Inventor · disambiguated record
Jacques Yves Gauthier
Also filed as: GAUTHIER JACQUES Y · GAUTHIER JACQUES YVES
42 granted patents·6 pending applications·3,467 citations·filing 1986–2014
98Inventor score
Files withMERCK FROSST CANADA INC34MERCK FROSST CANADA LTD4ALTMAN MICHAEL D2AXYS PHARM INC2ANDRESEN BRIAN M1
Top patents by PatentIndex Score
48 records- 0199US5861419ASubstituted pyridines as selective cyclooxygenase-2 inhibitorsMERCK FROSST CANADA INC·Filed 1997·Granted Jan 19, 1999·231 cites·19 claims
- 0299US5550142APhenyl heterocycles as cox-2 inhibitorsMERCK FROSST CANADA INC·Filed 1995·Granted Aug 27, 1996·379 cites·18 claims
- 0399US5536752APhenyl heterocycles as COX-2 inhibitorsMERCK FROSST CANADA INC·Filed 1995·Granted Jul 16, 1996·383 cites·18 claims
- 0499US5474995APhenyl heterocycles as cox-2 inhibitorsMERCK FROSST CANADA INC·Filed 1994·Granted Dec 12, 1995·543 cites·25 claims
- 0598US6020343A(Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitorsMERCK FROSST CANADA INC·Filed 1998·Granted Feb 1, 2000·156 cites·42 claims
- 0698US6001843ASubstituted pyridines as selective cyclooxygenase-2 inhibitorsMERCK FROSST CANADA INC·Filed 1998·Granted Dec 14, 1999·104 cites·10 claims
- 0798US5639780AN-benzyl indol-3-yl butanoic acid derivatives as cyclooxygenase inhibitorsMERCK FROSST CANADA INC·Filed 1995·Granted Jun 17, 1997·293 cites·13 claims
- 0898US5604253AN-benzylindol-3-yl propanoic acid derivatives as cyclooxygenase inhibitorsMERCK FROSST CANADA INC·Filed 1995·Granted Feb 18, 1997·319 cites·16 claims
- 0998US5552422AAryl substituted 5,5 fused aromatic nitrogen compounds as anti-inflammatory agentsMERCK FROSST CANADA INC·Filed 1995·Granted Sep 3, 1996·361 cites·21 claims
- 1096US5840746AUse of inhibitors of cyclooxygenase in the treatment of neurodegenerative diseasesMERCK FROSST CANADA INC·Filed 1997·Granted Nov 24, 1998·91 cites·9 claims
- 1196US5710140APhenyl heterocycles as COX-2 inhibitorsMERCK FROSST CANADA INC·Filed 1996·Granted Jan 20, 1998·156 cites·17 claims
- 1293US8735417B2Aminopyrimidines as Syk inhibitorsALTMAN MICHAEL D·Filed 2010·Granted May 27, 2014·35 cites·13 claims
- 1393US6498151B2Aryldifluoromethylphosphonic acids with sulfur-containing substituents as PTP-1B inhibitorsMERCK FROSST CANADA INC·Filed 2001·Granted Dec 24, 2002·56 cites·26 claims
- 1492US9353066B2Substituted phenyl-Spleen Tyrosine Kinase (Syk) inhibitorsMERCK SHARP & DOHME·Filed 2013·Granted May 31, 2016·11 cites·19 claims
- 1589US7973037B2Cathepsin cysteine protease inhibitorsAXYS PHARM INC·Filed 2008·Granted Jul 5, 2011·12 cites·10 claims
- 1688US6596736B2Substituted pyridines as selective cyclooxygenase-2 inhibitorsMERCK FROSST CANADA INC·Filed 2001·Granted Jul 22, 2003·13 cites·15 claims
- 1788US6071936ASubstituted pyridines as selective cyclooxygenase-2 inhibitorsMERCK FROSST CANADA INC·Filed 1999·Granted Jun 6, 2000·27 cites·19 claims
- 1888US5981576A(Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitorsMERCK FROSST CANADA INC·Filed 1998·Granted Nov 9, 1999·39 cites·12 claims
- 1986US7375134B2Cathepsin cysteine protease inhibitorsAXYS PHARM INC·Filed 2003·Granted May 20, 2008·21 cites·10 claims
- 2086US6486142B2Phosphonic acid derivatives as inhibitors of protein tyrosine phosphatase 1B (PTP-1B)MERCK FROSST CANADA INC·Filed 2000·Granted Nov 26, 2002·25 cites·29 claims
- 2181US6486141B2Phosphonic acid biaryl derivatives as inhibitors of protein tyrosine phosphatase 1B (PTP-1B)MERCK FROSST CANADA INC·Filed 2000·Granted Nov 26, 2002·16 cites·28 claims
- 2281US6169188B1(Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitorsMERCK FROSST CANADA INC·Filed 1999·Granted Jan 2, 2001·23 cites·3 claims
- 2380US6777433B2Protein tyrosine phosphatase 1B (PTP-1B) inhibitors containing two ortho-substituted aromatic phosphonatesMERCK FROSST CANADA INC·Filed 2002·Granted Aug 17, 2004·12 cites·21 claims
- 2479US8772336B2Cathepsin cysteine protease inhibitorsMERCK FROSST CANADA INC·Filed 2012·Granted Jul 8, 2014·3 cites·14 claims
- 2579US6448429B1Protein tyrosine phosphatase 1B (PTP-1B) inhibitors containing two ortho-substituted aromatic phosphonatesMERCK FROSST CANADA INC·Filed 2000·Granted Sep 10, 2002·13 cites·28 claims
- 2677US6174874B1Phosphonic acids derivatives as inhibitors of protein tyrosine phosphate 1B (PTP-1B)MERCK FROSST CANADA INC·Filed 1999·Granted Jan 16, 2001·21 cites·23 claims
- 2776US6486194B2Use of inhibitors of cyclooxygenase in the treatment of neurodegenerative diseasesMERCK FROSST CANADA INC·Filed 2001·Granted Nov 26, 2002·7 cites·6 claims
- 2875US7407959B2Cathepsin cysteine protease inhibitorsMERCK FROSST CANADA INC·Filed 2005·Granted Aug 5, 2008·2 cites·9 claims
- 2973US5204358AHetaryl styryl quinolines as leukotriene inhibitorsMERCK FROSST CANADA INC·Filed 1992·Granted Apr 20, 1993·14 cites·8 claims
- 3073US5182367A5-lipoxygenase activating proteinMERCK & CO INC·Filed 1990·Granted Jan 26, 1993·35 cites·3 claims
- 3172US8318748B2Cathepsin cysteine protease inhibitorsBAYLY CHRISTOPHER I·Filed 2011·Granted Nov 27, 2012·2 cites·18 claims
- 3272US6004960APyridazinones as inhibitors of cyclooxygenase-2MERCK FROSST CANADA INC·Filed 1998·Granted Dec 21, 1999·16 cites·15 claims
- 3371US5104882ADiarylstrylquinoline diacids and pharmaceutical compositions thereofMERCK FROSST CANADA INC·Filed 1990·Granted Apr 14, 1992·13 cites·9 claims
- 3465US7060715B2Substituted pyridines as selective cyclooxygenase-2 inhibitorsMERCK FROSST CANADA INC·Filed 2004·Granted Jun 13, 2006·1 cites·12 claims
- 3563US5506227APyridine-substituted benzyl alcohols as leukotriene antagonistsMERCK FROSST CANADA INC·Filed 1992·Granted Apr 9, 1996·18 cites·4 claims
- 3662US2014256743A1Cathepsin cysteine protease inhibitorsMERCK FROSST CANADA LTD·Filed 2014·Application pending·0 cites
- 3761US5004743APyridyl styrene dialkanoic acids as anti-leukotriene agentsMERCK FROSST CANADA INC·Filed 1987·Granted Apr 2, 1991·10 cites·10 claims
- 3856US2014243290A1Aminopyrimidines as SYK InhibitorsALTMAN MICHAEL D·Filed 2014·Application pending·0 cites
- 3955US7312353B2Cathespin cysteine protease inhibitorsMERCK FROST CANADA & CO·Filed 2004·Granted Dec 25, 2007·1 cites·11 claims
- 4049US2010298347A1Substituted 2-naphthoic acids as antagonists of gpr105 activityMERCK FROSST CANADA LTD·Filed 2008·Application pending·0 cites
- 4147US4857659AStereoselective synthesis of leukotriene antagonistsMERCK FROSST CANADA INC·Filed 1987·Granted Aug 15, 1989·2 cites·3 claims
- 4246US2009270511A1Prodrugs of inhibitors of cathepsin sMERCK FROSST CANADA LTD·Filed 2007·Application pending·0 cites
- 4345US2009099264A1Fluoroalkylamine Derivatives as Cathepsin InhibtorsMERCK FROSST CANADA LTD·Filed 2006·Application pending·0 cites
- 4445US2010048717A1Cathepsin b inhibitorsMERCK FROSST CANADA LTD MERK &·Filed 2007·Application pending·0 cites
- 4540US9822107B2Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitorsANDRESEN BRIAN M·Filed 2014·Granted Nov 21, 2017·0 cites·15 claims
- 4640US6211210B1Diphenyl-1,2,3-thiadiazol-3-oxides, compositions and methods of useMERCK FROSST CANADA INC·Filed 2000·Granted Apr 3, 2001·0 cites·12 claims
- 4734US4990526ALeukotriene antagonists, compositions and methods of use thereofMERCK FROSST CANADA INC·Filed 1986·Granted Feb 5, 1991·3 cites·9 claims
- 4830US5136034ASynthesis of chiral thioacetals and thioethersMERCK FROSST CANADA INC·Filed 1990·Granted Aug 4, 1992·0 cites·2 claims
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