Inventor · disambiguated record
Brian John Williams
Also filed as: WILLIAMS BRIAN · WILLIAMS BRIAN J · WILLIAMS BRIAN JOHN
52 granted patents·6 pending applications·1,113 citations·filing 1988–2014
99Inventor score
Files withMERCK SHARP & DOHME38MERCK & CO INC6ASTEX THERAPEUTICS LTD3BERDINI VALERIO1CARLING WILLIAM ROBERT1
Top patents by PatentIndex Score
58 records- 0199US5719147AMorpholine and thiomorpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 1995·Granted Feb 17, 1998·193 cites·27 claims
- 0294US6172077B1Spiro-azacyclic derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 1998·Granted Jan 9, 2001·149 cites·15 claims
- 0394US5637699AProcess for preparing morpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 1995·Granted Jun 10, 1997·85 cites·2 claims
- 0493US5494926A2/3-(heterocyclic alkyl amino)-1-(subst.-phenyl-methoxy)-ethanes/propanes as tachykinin-receptor antagonistsMERCK SHARP & DOHME·Filed 1994·Granted Feb 27, 1996·67 cites·15 claims
- 0587US5459270AAzacyclic compounds, processes for their preparation and pharmaceutical compositions containing themMERCK SHARP & DOHME·Filed 1992·Granted Oct 17, 1995·69 cites·14 claims
- 0686US8383619B2Pharmaceutical compoundsASTEX THERAPEUTICS LTD·Filed 2010·Granted Feb 26, 2013·8 cites·13 claims
- 0786US7138400B2Sulfamides as gamma-secretase inhibitorsMERCK SHARP & DOHME·Filed 2001·Granted Nov 21, 2006·32 cites·6 claims
- 0886US6235735B1Morpholine and thiomorpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 2000·Granted May 22, 2001·19 cites·18 claims
- 0986US5952315AUse of NK-1 receptor antagonists for treating bipolar disordersMERCK SHARP & DOHME·Filed 1997·Granted Sep 14, 1999·34 cites·5 claims
- 1086US5620989A4-Arylmethyloxymethyl piperidines as tachykinin antagonsitsMERCK SHARP & DOHME·Filed 1993·Granted Apr 15, 1997·61 cites·12 claims
- 1185US7304094B2Cyclohexyl sulphonesMERCK SHARP & DOHME·Filed 2005·Granted Dec 4, 2007·7 cites·8 claims
- 1280US6984663B2Cyclohexyl sulphonesMERCK SHARP & DOHME·Filed 2002·Granted Jan 10, 2006·11 cites·11 claims
- 1378US8664218B2Pharmaceutical compoundsASTEX THERAPEUTICS LTD·Filed 2013·Granted Mar 4, 2014·3 cites·12 claims
- 1477US8653084B2Hydrobenzamide derivatives as inhibitors of Hsp90FREDERICKSON MARTYN·Filed 2007·Granted Feb 18, 2014·5 cites·9 claims
- 1577US6489343B2Tetrahydropyran derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 2001·Granted Dec 3, 2002·9 cites·10 claims
- 1677US6060469ASpiro-piperidine derivatives and their use as tachykinin antagonistsMERCK SHARP & DOHME·Filed 1996·Granted May 9, 2000·42 cites·22 claims
- 1777US5166350AProcess for the manufacture of fluoran compoundsCIBA GEIGY CORP·Filed 1991·Granted Nov 24, 1992·22 cites·21 claims
- 1876US7595344B2Sulphones which modulate the action of gamma secretaseMERCK SHARP & DOHME·Filed 2008·Granted Sep 29, 2009·2 cites·12 claims
- 1975US9428439B2Hydrobenzamide derivatives as inhibitors of Hsp90ASTEX THERAPEUTICS LTD·Filed 2014·Granted Aug 30, 2016·2 cites·11 claims
- 2074US5872116AMorpholine and thiomorpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 1997·Granted Feb 16, 1999·14 cites·21 claims
- 2173US8796244B2Imidazopyridine derivatives as inhibitors of receptor tyrosine kinasesBERDINI VALERIO·Filed 2009·Granted Aug 5, 2014·2 cites·21 claims
- 2273US6458830B1Tetrahydropyran derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 2000·Granted Oct 1, 2002·7 cites·22 claims
- 2373US5929054AUse of NK-1 receptor antagonists for treating sexual dysfunctionsMERCK SHARP·Filed 1997·Granted Jul 27, 1999·41 cites·3 claims
- 2472US6048859AMorpholine and thiomorpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 1999·Granted Apr 11, 2000·26 cites·23 claims
- 2571US6638930B2Morpholine and thiomorpholine tachykinin receptor antagonistsMERCK & CO INC·Filed 2001·Granted Oct 28, 2003·1 cites·4 claims
- 2669US4863953A[3R]-3-amino-1-hydroxy pyrrolidin-2-one and its use as a neuroprotective agentMERCK SHARP & DOHME·Filed 1988·Granted Sep 5, 1989·13 cites·5 claims
- 2768US5633281A3,3-diphenyl prop-2-yl amino acid derivatives and their use as tachykinin antagonistsMERCK SHARP & DOHME·Filed 1993·Granted May 27, 1997·9 cites·8 claims
- 2867US6964981B2Tetrahydrofuran derivatives and their use as NK-1 antagonistsMERCK SHARP & DOHME·Filed 2001·Granted Nov 15, 2005·3 cites·14 claims
- 2967US5985874ASubstituted morpholine derivative and its use as a therapeutic agentMERCK SHARP & DOHME·Filed 1999·Granted Nov 16, 1999·10 cites·6 claims
- 3067US5977104AUse of NK-1 receptor antagonists for treating bipolar disordersMERCK SHARP & DOHME·Filed 1998·Granted Nov 2, 1999·29 cites·4 claims
- 3165US6114315AUse of NK-1 receptor antagonists for treating major depressive disorders with anxietyMERCK SHARP & DOHME·Filed 1998·Granted Sep 5, 2000·26 cites·4 claims
- 3262US4925867AHydrocarbon substituted pyrrolidinones, intermediates therefor, and anti-convulsant use thereofMERCK SHARP & DOHME·Filed 1989·Granted May 15, 1990·6 cites·8 claims
- 3361US5331089APeptides useful as tachykinin agonistsMERCK SHARPE & DOHME LTD·Filed 1992·Granted Jul 19, 1994·18 cites·9 claims
- 3459US5495047AFused tricyclic compounds, pharmaceutical compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1992·Granted Feb 27, 1996·6 cites·12 claims
- 3559US2008045533A1Novel cyclohexyl sulphonesCHURCHER IAN·Filed 2007·Application pending·0 cites
- 3658US7598386B2Sulphones which modulate the action of gamma-secretaseMERCK SHARP & DOHME·Filed 2007·Granted Oct 6, 2009·0 cites·5 claims
- 3758US7342009B2Cyclic sulfonamides for inhibition of gamma-secretaseMERCK SHARP & DOHME·Filed 2004·Granted Mar 11, 2008·0 cites·13 claims
- 3857US7410964B2Cyclohexyl sulphones as gamma-secretase inhibitorsMERCK SHARP & DOHME·Filed 2004·Granted Aug 12, 2008·0 cites·4 claims
- 3957US2008045515A1Cyclic sulfonamides for inhibition of gamma-secretaseDINNELL KEVIN·Filed 2007·Application pending·0 cites
- 4056US6071927ASpiro-piperidine derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 1997·Granted Jun 6, 2000·13 cites·24 claims
- 4155US5288730AAzabicyclic compounds, pharmaceutical compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1992·Granted Feb 22, 1994·10 cites·11 claims
- 4254US5610183APhenylglycine derivatives pharmaceutical compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1992·Granted Mar 11, 1997·10 cites·11 claims
- 4353US5610159AN-oxides of morpholine derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 1996·Granted Mar 11, 1997·6 cites·19 claims
- 4448US5925627AUse of NK-1 receptor antagonists for treating movement disordersMERCK SHARP & DOHME·Filed 1997·Granted Jul 20, 1999·7 cites·11 claims
- 4548US5633266AAzacyclic compounds compositions containing them and their use as tachykinin antagonistsMERCK SHARP & DOHME·Filed 1994·Granted May 27, 1997·7 cites·17 claims
- 4647US2004116404A1Sulphones which modulate the action of gamma secretaseFiled 2001·Application pending·0 cites
- 4746US5629347AAromatic compounds, pharmaceutical compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1992·Granted May 13, 1997·6 cites·12 claims
- 4845US2009054440A1Quinoline derivatives as neurokinin receptor antagonistsCARLING WILLIAM ROBERT·Filed 2006·Application pending·0 cites
- 4943US7265110B2Tetrahydropyran derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 2002·Granted Sep 4, 2007·0 cites·20 claims
- 5043US6271230B1Use of NK-1 receptor antagonists for treating cognitive disordersMERCK SHARP & DOHME·Filed 1999·Granted Aug 7, 2001·6 cites·5 claims
Showing the top 50 of 58 patent records by PatentIndex Score.
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