11447770B1Methods and compositions for prime editing nucleotide sequences81 cites · 202278% earned
- 583US10925842B2Bupropion as a modulator of drug activity97 cites · 202193% earned
- 679US11197839B2Bupropion as a modulator of drug activity78 cites · 202193% earned
- 775US10980800B2Bupropion as a modulator of drug activity93 cites · 202193% earned
- 871US11253492B2Bupropion as a modulator of drug activity77 cites · 202193% earned
- 967US11298352B2Bupropion as a modulator of drug activity74 cites · 202193% earned
- 1063US11020389B2Bupropion as a modulator of drug activity87 cites · 202193% earned
- 1158US11291638B2Bupropion as a modulator of drug activity72 cites · 202193% earned
- 1254US11344544B2Bupropion as a modulator of drug activity71 cites · 202189% earned
- 1350US11253491B2Bupropion as a modulator of drug activity71 cites · 202193% earned
- 1446US11291665B2Bupropion as a modulator of drug activity71 cites · 202193% earned
- 1542US11207281B2Bupropion as a modulator of drug activity84 cites · 202193% earned
- 1638US11285118B2Bupropion as a modulator of drug activity69 cites · 202286% earned
- 1733US11229640B2Combination of dextromethorphan and bupropion for treating depression80 cites · 202193% earned
- 1829US11419867B2Bupropion as a modulator of drug activity66 cites · 202292% earned
- 1925US11123343B2Bupropion as a modulator of drug activity79 cites · 202193% earned
- 2021US11213521B2Bupropion as a modulator of drug activity79 cites · 202193% earned
- 2117US11111309B2Method of reducing expression of DUX4 in a muscle cell by administering an anti-transferri65 cites · 202177% earned
- 2213US11730706B1Treatment of depression in certain patient populations39 cites · 202373% earned
- 238US11141388B2Bupropion as a modulator of drug activity78 cites · 202189% earned
- 244US11426370B2Bupropion as a modulator of drug activity65 cites · 202192% earned
- 251US11058648B2Bupropion as a modulator of drug activity77 cites · 202193% earned
All-time canon
The defining A61P patents of the whole record
- 199US5585089A✦ AIHumanized immunoglobulins7,465 cites · 199690% earned
- 296US5530101A✦ AIHumanized immunoglobulins5,773 cites · 199690% earned
- 392US5693762A✦ AIHumanized immunoglobulins5,271 cites · 199790% earned
- 488US5821337AImmunoglobulin variants4,043 cites · 199891% earned
- 583US6180370B1Humanized immunoglobulins and methods of making the same3,646 cites · 200189% earned
- 679US6737056B1Polypeptide variants with altered effector function3,376 cites · 200487% earned
- 775US5693761APolynucleotides encoding improved humanized immunoglobulins3,290 cites · 199789% earned
- 871US4816397AMultichain polypeptides or proteins and processes for their production3,126 cites · 198996% earned
- 967US6506559B1Genetic inhibition by double-stranded RNA3,119 cites · 200387% earned
- 1063US5013556ALiposomes with enhanced circulation time2,874 cites · 199194% earned
- 1158US5770429ATransgenic non-human animals capable of producing heterologous antibodies2,663 cites · 199896% earned
- 1254US5731168AMethod for making heteromultimeric polypeptides2,644 cites · 199888% earned
- 1350US6054297AHumanized antibodies and methods for making them2,266 cites · 200096% earned
- 1446US8008449B2Human monoclonal antibodies to programmed death 1 (PD-1) and methods for treating cancer u2,199 cites · 200987% earned
- 1542US6407213B1Method for making humanized antibodies2,158 cites · 200291% earned
- 1638US5539082APeptide nucleic acids2,083 cites · 199693% earned
- 1733US6544212B2Diabetes management system2,056 cites · 200396% earned
- 1829US4670417AHemoglobin combined with a poly(alkylene oxide)2,034 cites · 198796% earned
- 1925US4496689ACovalently attached complex of alpha-1-proteinase inhibitor with a water soluble polymer1,835 cites · 198596% earned
- 2021US6596296B1Drug releasing biodegradable fiber implant1,834 cites · 200392% earned
- 2117US6248363B1Solid carriers for improved delivery of active ingredients in pharmaceutical compositions1,826 cites · 200187% earned
- 2213US6602684B1Glycosylation engineering of antibodies for improving antibody-dependent cellular cytotoxi1,819 cites · 200387% earned
- 238US5641870ALow pH hydrophobic interaction chromatography for antibody purification1,818 cites · 199789% earned
- 244US7108701B2Drug releasing anastomosis devices and methods for treating anastomotic sites1,784 cites · 200396% earned
- 251US6749587B2Modular infusion device and method1,768 cites · 200293% earned
Rising· last 2 yrs
Assignees whose newest A61P patents became public in the last 2 years — the current frontier
- 199GENENTECH INC1,383 patents · 60,723 citations
- 296LIPOCINE INC52 patents · 6,133 citations
- 392UNIV IOWA RES FOUND141 patents · 8,001 citations
- 488UNIV TEXAS927 patents · 20,041 citations
- 583UNIV PENNSYLVANIA634 patents · 13,492 citations
- 679US HEALTH1,266 patents · 28,710 citations
- 775AMGEN INC960 patents · 22,626 citations
- 871UNIV CALIFORNIA1,901 patents · 30,707 citations
- 967CHILDRENS MEDICAL CENTER259 patents · 7,651 citations
- 1063IMMUNOMEDICS INC226 patents · 11,272 citations
- 1158BRISTOL MYERS SQUIBB CO2,066 patents · 40,102 citations
- 1254IMMUNOGEN INC163 patents · 9,285 citations
- 1350PURDUE PHARMA LP381 patents · 8,617 citations
- 1446CELGENE CORP353 patents · 8,962 citations
- 1542BROAD INST INC120 patents · 3,413 citations
- 1638PURDUE RESEARCH FOUNDATION194 patents · 7,278 citations
- 1733RIGEL PHARMACEUTICALS INC264 patents · 4,427 citations
- 1829PFIZER2,457 patents · 43,131 citations
- 1925UNIV MASSACHUSETTS255 patents · 5,264 citations
- 2021UNIV ARIZONA154 patents · 7,233 citations
- 2117UNIV NEW YORK232 patents · 4,046 citations
- 2213SCRIPPS RESEARCH INST362 patents · 9,599 citations
- 238MILLENNIUM PHARM INC361 patents · 6,299 citations
- 244REGENERON PHARMA665 patents · 9,329 citations
- 251VERTEX PHARMA719 patents · 22,769 citations
Active· last 5 yrs
Sustained A61P output across the last 5 years
- 199GENENTECH INC1,383 patents · 60,723 citations
- 296LIPOCINE INC52 patents · 6,133 citations
- 392UNIV IOWA RES FOUND141 patents · 8,001 citations
- 488UNIV TEXAS927 patents · 20,041 citations
- 583UNIV PENNSYLVANIA634 patents · 13,492 citations
- 679WISCONSIN ALUMNI RES FOUND457 patents · 11,086 citations
- 775GLAUKOS CORP12 patents · 2,133 citations
- 871US HEALTH1,266 patents · 28,710 citations
- 967AMGEN INC960 patents · 22,626 citations
- 1063MAX PLANCK GESELLSCHAFT132 patents · 4,686 citations
- 1158UNIV CALIFORNIA1,901 patents · 30,707 citations
- 12543M INNOVATIVE PROPERTIES CO230 patents · 18,111 citations
- 1350CHILDRENS MEDICAL CENTER259 patents · 7,651 citations
- 1446IMMUNOMEDICS INC226 patents · 11,272 citations
- 1542BRISTOL MYERS SQUIBB CO2,066 patents · 40,102 citations
- 1638ETHICON INC51 patents · 5,533 citations
- 1733IMMUNOGEN INC163 patents · 9,285 citations
- 1829PURDUE PHARMA LP381 patents · 8,617 citations
- 1925CELGENE CORP353 patents · 8,962 citations
- 2021BROAD INST INC120 patents · 3,413 citations
- 2117PURDUE RESEARCH FOUNDATION194 patents · 7,278 citations
- 2213RIGEL PHARMACEUTICALS INC264 patents · 4,427 citations
- 238ALEXZA PHARMACEUTICALS INC73 patents · 4,579 citations
- 244WARNER LAMBERT CO636 patents · 23,110 citations
- 251PFIZER2,457 patents · 43,131 citations
All-time canon
All-time PatentIndex Score in A61P
- 199PROTEIN DESIGN LABS INC13 patents · 26,501 citations
- 296GENENTECH INC1,383 patents · 60,723 citations
- 392SANGAMO BIOSCIENCES INC67 patents · 6,793 citations
- 488ISIS PHARMACEUTICALS INC300 patents · 33,197 citations
- 583MEDICAL RES COUNCIL56 patents · 6,150 citations
- 679LIPOCINE INC52 patents · 6,133 citations
- 775UNIV IOWA RES FOUND141 patents · 8,001 citations
- 871MEDAREX INC67 patents · 10,134 citations
- 967UNIV TEXAS927 patents · 20,041 citations
- 1063UNIV PENNSYLVANIA634 patents · 13,492 citations
- 1158WISCONSIN ALUMNI RES FOUND457 patents · 11,086 citations
- 1254AMERICAN CYANAMID CO281 patents · 12,024 citations
- 1350EURO CELTIQUE SA145 patents · 15,354 citations
- 1446COLLAGEN CORP14 patents · 5,790 citations
- 1542CIBA GEIGY CORP460 patents · 15,521 citations
- 1638GLAUKOS CORP12 patents · 2,133 citations
- 1733US HEALTH1,266 patents · 28,710 citations
- 1829AMGEN INC960 patents · 22,626 citations
- 1925MAX PLANCK GESELLSCHAFT132 patents · 4,686 citations
- 2021UNIV CALIFORNIA1,901 patents · 30,707 citations
- 2117PHARMACYCLICS INC47 patents · 3,405 citations
- 2213SEATTLE GENETICS INC74 patents · 5,502 citations
- 2383M INNOVATIVE PROPERTIES CO230 patents · 18,111 citations
- 244ALEXZA MOLECULAR DELIVERY CORP20 patents · 2,255 citations
- 251IDEC PHARMA CORP25 patents · 4,719 citations
90–99 field-defining50–89 strong<50 emergingearned by citationsfrom family breadth