Assignee
PFIZER
4,152 granted patents·1,348 pending applications·74,074 citations·filing 1970–2025
Top patents by PatentIndex Score
5,500 records- 0199US5834450A9- (substituted amino) -alpha-6-deoxy-5-oxy tetracycline derivatives, their preparation and their use as antibioticsPFIZER·Filed 1995·Granted Nov 10, 1998·252 cites·8 claims
- 0299US5747498AAlkynyl and azido-substituted 4-anilinoquinazolinesPFIZER·Filed 1996·Granted May 5, 1998·1.2k cites·32 claims
- 0399US4831031AAryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activityPFIZER·Filed 1988·Granted May 16, 1989·307 cites·9 claims
- 0499US4188390AAntihypertensive 4-amino-2-[4-(1,4-benzodioxan-2-carbonyl) piperazin-1-yl or homopiperazin-1-yl]quinazolinesPFIZER·Filed 1978·Granted Feb 12, 1980·135 cites·6 claims
- 0598US11110160B2Glycoconjugation processes and compositionsPFIZER·Filed 2020·Granted Sep 7, 2021·6 cites·20 claims
- 0698US10851081B2GLP-1 receptor agonists and uses thereofPFIZER·Filed 2020·Granted Dec 1, 2020·12 cites·19 claims
- 0798US7655232B2Anti-NGF antibodies and methods using samePFIZER·Filed 2007·Granted Feb 2, 2010·60 cites·12 claims
- 0898US7288251B2Antibodies to CD40PFIZER·Filed 2002·Granted Oct 30, 2007·158 cites·22 claims
- 0998US7132281B2Methods and host cells for producing human monoclonal antibodies to CTLA-4PFIZER·Filed 2004·Granted Nov 7, 2006·220 cites·262 claims
- 1098US7125880B1Corticotropin releasing factor antagonistsPFIZER·Filed 2000·Granted Oct 24, 2006·97 cites·21 claims
- 1198US7109003B2Methods for expressing and recovering human monoclonal antibodies to CTLA-4PFIZER·Filed 2003·Granted Sep 19, 2006·287 cites·101 claims
- 1298US6706283B1Controlled release by extrusion of solid amorphous dispersions of drugsPFIZER·Filed 2000·Granted Mar 16, 2004·202 cites·71 claims
- 1398US6603008B1Sulfamoylheleroaryl pyrazole compounds as anti-inflammatory/analgesic agentsPFIZER·Filed 2000·Granted Aug 5, 2003·600 cites·3 claims
- 1498US6436938B1Combination treatment for depressionPFIZER·Filed 2001·Granted Aug 20, 2002·176 cites·30 claims
- 1598US6235764B1Isothiazole derivatives useful as anticancer agentsPFIZER·Filed 1999·Granted May 22, 2001·261 cites·23 claims
- 1698US5863949AArylsulfonylamino hydroxamic acid derivativesPFIZER·Filed 1995·Granted Jan 26, 1999·528 cites·13 claims
- 1798US5861510AArylsulfonyl hydroxamic acid derivatives as MMP and TNF inhibitorsPFIZER·Filed 1995·Granted Jan 19, 1999·536 cites·11 claims
- 1898US5593997A4-aminopyrazolo(3-,4-D)pyrimidine and 4-aminopyrazolo-(3,4-D)pyridine tyrosine kinase inhibitorsPFIZER·Filed 1995·Granted Jan 14, 1997·355 cites·16 claims
- 1998US5431921ADispensing device containing a hydrophobic mediumPFIZER·Filed 1991·Granted Jul 11, 1995·834 cites·9 claims
- 2098US5306726A3-aryl-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agentsPFIZER·Filed 1992·Granted Apr 26, 1994·112 cites·4 claims
- 2198US5250534APyrazolopyrimidinone antianginal agentsPFIZER·Filed 1992·Granted Oct 5, 1993·276 cites·8 claims
- 2298US5059609ASubstituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseasesPFIZER·Filed 1989·Granted Oct 22, 1991·98 cites·35 claims
- 2398US5030654AGlutaramide diuretic agentsPFIZER·Filed 1989·Granted Jul 9, 1991·172 cites·38 claims
- 2498US4939140AHeterocyclic oxophthalazinyl acetic acidsPFIZER·Filed 1988·Granted Jul 3, 1990·112 cites·29 claims
- 2598US4803076AControlled release device for an active substancePFIZER·Filed 1986·Granted Feb 7, 1989·238 cites·39 claims
- 2698US4710507AQuinolone inotropic agentsPFIZER·Filed 1984·Granted Dec 1, 1987·57 cites·6 claims
- 2798US4619924A2-alkylthiopenem derivativesPFIZER·Filed 1984·Granted Oct 28, 1986·66 cites·24 claims
- 2898US4572909A2-(Secondary aminoalkoxymethyl) dihydropyridine derivatives as anti-ischaemic and antihypertensive agentsPFIZER·Filed 1984·Granted Feb 25, 1986·241 cites·17 claims
- 2998US4536518AAntidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenaminePFIZER·Filed 1979·Granted Aug 20, 1985·278 cites·22 claims
- 3098US4474768AN-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates thereforPFIZER·Filed 1982·Granted Oct 2, 1984·246 cites·8 claims
- 3198US4411925ABranched amides of L-aspartyl-d-amino acid dipeptidesPFIZER·Filed 1980·Granted Oct 25, 1983·155 cites·94 claims
- 3298US4404216AAntifungal 1,3-bis-triazolyl-2-propanol derivativePFIZER·Filed 1982·Granted Sep 13, 1983·83 cites·3 claims
- 3398US4399163ABranched amides of L-aspartyl-D-amino acid dipeptidesPFIZER·Filed 1981·Granted Aug 16, 1983·120 cites·20 claims
- 3498US4130714AHydantoin therapeutic agentsPFIZER·Filed 1977·Granted Dec 19, 1978·71 cites·5 claims
- 3598US4117230AHydantoin derivatives as therapeutic agentsPFIZER·Filed 1977·Granted Sep 26, 1978·62 cites·11 claims
- 3698US4024179ASubstituted ω-pentanorprostaglandinsPFIZER·Filed 1973·Granted May 17, 1977·52 cites·18 claims
- 3797US11702424B2Bicyclic-fused heteroaryl or aryl compoundsPFIZER·Filed 2020·Granted Jul 18, 2023·4 cites·8 claims
- 3897US11566006B2Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereofPFIZER·Filed 2021·Granted Jan 31, 2023·7 cites·20 claims
- 3997US11512070B2GLP-1 receptor agonists and uses thereofPFIZER·Filed 2020·Granted Nov 29, 2022·11 cites·16 claims
- 4097US11117928B2Glycoconjugation processPFIZER·Filed 2020·Granted Sep 14, 2021·4 cites·21 claims
- 4197US11014911B2CDK2 inhibitorsPFIZER·Filed 2020·Granted May 25, 2021·11 cites·4 claims
- 4297US10710966B1Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereofPFIZER·Filed 2020·Granted Jul 14, 2020·20 cites·24 claims
- 4397US10590087B1Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereofPFIZER·Filed 2019·Granted Mar 17, 2020·39 cites·18 claims
- 4497US10583187B2Glycoconjugation processes and compositionsPFIZER·Filed 2018·Granted Mar 10, 2020·17 cites·10 claims
- 4597US10550159B2Neisseria meningitidis composition and methods thereofPFIZER·Filed 2018·Granted Feb 4, 2020·11 cites·15 claims
- 4697US10208019B2GLP-1 receptor agonists and uses thereofPFIZER·Filed 2017·Granted Feb 19, 2019·50 cites·26 claims
- 4797US10196429B2Neisseria meningitidis composition and methods thereofPFIZER·Filed 2017·Granted Feb 5, 2019·12 cites·5 claims
- 4897US10071992B2Diacylglycerol acyl transferase 2 inhibitorsPFIZER·Filed 2017·Granted Sep 11, 2018·24 cites·24 claims
- 4997US9950054B2Glycoconjugation processes and compositionsPFIZER·Filed 2016·Granted Apr 24, 2018·24 cites·16 claims
- 5097US7803832B2N-(1-arylpyrazol-4L)sulfonamides and their use as parasiticidesPFIZER·Filed 2009·Granted Sep 28, 2010·88 cites·13 claims
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