US2003040093A1PendingUtilityA1

Platelet activating factor acetylhydrolase, and gene thereof

Assignee: SUNTORY LTDPriority: Jun 28, 1996Filed: Sep 25, 2001Published: Feb 27, 2003
Est. expiryJun 28, 2016(expired)· nominal 20-yr term from priority
C12N 9/18
55
PatentIndex Score
0
Cited by
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Claims

Abstract

A protein having activities of a human platelet activating factor acetylhydrolase, and represented by an amino acid sequence represented by the following formula (I) or an amino acid sequence having homology therewith; and a DNA encoding the protein: Met Gly Val Asn Gln Ser Val Gly Phe Pro Pro Val Thr Gly Pro His Leu Val Gly Cys Gly Asp Val Met Glu Gly Gln Asn Leu Gln Gly Ser Phe Phe Arg Leu Phe Tyr Pro Cys Gln Lys Ala Glu Glu Thr Met Glu Gln Pro Leu Trp Ile Pro Arg Tyr Glu Tyr Cys Thr Gly Leu Ala Glu Tyr Leu Gln Phe Asn Lys Arg Cys Gly Gly Leu Leu Phe Asn Leu Ala Val Gly Ser Cys Arg Leu Pro Val Ser Trp Asn Gly Pro Phe Lys Thr Lys Asp Ser Gly Tyr Pro Leu Ile Ile Phe Ser His Gly Leu Gly Ala Phe Arg Thr Leu Tyr Ser Ala Phe Cys Met Glu Leu Ala Ser Arg Gly Phe Val Val Ala Val Pro Glu His Arg Asp Arg Ser Ala Ala Thr Thr Tyr Phe Cys Lys Gln Ala Pro Glu Glu Asn Gln Pro Thr Asn Glu Ser Leu Gln Glu Glu Trp Ile Pro Phe Arg Arg Val Glu Glu Gly Glu Lys Glu Phe His Val Arg Asn Pro Gln Val His Gln Arg Val Ser Glu Cys Leu Arg Val Leu Lys Ile Leu Gln Glu Val Thr Ala Gly Gln Thr Val Phe Asn Ile Leu Pro Gly Gly Leu Asp Leu Met Thr Leu Lys Gly Asn Ile Asp Met Ser Arg Val Ala Val Met Gly His Ser Phe Gly Gly Ala Thr Ala Ile Leu Ala Leu Ala Lys Glu Thr Gln Phe Arg Cys Ala Val Ala Leu Asp Ala Trp Met Phe Pro Leu Glu Arg Asp Phe Tyr Pro Lys Ala Arg Gly Pro Val Phe Phe Ile Asn Thr Glu Lys Phe Gln Thr Met Glu Ser Val Asn Leu Met Lys Lys Ile Cys Ala Gln His Glu Gln Ser Arg Ile Ile Thr Val Leu Gly Ser Val His Arg Ser Gln Thr Asp Phe Ala Phe Val Thr Gly Asn Leu Ile Gly Lys Phe Phe Ser Thr Glu Thr Arg Gly Ser Leu Asp Pro Tyr Glu Gly Gln Glu Val Met Val Arg Ala Met Leu Ala Phe Leu Gln Lys His Leu Asp Leu Lys Glu Asp Tyr Asn Gln Trp Asn Asn Leu Ile Glu Gly Ile Gly Pro Ser Leu Thr Pro Gly Ala Pro His His Leu Ser Ser Leu

Claims

exact text as granted — not AI-modified
1 . A protein having activities of a human platelet activating factor acetylhydrolase, and represented by an amino acid sequence represented by the following formula (I) or an amino acid sequence having homology therewith:  
       
         
           
                 
               
                     
                 
                   Met Gly Val Asn Gln Ser Val Gly Phe Pro Pro Val 
                 
                     
                 
                   Thr Gly Pro His Leu Val Gly Cys Gly Asp Val Met 
                 
                     
                 
                   Glu Gly Gln Asn Leu Gln Gly Ser Phe Phe Arg Leu 
                 
                     
                 
                   Phe Tyr Pro Cys Gln Lys Ala Glu Glu Thr Met Glu 
                 
                     
                 
                   Gln Pro Leu Trp Ile Pro Arg Tyr Glu Tyr Cys Thr 
                 
                     
                 
                   Gly Leu Ala Glu Tyr Leu Gln Phe Asn Lys Arg Cys 
                 
                     
                 
                   Gly Gly Leu Leu Phe Asn Leu Ala Val Gly Ser Cys 
                 
                     
                 
                   Arg Leu Pro Val Ser Trp Asn Gly Pro Phe Lys Thr 
                 
                     
                 
                   Lys Asp Ser Gly Tyr Pro Leu Ile Ile Phe Ser His 
                 
                     
                 
                   Gly Leu Gly Ala Phe Arg Thr Leu Tyr Ser Ala Phe 
                 
                     
                 
                   Cys Met Glu Leu Ala Ser Arg Gly Phe Val Val Ala 
                 
                     
                 
                   Val Pro Glu His Arg Asp Arg Ser Ala Ala Thr Thr 
                 
                     
                 
                   Tyr Phe Cys Lys Gln Ala Pro Glu Glu Asn Gln Pro 
                 
                     
                 
                   Thr Asn Glu Ser Leu Gln Glu Glu Trp Ile Pro Phe 
                 
                     
                 
                   Arg Arg Val Glu Glu Gly Glu Lys Glu Phe His Val 
                 
                     
                 
                   Arg Asn Pro Gln Val His Gln Arg Val Ser Glu Cys 
                 
                     
                 
                   Leu Arg Val Leu Lys Ile Leu Gln Glu Val Thr Ala 
                 
                     
                 
                   Gly Gln Thr Val Phe Asn Ile Leu Pro Gly Gly Leu 
                 
                     
                 
                   Asp Leu Met Thr Leu Lys Gly Asn Ile Asp Met Ser 
                 
                     
                 
                   Arg Val Ala Val Met Gly His Ser Phe Gly Gly Ala 
                 
                     
                 
                   Thr Ala Ile Leu Ala Leu Ala Lys Glu Thr Gln Phe 
                 
                     
                 
                   Arg Cys Ala Val Ala Leu Asp Ala Trp Met Phe Pro 
                 
                     
                 
                   Leu Glu Arg Asp Phe Tyr Pro Lys Ala Arg Gly Pro 
                 
                     
                 
                   Val Phe Phe Ile Asn Thr Glu Lys Phe Gln Thr Met 
                 
                     
                 
                   Glu Ser Val Asn Leu Met Lys Lys Ile Cys Ala Gln 
                 
                     
                 
                   His Glu Gln Ser Arg Ile Ile Thr Val Leu Gly Ser 
                 
                     
                 
                   Val His Arg Ser Gln Thr Asp Phe Ala Phe Val Thr 
                 
                     
                 
                   Gly Asn Leu Ile Gly Lys Phe Phe Ser Thr Glu Thr 
                 
                     
                 
                   Arg Gly Ser Leu Asp Pro Tyr Glu Gly Gln Glu Val 
                 
                     
                 
                   Met Val Arg Ala Met Leu Ala Phe Leu Gln Lys His 
                 
                     
                 
                   Leu Asp Leu Lys Glu Asp Tyr Asn Gln Trp Asn Asn 
                 
                     
                 
                   Leu Ile Glu Gly Ile Gly Pro Ser Leu Thr Pro Gly 
                 
                     
                 
                   Ala Pro His His Leu Ser Ser Leu 
                 
                     
                 
             
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
               
            
           
         
       
     
     
         2 . A DNA encoding said protein of  claim 1 .  
     
     
         3 . An expression vector having said DNA of  claim 2 .  
     
     
         4 . Recombinant host cells transformed by said expression vector of  claim 3 .  
     
     
         5 . A process for the production of a protein having activities of a human platelet activating factor acetylhydrolase, which comprises culturing said recombinant host cells of  claim 4  and collecting said protein from the resulting cultured matter.  
     
     
         6 . An antibody against said protein of  claim 1 .  
     
     
         7 . A DNA encoding a protein having activities of a bovine platelet activating factor acetylhydrolase, and represented by an amino acid sequence represented by the following formula (III) or an amino acid sequence having homology therewith:  
       
         
           
                 
               
                     
                 
                   Met Gly Val Asn Gln Ser Val Ser Phe Pro Pro Val 
                 
                     
                 
                   Thr Gly Pro His Leu Val Gly Cys Gly Asp Val Met 
                 
                     
                 
                   Glu Gly Gln Ser Leu Gln Gly Ser Phe Phe Arg Leu 
                 
                     
                 
                   Phe Tyr Pro Cys Gln Glu Ala Glu Glu Thr Ser Glu 
                 
                     
                 
                   Gln Pro Leu Trp Ile Pro Arg Tyr Glu Tyr Cys Ala 
                 
                     
                 
                   Gly Leu Ala Glu Tyr Leu Lys Phe Asn Lys Arg Trp 
                 
                     
                 
                   Gly Gly Leu Leu Phe Asn Leu Gly Val Gly Ser Cys 
                 
                     
                 
                   Arg Leu Pro Val Ser Trp Asn Gly Pro Phe Lys Thr 
                 
                     
                 
                   Lys Asp Ser Gly Tyr Pro Leu Ile Ile Phe Ser His 
                 
                     
                 
                   Gly Met Gly Ala Phe Arg Thr Val Tyr Ser Ala Phe 
                 
                     
                 
                   Cys Met Glu Leu Ala Ser Arg Gly Phe Val Val Ala 
                 
                     
                 
                   Val Pro Glu His Arg Asp Gly Ser Ala Ala Ala Thr 
                 
                     
                 
                   Cys Phe Cys Lys Gln Thr Pro Glu Glu Asn Gln Pro 
                 
                     
                 
                   Asp Asn Glu Ala Leu Lys Glu Glu Trp Ile Pro His 
                 
                     
                 
                   Arg Gln Ile Glu Glu Gly Glu Lys Glu Phe Tyr Val 
                 
                     
                 
                   Arg Asn Tyr Gln Val His Gln Arg Val Ser Glu Cys 
                 
                     
                 
                   Val Arg Val Leu Lys Ile Leu Gln Glu Val Thr Ala 
                 
                     
                 
                   Gly Gln Ala Val Leu Asn Ile Leu Pro Gly Gly Leu 
                 
                     
                 
                   Asp Leu Met Thr Leu Lys Gly Gly Ile Asp Val Ser 
                 
                     
                 
                   Arg Val Ala Val Met Gly His Ser Phe Gly Gly Ala 
                 
                     
                 
                   Thr Ala Ile Leu Ala Leu Ala Lys Glu Met Gln Phe 
                 
                     
                 
                   Arg Cys Ala Val Ala Leu Asp Ala Trp Met Phe Pro 
                 
                     
                 
                   Leu Glu His Asp Phe Tyr Pro Thr Ala Arg Gly Pro 
                 
                     
                 
                   Ile Phe Phe Ile Asn Ala Glu Lys Phe Gln Thr Val 
                 
                     
                 
                   Glu Thr Val Asn Leu Met Lys Lys Ile Cys Asp Gln 
                 
                     
                 
                   His His Gln Ser Arg Ile Ile Thr Val Leu Gly Ser 
                 
                     
                 
                   Val His Arg Ser Leu Thr Asp Phe Val Phe Val Ala 
                 
                     
                 
                   Gly Asn Trp Ile Ser Lys Phe Phe Ser Ser His Thr 
                 
                     
                 
                   Arg Gly Ser Leu Asp Pro Tyr Glu Gly Gln Glu Thr 
                 
                     
                 
                   Val Val Arg Ala Met Leu Ala Phe Leu Gln Lys His 
                 
                     
                 
                   Leu Asp Leu Lys Glu Asp Tyr Asp Gln Trp Asn Asn 
                 
                     
                 
                   Phe Ile Glu Gly Ile Gly Pro Ser Leu Thr Pro Gly 
                 
                     
                 
                   Ala Pro His His Leu Ser Ser Leu 
                 
                     
                 
             
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
                
               
            
           
         
       
     
     
         8 . An expression vector having said DNA of  claim 7 .  
     
     
         9 . Recombinant eucaryotic host cells transformed by said expression vector of  claim 8 .  
     
     
         10 . A process for the production of a protein having activities of a bovine platelet activating factor acetylhydrolase, which comprises culturing said recombinant eucaryotic host cells of  claim 9  and collecting said protein from the resulting cultured matter.  
     
     
         11 . An antibody against a protein having activities of a bovine platelet activating factor acetylhydrolase, and represented by an amino acid sequence represented by the following formula (III) or an amino acid sequence having homology therewith:  
       
         
           
                 
               
                     
                 
                   Met Gly Val Asn Gln Ser Val Ser Phe Pro Pro Val 
                 
                     
                 
                   Thr Gly Pro His Leu Val Gly Cys Gly Asp Val Met 
                 
                     
                 
                   Glu Gly Gln Ser Leu Gln Gly Ser Phe Phe Arg Leu 
                 
                     
                 
                   Phe Tyr Pro Cys Gln Glu Ala Glu Glu Thr Ser Glu 
                 
                     
                 
                   Gln Pro Leu Trp Ile Pro Arg Tyr Glu Tyr Cys Ala 
                 
                     
                 
                   Gly Leu Ala Glu Tyr Leu Lys Phe Asn Lys Arg Trp 
                 
                     
                 
                   Gly Gly Leu Leu Phe Asn Leu Gly Val Gly Ser Cys 
                 
                     
                 
                   Arg Leu Pro Val Ser Trp Asn Gly Pro Phe Lys Thr 
                 
                     
                 
                   Lys Asp Ser Gly Tyr Pro Leu Ile Ile Phe Ser His 
                 
                     
                 
                   Gly Met Gly Ala Phe Arg Thr Val Tyr Ser Ala Phe 
                 
                     
                 
                   Cys Met Glu Leu Ala Ser Arg Gly Phe Val Val Ala 
                 
                     
                 
                   Val Pro Glu His Arg Asp Gly Ser Ala Ala Ala Thr 
                 
                     
                 
                   Cys Phe Cys Lys Gln Thr Pro Glu Glu Asn Gln Pro 
                 
                     
                 
                   Asp Asn Glu Ala Leu Lys Glu Glu Trp Ile Pro His 
                 
                     
                 
                   Arg Gln Ile Glu Glu Gly Glu Lys Glu Phe Tyr Val 
                 
                     
                 
                   Arg Asn Tyr Gln Val His Gln Arg Val Ser Glu Cys 
                 
                     
                 
                   Val Arg Val Leu Lys Ile Leu Gln Glu Val Thr Ala 
                 
                     
                 
                   Gly Gln Ala Val Leu Asn Ile Lue Pro Gly Gly Leu 
                 
                     
                 
                   Asp Leu Met Thr Leu Lys Gly Gly Ile Asp Val Ser 
                 
                     
                 
                   Arg Val Ala Val Met Gly His Ser Phe Gly Gly Ala 
                 
                     
                 
                   Thr Ala Ile Leu Ala Leu Ala Lys Glu Met Gln Phe 
                 
                     
                 
                   Arg Cys Ala Val Ala Leu Asp Ala Trp Met Phe Pro 
                 
                     
                 
                   Leu Glu His Asp Phe Tyr Pro Thr Ala Arg Gly Pro 
                 
                     
                 
                   Ile Phe Phe Ile Asn Ala Glu Lys Phe Gln Thr Val 
                 
                     
                 
                   Glu Thr Val Asn Leu Met Lys Lys Ile Cys Asp Gln 
                 
                     
                 
                   His His Gln Ser Arg Ile Ile Thr Val Leu Gly Ser 
                 
                     
                 
                   Val His Arg Ser Leu Thr Asp Phe Val Phe Val Ala 
                 
                     
                 
                   Gly Asn Trp Ile Ser Lys Phe Phe Ser Ser His Thr 
                 
                     
                 
                   Arg Gly Ser Leu Asp Pro Tyr Glu Gly Gln Glu Thr 
                 
                     
                 
                   Val Val Arg Ala Met Leu Ala Phe Leu Gln Lys His 
                 
                     
                 
                   Leu Asp Leu Lys Glu Asp Tyr Asp Gln Trp Asn Asn 
                 
                     
                 
                   Phe Ile Glu Gly Ile Gly Pro Ser Leu Thr Pro Gly 
                 
                     
                 
                   Ala Pro His His Leu Ser Ser Leu

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