Inventor · disambiguated record
Rogelio P. Frutos
Also filed as: FRUTOS ROGELIO · FRUTOS ROGELIO P · FRUTOS ROGELIO PEREZ
17 granted patents·6 pending applications·155 citations·filing 2001–2024
94Inventor score
Files withBOEHRINGER INGELHEIM INT11BOEHRINGER INGELHEIM PHARMA6POUZET PASCALE A J2BUSACCA CARL ALAN1DOLLINGER HORST1
Top patents by PatentIndex Score
23 records- 0194US7514557B2Process for preparing acyclic HCV protease inhibitorsBOEHRINGER INGELHEIM INT·Filed 2005·Granted Apr 7, 2009·41 cites·12 claims
- 0288US8017771B2Process for preparing acyclic HCV protease inhibitorsBOEHRINGER INGELHEIM INT·Filed 2009·Granted Sep 13, 2011·11 cites·1 claims
- 0387US7858804B2Process for making cytokine inhibiting compounds containing 4- and 5-imidazolyl rings and the intermediates thereofBOEHRINGER INGELHEIM INT·Filed 2007·Granted Dec 28, 2010·9 cites·1 claims
- 0486US8609670B2Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthmaPOUZET PASCALE A J·Filed 2012·Granted Dec 17, 2013·13 cites·34 claims
- 0586US8101765B2Process for preparing acyclic HCV protease inhibitorsBUSACCA CARL ALAN·Filed 2009·Granted Jan 24, 2012·11 cites·6 claims
- 0685US7148347B2Process for preparing macrocyclic compoundsBOEHRINGER INGELHEIM INT·Filed 2004·Granted Dec 12, 2006·35 cites·22 claims
- 0782US10745411B2Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthmaBOEHRINGER INGELHEIM INT·Filed 2019·Granted Aug 18, 2020·1 cites·2 claims
- 0882US6437148B1Intermediates for (R)-3(4-bromobenzyl)-1-(3,5-dichlorophenyl)-5-iodo-3-methyl-1-H-imidazo[1,2-a]imidazol-2-oneBOEHRINGER INGELHEIM PHARMA·Filed 2002·Granted Aug 20, 2002·12 cites·2 claims
- 0981US9802954B2Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthmaBOEHRINGER INGELHEIM INT·Filed 2013·Granted Oct 31, 2017·2 cites·21 claims
- 1075US6414161B1Synthesis of (R)-3-(4-Bromobenzyl)-1-(3,5-dichlorophenyl)-5-iodo-3-methyl-1-H-imidazo[1,2-a]imidazol-2-oneBOEHRINGER INGELHEIM PHARMA·Filed 2001·Granted Jul 2, 2002·6 cites·21 claims
- 1174US7470795B2Synthesis of 6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-sulfonic acid amidesBOEHRINGER INGELHEIM PHARMA·Filed 2005·Granted Dec 30, 2008·2 cites·4 claims
- 1274US6458986B1Intermediate for (R)-3-(4-Bromobenzyl)-1-(3,5-dichlorophenyl)-5-iodo-3-methyl-1-H-imidazo[1,2-α]imidazol-2-oneBOEHRINGER INGELHEIM PHARMA·Filed 2002·Granted Oct 1, 2002·5 cites·2 claims
- 1371US8653282B2Preparation of dihydrothieno [3,2-D] pyrimidines and intermediates used thereinFRUTOS ROGELIO·Filed 2008·Granted Feb 18, 2014·2 cites·11 claims
- 1467US6441183B1Intermediate for (R)-3-(4-Bromobenzyl)-1-(3,5-dichlorophenyl)-5-iodo-3-methyl-1-H-imidazo[1,2-a]imidazol-2-oneBOEHRINGER INGELHEIM PHARMA·Filed 2002·Granted Aug 27, 2002·2 cites·2 claims
- 1567US6433183B1(R)-3-(4-bromobenzyl)-1-(3,5-dichlorophenyl)-3-methyl-1,6-dihydroimidazo[1,2-a]imidazole-2,5-dioneBOEHRINGER INGELHEIM PHARMA·Filed 2002·Granted Aug 13, 2002·2 cites·3 claims
- 1665US8471010B2Synthesis of dihydrothieno[3,2-d]pyrimidine diolsFRUTOS ROGELIO P·Filed 2009·Granted Jun 25, 2013·1 cites·21 claims
- 1760US2025270230A1Novel synthetic steps for the manufacturing method of the pde4b-inhibitor 1-({(5r)-2-[4-(5-chloropyrimidine-2-yl)piperidine-1-yl]-5-oxido-6,7-dihydrothieno[3,2-d]pyrimidine-4-yl}amino)cyclobutyl]methanolBOEHRINGER INGELHEIM INT·Filed 2024·Application pending·0 cites
- 1859US2024083889A1Scalable process for the preparation of a GlyT-1 InhibitorBOEHRINGER INGELHEIM INT·Filed 2023·Application pending·0 cites
- 1959US2018072754A1Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthmaBOEHRINGER INGELHEIM INT·Filed 2017·Application pending·0 cites
- 2057US2009088571A1Synthesis of 6,7-Dihydro-5H-imidazo[1,2-a]imidazole-3-sulfonic acid amidesBOEHRINGER INGELHEIM INT·Filed 2008·Application pending·0 cites
- 2154US9150586B2Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthmaPOUZET PASCALE A J·Filed 2012·Granted Oct 6, 2015·0 cites·3 claims
- 2245US2013059866A1Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthmaDOLLINGER HORST·Filed 2012·Application pending·0 cites
- 2340US2006258888A1Bis-Amination of Aryl HalidesBOEHRINGER INGELHEIM INT·Filed 2006·Application pending·0 cites
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Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →