Inventor · disambiguated record
Leslie Joseph Street
Also filed as: STREET LESLIE J · STREET LESLIE JOSEPH · STREET Leslie
80 granted patents·9 pending applications·1,340 citations·filing 1989–2025
99Inventor score
Files withMERCK SHARP & DOHME66MUELLER RUDOLF6PGI DRUG DISCOVERY LLC4CORTEX PHARMA INC3MERCK & CO INC2
Top patents by PatentIndex Score
89 records- 0194US5298520ATriazole containing indole derivativesMERCK SHARP & DOHME·Filed 1992·Granted Mar 29, 1994·97 cites·6 claims
- 0293US7176203B2Imidazo-triazine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2003·Granted Feb 13, 2007·63 cites·7 claims
- 0393US5317103AIndole-substituted five-membered heteroaromatic compounds as 5-HT1 agonistsMERCK SHARP & DOHME·Filed 1992·Granted May 31, 1994·63 cites·7 claims
- 0492US8013003B2Di-substituted amides for enhancing glutamatergic synaptic responsesCORTEX PHARMA INC·Filed 2008·Granted Sep 6, 2011·21 cites·21 claims
- 0592US5260293APyrazines, pyrimidines and pyridazines useful in the treatment of senile dementiaMERCK SHARP & DOHME·Filed 1991·Granted Nov 9, 1993·51 cites·9 claims
- 0691US6476030B1Pyrazolo-triazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 1999·Granted Nov 5, 2002·70 cites·9 claims
- 0791US5208248AIndazole-substituted five-membered heteroaromatic compoundsMERCK SHARPE & DOHME LTD·Filed 1991·Granted May 4, 1993·49 cites·7 claims
- 0889US5106853AOxadiazole and its salts, their use in treating dementiaMERCK SHARP & DOHME·Filed 1990·Granted Apr 21, 1992·77 cites·5 claims
- 0988US6310203B1Precursor compounds to substituted 1,2,4-triazolo[3,4,-a]phathalazine GABA alpha 5 ligandsMERCK SHARPE & DOHME LTD·Filed 2000·Granted Oct 30, 2001·28 cites·2 claims
- 1087US6696444B2Imidazo-triazine derivatives as ligands for GABA receptorsMERCK SHARPE & DOHME·Filed 2003·Granted Feb 24, 2004·26 cites·9 claims
- 1186US6617326B2Imidazo-triazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2002·Granted Sep 9, 2003·21 cites·13 claims
- 1285US6900215B2Imidazo-pyrimidine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2002·Granted May 31, 2005·16 cites·28 claims
- 1385US6730681B2Triazolo-pyrimidine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2000·Granted May 4, 2004·18 cites·12 claims
- 1485US6500828B1Triazolo-pyridazine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2000·Granted Dec 31, 2002·18 cites·9 claims
- 1584US6914063B2Imidazo-pyrazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2001·Granted Jul 5, 2005·14 cites·11 claims
- 1684US6642229B23-Phenyl-imidazo-pyrimidine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2001·Granted Nov 4, 2003·21 cites·11 claims
- 1784US5451588AImidazole, triazole and tetrazole derivativesMERCK SHARP & DOHME·Filed 1993·Granted Sep 19, 1995·39 cites·6 claims
- 1883US7626056B2Cyclohexanesulfonyl derivatives as GlyT1 inhibitors to treat schizophreniaMERCK SHARP & DOHME·Filed 2006·Granted Dec 1, 2009·5 cites·11 claims
- 1982US8119632B2Bicyclic amide derivatives for enhancing glutamatergic synaptic responsesMUELLER RUDOLF·Filed 2010·Granted Feb 21, 2012·4 cites·6 claims
- 2082US6936608B2Imidazo-triazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2001·Granted Aug 30, 2005·20 cites·17 claims
- 2182US6828322B2Triazolo-pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2003·Granted Dec 7, 2004·14 cites·15 claims
- 2282US6541484B2Pyrazolo-pyridine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2000·Granted Apr 1, 2003·19 cites·9 claims
- 2381US7825135B2Heteroaryl piperidine glycine transporter inhibitorsMERCK SHARP & DOHME·Filed 2005·Granted Nov 2, 2010·6 cites·13 claims
- 2481US5510362AImidazole, triazole and tetrazole derivativesMERCK SHARP & DOHME·Filed 1993·Granted Apr 23, 1996·53 cites·8 claims
- 2580US6593325B1Pyrido-pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2000·Granted Jul 15, 2003·15 cites·9 claims
- 2679US6914065B2Imidazo[1,2-C]pyrimidine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2001·Granted Jul 5, 2005·12 cites·8 claims
- 2779US6872720B2Pyrazolo-triazine derivatives as ligands for gaba receptorsMERCK SHARP & DOHME·Filed 2001·Granted Mar 29, 2005·13 cites·8 claims
- 2879US6730676B2Pyrazino-pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2001·Granted May 4, 2004·13 cites·9 claims
- 2979US6608062B1Imidazo-triazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2000·Granted Aug 19, 2003·12 cites·9 claims
- 3079US6255305B1Substituted triazolo-pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 1997·Granted Jul 3, 2001·49 cites·15 claims
- 3179US6200975B1Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligandsMERCK SHARP & DOHME·Filed 1998·Granted Mar 13, 2001·42 cites·24 claims
- 3278US7030128B2Imidazo-pyrimidine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2002·Granted Apr 18, 2006·11 cites·10 claims
- 3376US5854268AAzetidine, pyrrolidine and piperidine derivativesMERCK SHARP & DOHME·Filed 1995·Granted Dec 29, 1998·45 cites·10 claims
- 3475US5602162AImidazole, triazole and tetrazole derivativesMERCK SHARP & DOHME·Filed 1995·Granted Feb 11, 1997·27 cites·8 claims
- 3574US8263591B2Bicyclic amides for enhancing glutamatergic synaptic responsesMUELLER RUDOLF·Filed 2008·Granted Sep 11, 2012·1 cites·14 claims
- 3674US6211219B1Aminocyclohexane derivatives as 5-HT receptor agonistsMERCK SHARP & DOHME·Filed 1997·Granted Apr 3, 2001·18 cites·10 claims
- 3773US6969716B25-phenyl[1,2,4]triazines as ligands for GABA-A α2/α3 receptors for treating anxiety or depressionMERCK SHARP & DOHME·Filed 2004·Granted Nov 29, 2005·6 cites·10 claims
- 3873US6140347AAzetidine, pyrrolidine and piperidine derivatives as 5-HT receptor agonistsMERCK SHARP & DOHME·Filed 1997·Granted Oct 31, 2000·18 cites·9 claims
- 3972US8507482B2Bicyclic amide derivatives for enhancing glutamatergic synaptic responsesMUELLER RUDOLF·Filed 2012·Granted Aug 13, 2013·1 cites·17 claims
- 4071US8168632B2Bicyclic amide derivatives for the treatment of respiratory disordersMUELLER RUDOLF·Filed 2010·Granted May 1, 2012·1 cites·17 claims
- 4171US8110584B2Methods for the treatment of respiratory depressionMUELLER RUDOLF·Filed 2010·Granted Feb 7, 2012·1 cites·15 claims
- 4270US6579875B1Triazolo-pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 1999·Granted Jun 17, 2003·22 cites·20 claims
- 4370US6444666B1Triazolopyridazine Derivatives for treating anxiety and enhancing cognitionMERCK SHARP & DOHME·Filed 1998·Granted Sep 3, 2002·15 cites·8 claims
- 4467US8642633B2Di-substituted amides for enhancing glutamatergic synaptic responsesCORTEX PHARMACEUTICAL INC·Filed 2013·Granted Feb 4, 2014·1 cites·15 claims
- 4564US8404682B2Di-substituted amides for enhancing glutamatergic synaptic responsesSTREET Leslie·Filed 2011·Granted Mar 26, 2013·1 cites·38 claims
- 4664US6337331B1Triazolo-pyrimidine as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 1999·Granted Jan 8, 2002·21 cites·10 claims
- 4764US2025129035A1Compounds for the treatment of a central nervous system disease or disorderPGI DRUG DISCOVERY LLC·Filed 2024·Application pending·0 cites
- 4863US7851638B2Cyclohexanesulfonyl derivatives as GLYT1 inhibitors to treat schizophreniaMERCK SHARP & DOHME·Filed 2009·Granted Dec 14, 2010·0 cites·9 claims
- 4963US7485640B2Imidazopyrazinones as GABA-A receptor anxiolyticsMERCK SHARP & DOHME·Filed 2003·Granted Feb 3, 2009·1 cites·8 claims
- 5062US6960598B2(1,8) naphthyridines as gaba ligands, their pharmaceutical compositions and usesMERCK SHARP & DOHME·Filed 2002·Granted Nov 1, 2005·2 cites·11 claims
Showing the top 50 of 89 patent records by PatentIndex Score.
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