US2018291049A1PendingUtilityA1

Crystalline Forms of Fosnetupitant

Assignee: HELSINN HEALTHCARE SAPriority: Oct 6, 2015Filed: Jun 8, 2018Published: Oct 11, 2018
Est. expiryOct 6, 2035(~9.2 yrs left)· nominal 20-yr term from priority
A61P 1/08C07F 9/650952C07F 9/091C07B 2200/13A61K 31/675C07F 9/65583C07F 9/650958
49
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Claims

Abstract

The present invention provides crystalline forms of the chloride monohydrochloride salt of fosnetupitant, methods of making the crystalline forms, and pharmaceutical dosage forms that make use of the crystalline forms.

Claims

exact text as granted — not AI-modified
1 - 38 ) (canceled) 
     
     
         39 ) Amorphous (4-(5-(2-(3,5-bis(trifluoromethyl)phenyl)-N,2-dimethylpropanamido)-4-(o-tolyl)pyridin-2-yl)-1-methylpiperazin-1-ium-1-yl)methyl hydrogen phosphate (fosnetupitant) chloride hydrochloride. 
     
     
         40 ) A pharmaceutical composition comprising the amorphous fosnetupitant chloride hydrochloride of  claim 39  and one or more pharmaceutically acceptable excipients. 
     
     
         41 ) A pharmaceutical composition comprising the amorphous fosnetupitant chloride hydrochloride of  claim 39 , palonosetron hydrochloride, and one or more pharmaceutically acceptable excipients. 
     
     
         42 ) A composition comprising the amorphous fosnetupitant chloride hydrochloride of  claim 39  and Form I fosnetupitant chloride hydrochloride. 
     
     
         43 ) A pharmaceutical composition comprising the amorphous fosnetupitant chloride hydrochloride of  claim 39 , Form I fosnetupitant chloride hydrochloride, and palonosetron hydrochloride.

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