US2023381119A1PendingUtilityA1

Use of histone acetyltransferase inhibitor amidoximes as anti-proliferative agents

Assignee: TEXAS WOMAN’S UNIVPriority: Oct 2, 2017Filed: Apr 7, 2023Published: Nov 30, 2023
Est. expiryOct 2, 2037(~11.2 yrs left)· nominal 20-yr term from priority
A61K 31/155A61K 33/24A61K 45/06A61P 35/00A61K 31/15
60
PatentIndex Score
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Claims

Abstract

Described herein is the use of bisamidoximes compounds for the treatment of HAT malfunction related pathologies.

Claims

exact text as granted — not AI-modified
1 - 7 . (canceled) 
     
     
         8 . A pharmaceutical composition comprising one or more bisamidoximes, wherein the one or more bisamidoximes are selected from the group of compounds consisting of JJMB 5, JJMB6, and JJMB 9: 
       
         
           
           
               
               
           
         
       
     
     
         9 . The pharmaceutical composition of  claim 8 , comprising two or more bisamidoximes. 
     
     
         10 . The pharmaceutical composition of  claim 8 , comprising JJMB5 and JJMB 9. 
     
     
         11 . The pharmaceutical composition of  claim 8 , comprising JJMB5. 
     
     
         12 . The pharmaceutical composition of  claim 8 , comprising JJMB6. 
     
     
         13 . The pharmaceutical composition of  claim 8 , comprising JJMB 9. 
     
     
         14 . The pharmaceutical composition of  claim 8 , further comprising an anticancer agent. 
     
     
         15 . The pharmaceutical composition of  claim 14 , wherein the anticancer agent is cisplatin. 
     
     
         16 . The pharmaceutical composition of  claim 8  being a therapeutically effective amount for inhibiting histone acetyltransferases (HATs) in a HAT malfunction related pathology. 
     
     
         17 . The pharmaceutical composition of  claim 8  being a therapeutically effective amount for treating colon cancer, breast cancer, or lung cancer in a subject. 
     
     
         18 . A pharmaceutical composition comprising one or more bisamidoximes, wherein the one or more bisamidoximes are selected from the group of compounds consisting of JJMB 5, JJMB6, JJMB 7, and JJMB 9: 
       
         
           
           
               
               
           
         
       
     
     
         19 . The pharmaceutical composition of  claim 18 , comprising two or more bisamidoximes. 
     
     
         20 . The pharmaceutical composition of  claim 18 , comprising JJMB5 and JJMB 9. 
     
     
         21 . The pharmaceutical composition of  claim 18 , comprising JJMB5 and JJMB7. 
     
     
         22 . The pharmaceutical composition of  claim 18 , comprising JJMB7 and JJMB 9. 
     
     
         23 . The pharmaceutical composition of  claim 18 , comprising JJMB 7. 
     
     
         24 . The pharmaceutical composition of  claim 18 , further comprising an anticancer agent. 
     
     
         25 . The pharmaceutical composition of  claim 24 , wherein the anticancer agent is cisplatin. 
     
     
         26 . The pharmaceutical composition of  claim 18  being a therapeutically effective amount for inhibiting histone acetyltransferases (HATs) in a HAT malfunction related pathology. 
     
     
         27 . The pharmaceutical composition of  claim 18  being a therapeutically effective amount for treating colon cancer, breast cancer, or lung cancer in a subject.

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