Assignee
AXYS PHARM INC
US·40 granted patents·25 pending applications·831 citations·filing 1994–2008
Top patents by PatentIndex Score
65 records- 0195US6506733B1Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2000·Granted Jan 14, 2003·40 cites·18 claims
- 0292US6455502B1Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2000·Granted Sep 24, 2002·39 cites·15 claims
- 0391US6287840B1Irreversible cysteine protease inhibitors containing vinyl groups conjugated to electron withdrawing groupsAXYS PHARM INC·Filed 1999·Granted Sep 11, 2001·49 cites·32 claims
- 0489US7973037B2Cathepsin cysteine protease inhibitorsAXYS PHARM INC·Filed 2008·Granted Jul 5, 2011·12 cites·10 claims
- 0588US7012075B2Cathepsin cysteine protease inhibitorsAXYS PHARM INC·Filed 2002·Granted Mar 14, 2006·52 cites·29 claims
- 0688US6492362B1Compounds and compositions as cathepsin S inhibitorsAXYS PHARM INC·Filed 2000·Granted Dec 10, 2002·28 cites·9 claims
- 0788US6476026B1Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2000·Granted Nov 5, 2002·27 cites·13 claims
- 0887US6562854B2Compositions comprising a substituted benzimidazole useful for treating immunomediated inflammatory disordersAXYS PHARM INC·Filed 2001·Granted May 13, 2003·19 cites·16 claims
- 0986US7375134B2Cathepsin cysteine protease inhibitorsAXYS PHARM INC·Filed 2003·Granted May 20, 2008·21 cites·10 claims
- 1086US6867200B1(Hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitorsAXYS PHARM INC·Filed 1999·Granted Mar 15, 2005·93 cites·13 claims
- 1186US6030946AReversible cysteine protease inhibitorsAXYS PHARM INC·Filed 1996·Granted Feb 29, 2000·78 cites·21 claims
- 1283US6576630B1Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2000·Granted Jun 10, 2003·21 cites·16 claims
- 1383US6278039B1C. elegans deletion mutantsAXYS PHARM INC·Filed 1998·Granted Aug 21, 2001·60 cites·1 claims
- 1482US6081766AMachine-learning approach to modeling biological activity for molecular design and to modeling other characteristicsAXYS PHARM INC·Filed 1994·Granted Jun 27, 2000·58 cites·32 claims
- 1581US6593327B2Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2001·Granted Jul 15, 2003·11 cites·13 claims
- 1679US6103879ABivalent molecules that form an activating complex with an erythropoietin receptorAXYS PHARM INC·Filed 1997·Granted Aug 15, 2000·46 cites·3 claims
- 1774US7226921B2Compounds and compositions as cathepsin S inhibitorsAXYS PHARM INC·Filed 2005·Granted Jun 5, 2007·2 cites·20 claims
- 1874US6022969ACompositions and methods for treating mast-cell mediated conditionsAXYS PHARM INC·Filed 1995·Granted Feb 8, 2000·35 cites·31 claims
- 1973US7196099B2Compounds and compositions as cathepsin inhibitorsAXYS PHARM INC·Filed 2004·Granted Mar 27, 2007·6 cites·13 claims
- 2071US6069010AHigh throughput gene inactivation with large scale gene targetingAXYS PHARM INC·Filed 1996·Granted May 30, 2000·34 cites·14 claims
- 2169US6355460B1Metal mediated serine protease inhibitorsAXYS PHARM INC·Filed 1999·Granted Mar 12, 2002·12 cites·9 claims
- 2269US6069234AModified coagulation agentAXYS PHARM INC·Filed 1997·Granted May 30, 2000·26 cites·14 claims
- 2368US6977256B2Compounds and compositions as cathepsin S inhibitorsAXYS PHARM INC·Filed 2002·Granted Dec 20, 2005·4 cites·21 claims
- 2467US7064123B1Compounds and compositions as cathepsin inhibitorsAXYS PHARM INC·Filed 2001·Granted Jun 20, 2006·4 cites·22 claims
- 2562US7030116B2Compounds and compositions as cathepsin inhibitorsAXYS PHARM INC·Filed 2002·Granted Apr 18, 2006·1 cites·9 claims
- 2662US6087485AAsthma related genesAXYS PHARM INC·Filed 1998·Granted Jul 11, 2000·16 cites·7 claims
- 2761US2007015755A1Novel compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2006·Application pending·0 cites
- 2860US2007232654A1Novel Compounds and Compositions as Cathepsin InhibitorsAXYS PHARM INC·Filed 2007·Application pending·0 cites
- 2957US2004147745A1Novel compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2004·Application pending·0 cites
- 3056US2007203138A1Novel Compounds and Compositions as Cathepsin S InhibitorsAXYS PHARM INC·Filed 2007·Application pending·0 cites
- 3156US2006135781A1Process for preparing heteroaryl and unsaturated heterocycloalkylmagnesium reagents and uses thereofAXYS PHARM INC·Filed 2006·Application pending·0 cites
- 3254US2007135386A1Novel Compounds and Compositions as Cathepsin InhibitorsAXYS PHARM INC·Filed 2007·Application pending·0 cites
- 3353US2003119788A1Novel compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2002·Application pending·0 cites
- 3453US2003096796A1Novel compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2002·Application pending·0 cites
- 3550US6544767B1Cathespin O2 proteaseAXYS PHARM INC·Filed 1995·Granted Apr 8, 2003·7 cites·3 claims
- 3650US2007049594A1Novel compounds and compositions as cathepsin inhibitorsAXYS PHARM INC·Filed 2005·Application pending·0 cites
- 3750US2006089357A1Novel compounds and compositions as cathepsin inhibitorsAXYS PHARM INC·Filed 2005·Application pending·0 cites
- 3849US2004014796A1Novel compounds and compositions as cathepsin S inhititorsAXYS PHARM INC·Filed 2002·Application pending·0 cites
- 3948US2006058553A1Novel bicyclic hydroxamates as inhibitors of histone deacetylaseAXYS PHARM INC·Filed 2003·Application pending·0 cites
- 4048US2005176797A12-[5-(5-Carbamimidoyl-1H-heteroaryl)-6-hydroxybiphenyl-3-YL]-succinic acid derivatives as factor viia inhibitorsAXYS PHARM INC·Filed 2004·Application pending·0 cites
- 4148US2007105892A1Amidino compounds as cysteine protease inhibitorsAXYS PHARM INC·Filed 2004·Application pending·0 cites
- 4248US2007276019A1Haloalkyl Containing Compounds as Cysteine Protease InhibitorsAXYS PHARM INC·Filed 2004·Application pending·0 cites
- 4347US6465503B2Selective urokinase inhibitorsAXYS PHARM INC·Filed 2001·Granted Oct 15, 2002·0 cites·10 claims
- 4447US2004091951A1Assay for measuring acetylation or deacetylation activity of an enzymeAXYS PHARM INC·Filed 2003·Application pending·0 cites
- 4547US2003232864A1Novel Compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2003·Application pending·0 cites
- 4646US2003212120A1Compositions comprising a substituted benzimidazole useful for treating immunomediated inflammatory disordersAXYS PHARM INC·Filed 2003·Application pending·0 cites
- 4745US2003114457A12- [5- (5-carbamimidoyl-1H-heteroaryl)-6-hydroxybiphenyl-3-yl]-succinic acid derivatives as factor viia inhibitorsAXYS PHARM INC·Filed 2002·Application pending·0 cites
- 4845US2003092634A1Novel compounds and compositions as protease inhibitorsAXYS PHARM INC·Filed 2002·Application pending·0 cites
- 4944US2005288336A1Cysteine protease inhibitorsAXYS PHARM INC·Filed 2003·Application pending·0 cites
- 5043US6150379ACompounds and compositions as anticoagulantsAXYS PHARM INC·Filed 1998·Granted Nov 21, 2000·2 cites·6 claims
Showing the top 50 of 65 patent records by PatentIndex Score.
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