US2020071328A1PendingUtilityA1

1,6- diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections

Assignee: WOCKHARDT LTDPriority: Aug 25, 2012Filed: Nov 7, 2019Published: Mar 5, 2020
Est. expiryAug 25, 2032(~6.1 yrs left)· nominal 20-yr term from priority
A61K 31/4545C07C 211/63A61K 31/55A61K 31/439A61K 9/0053C07D 487/08C07D 471/08A61K 31/496A61K 9/20A61K 31/546A61K 45/06A61P 31/04A61K 9/48A61K 31/407
72
PatentIndex Score
0
Cited by
0
References
0
Claims

Abstract

Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.

Claims

exact text as granted — not AI-modified
1 . A pharmaceutical composition, comprising: (a) at least one antibacterial agent independently selected from cefpodoxime, ceftibuten, cefuroxime, cefixime and pharmaceutically acceptable salts thereof; and (b) at least one compound independently selected from: 
       
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
       
       and
 stereoisomers and pharmaceutically acceptable salts thereof. 
 
     
     
         2 . The pharmaceutical composition of  claim 1 , further comprising at least one pharmaceutically acceptable excipient. 
     
     
         3 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefpodoxime or a pharmaceutically acceptable salt thereof. 
     
     
         4 . The pharmaceutical composition of  claim 3 , wherein the cefpodoxime is cefpodoxime axetil. 
     
     
         5 . The pharmaceutical composition of  claim 3 , wherein the cefpodoxime is cefpodoxime proxetil. 
     
     
         6 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is ceftibuten or a pharmaceutically acceptable salt thereof. 
     
     
         7 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefuroxime or a pharmaceutically acceptable salt thereof. 
     
     
         8 . The pharmaceutical composition of  claim 7 , where the cefuroxime is cefuroxime axetil. 
     
     
         9 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefiximeor a pharmaceutically acceptable salt thereof. 
     
     
         10 . The pharmaceutical composition of  claim 1 , wherein the at least one compound is in the form of a sodium salt. 
     
     
         11 . The pharmaceutical composition of  claim 1 , wherein the at least one compound is 
       
         
           
           
               
               
           
         
         or a stereoisomer or pharmaceutically acceptable salt thereof. 
       
     
     
         12 . The pharmaceutical composition of  claim 1 , wherein the at least one compound is 
       
         
           
           
               
               
           
         
         or a stereoisomer or pharmaceutically acceptable salt thereof. 
       
     
     
         13 . The pharmaceutical composition of  claim 1 , wherein the at least one compound is 
       
         
           
           
               
               
           
         
         or a stereoisomer or pharmaceutically acceptable salt thereof. 
       
     
     
         14 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefpodoxime, and the at least one compound is 
       
         
           
           
               
               
           
         
       
     
     
         15 . The pharmaceutical composition of  claim 14 , wherein the cefpodoxime is cefpodoxime axetil. 
     
     
         16 . The pharmaceutical composition of  claim 14 , wherein the cefpodoxime is cefpodoxime proxetil. 
     
     
         17 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is ceftibuten, and the at least one compound is 
       
         
           
           
               
               
           
         
       
     
     
         18 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefuroxime, and the at least one compound is 
       
         
           
           
               
               
           
         
       
     
     
         19 . The pharmaceutical composition of  claim 18 , wherein the cefuroxime is cefuroxime axetil. 
     
     
         20 . The pharmaceutical composition of  claim 1 , wherein the at least one antibacterial agent is cefixime, and the at least one compound is

Join the waitlist — get patent alerts

Track US2020071328A1 — get alerts on status changes and closely related new filings.

We store only your email — no account needed. See our privacy policy.