US2012302587A1PendingUtilityA1

Rho-kinase inhibitors

Assignee: NAGARAHNAM DHANAPALANPriority: Jan 23, 2002Filed: Aug 6, 2012Published: Nov 29, 2012
Est. expiryJan 23, 2022(expired)· nominal 20-yr term from priority
A61P 43/00A61P 35/00A61P 9/10A61P 7/02A61P 9/12A61P 9/00A61P 25/28A61P 27/06A61P 25/00A61P 25/06A61P 19/10A61P 11/06A61P 15/00C07D 401/14C07D 401/12A61P 15/10A61P 19/08
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Claims

Abstract

Disclosed are compounds and derivatives thereof, their synthesis, and their use as Rho-kinase inhibitors. These compounds are useful for inhibiting tumor growth, treating erectile dysfunction, and treating other indications mediated by Rho-kinase, e.g., coronary heart disease.

Claims

exact text as granted — not AI-modified
1 . A compound of the formula 
       
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
       
     
     
         2 . A method of treating an indication mediated by Rho-kinase, comprising administering a compound of  claim 1 . 
     
     
         3 . A process according to  claim 1 , wherein the host is a human. 
     
     
         4 . A method of treating hypertension, atherosclerosis, restenosis, cerebral ischemia, cerebral vasospasm, neuronal degeneration, spinal cord injury, cancer of the breast, colon, prostate, ovaries, brain or lung, thrombotic disorders, asthma, glaucoma, osteoporosis or erectile dysfunction, comprising administering to host in need thereof a compound according to  claim 1 . 
     
     
         5 . A process according to  claim 4 , wherein the host is a human.

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