Inventor · disambiguated record
John P. Dusza
Also filed as: ALBRIGHT JAY D · DUSZA JOHN · DUSZA JOHN P · DUSZA JOHN PAUL
54 granted patents·2 pending applications·1,343 citations·filing 1978–2008
99Inventor score
Top patents by PatentIndex Score
56 records- 0198US4626538A[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1985·Granted Dec 2, 1986·106 cites·15 claims
- 0298US4521422AAryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanonesAMERICAN CYANAMID CO·Filed 1984·Granted Jun 4, 1985·71 cites·31 claims
- 0398US4178449APyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1978·Granted Dec 11, 1979·62 cites·18 claims
- 0497US6399621B1N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1, 5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related theretoAMERICAN CYANAMID CO·Filed 2000·Granted Jun 4, 2002·78 cites·9 claims
- 0597US4209621A(Substituted-phenyl)-1,2,4-triazolo[4,3-a]-pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1979·Granted Jun 24, 1980·47 cites·16 claims
- 0696US4876252A4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinaminesAMERICAN CYANAMID CO·Filed 1988·Granted Oct 24, 1989·89 cites·1 claims
- 0796US4788195A4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinaminesAMERICAN CYANAMID CO·Filed 1986·Granted Nov 29, 1988·104 cites·16 claims
- 0894US4900836A(3-amino-1H-pyrazol-4-yl) (aryl)methanonesAMERICAN CYANAMID CO·Filed 1984·Granted Feb 13, 1990·38 cites·1 claims
- 0993US4654347AAryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanonesAMERICAN CYANAMID CO·Filed 1985·Granted Mar 31, 1987·43 cites·15 claims
- 1093US4576943APyrazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1984·Granted Mar 18, 1986·30 cites·22 claims
- 1193US4281000ASubstituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agentsAMERICAN CYANAMID CO·Filed 1980·Granted Jul 28, 1981·30 cites·18 claims
- 1293US4260756A6- And 8-heteroaryl-1,2,4-triazolo[4,3-b]pyridazinesAMERICAN CYANAMID CO·Filed 1979·Granted Apr 7, 1981·26 cites·14 claims
- 1392US4421753A1-(5-Amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazinesAMERICAN CYANAMID CO·Filed 1982·Granted Dec 20, 1983·26 cites·30 claims
- 1492US4236005AImidazo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1979·Granted Nov 25, 1980·23 cites·10 claims
- 1591US5536718ATricyclic benzazepine vasopressin antagonistsAMERICAN CYANAMID CO·Filed 1995·Granted Jul 16, 1996·86 cites·37 claims
- 1691US4654343AN-substituted-N[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureasAMERICAN CYANAMID CO·Filed 1985·Granted Mar 31, 1987·60 cites·15 claims
- 1789US6903091B2Biphenyl vasopressin agonistsWYETH CORP·Filed 2002·Granted Jun 7, 2005·26 cites·6 claims
- 1888US4582833A2-(substituted-1-piperazinyl)[1,2,4]triazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1984·Granted Apr 15, 1986·19 cites·19 claims
- 1987US6511974B1Tricyclic vasopressin agonistsWYETH CORP·Filed 1998·Granted Jan 28, 2003·42 cites·88 claims
- 2086US7053083B2Cyclohexylphenyl vasopressin agonistsWYETH CORP·Filed 2002·Granted May 30, 2006·23 cites·9 claims
- 2186US5169850AN-(dialkylamino)methylene)-substituted pyrazolo(1,5-a)-pyrimidine-3-carboxamides and N-(dialkylamino)methylene-substituted-4,5-dihydropyrazolo-(1,5-a)-pyrimidine-3-carboxamidesAMERICAN CYANAMID CO·Filed 1991·Granted Dec 8, 1992·30 cites·10 claims
- 2285US5753648ATricyclic benzazepine vasopressin antagonistsAMERICAN CYANAMID CO·Filed 1996·Granted May 19, 1998·70 cites·36 claims
- 2384US4847256A4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidinesAMERICAN CYANAMID CO·Filed 1986·Granted Jul 11, 1989·34 cites·15 claims
- 2483US4444774A7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1982·Granted Apr 24, 1984·13 cites·7 claims
- 2581US7465722B2Biphenyl vasopressin agonistsWYETH CORP·Filed 2006·Granted Dec 16, 2008·3 cites·12 claims
- 2681US7202239B2Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonistsWYETH CORP·Filed 2002·Granted Apr 10, 2007·16 cites·21 claims
- 2779US4260767A2-PyridylhydrazidesAMERICAN CYANAMID CO·Filed 1979·Granted Apr 7, 1981·8 cites·7 claims
- 2878US4347251ANovel 3-substituted amino-1-substituted heteroaryl-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1981·Granted Aug 31, 1982·12 cites·8 claims
- 2976US5538977A3-Substituted-7-[3-(imidazol-1-yl)phenyl]-pyrazolo[1,5-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1995·Granted Jul 23, 1996·19 cites·33 claims
- 3074US4451479ATherapeutically active 3-amino-1-halogenated phenyl-2-pyrazolines and their C4 and C5 analogsAMERICAN CYANAMID CO·Filed 1982·Granted May 29, 1984·8 cites·58 claims
- 3173US4432991ATherapeutically active 3-amino-1-phenyl(and substituted phenyl)-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1982·Granted Feb 21, 1984·10 cites·6 claims
- 3270US4980472AMethod of making (3-amino-1H-pyrazol-4-yl) (aryl)methanonesAMERICAN CYANAMID CO·Filed 1989·Granted Dec 25, 1990·8 cites·7 claims
- 3369US4374988A4-Heteroarylimidazo-[1,5-A]pyrimidinesAMERICAN CYANAMID CO·Filed 1981·Granted Feb 22, 1983·6 cites·16 claims
- 3467US4551530APyridyl imidazo[1,2-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1984·Granted Nov 5, 1985·5 cites·2 claims
- 3566US5700796ATricyclic benzazepine vasopressin antagonistsAMERICAN CYANAMID CO·Filed 1996·Granted Dec 23, 1997·20 cites·18 claims
- 3666US2009227565A1Biphenyl Vasopressin AgonistsWYETH CORP·Filed 2008·Application pending·0 cites
- 3764US5059691AN-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamidesAMERICAN CYANAMID CO·Filed 1990·Granted Oct 22, 1991·8 cites·9 claims
- 3862US4376122ANovel 3-substituted amino-1-heteroaryl-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1981·Granted Mar 8, 1983·4 cites·4 claims
- 3961US7223752B2Biphenyl vasopressin agonistsWYETH CORP·Filed 2004·Granted May 29, 2007·0 cites·27 claims
- 4060US5612334ATricyclic benzazepine vasopressin antagonistsAMERICAN CYANAMID CO·Filed 1995·Granted Mar 18, 1997·12 cites·9 claims
- 4157US4393217ASubstituted phenyl-5-aminopyrazolesAMERICAN CYANAMID CO·Filed 1981·Granted Jul 12, 1983·3 cites·3 claims
- 4256US4767765AN-substituted-N-[3-(1,2,4-triazolo-[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureasAMERICAN CYANAMID CO·Filed 1987·Granted Aug 30, 1988·4 cites·12 claims
- 4355US4447442A3-Trifluoroacetylamino-1-aryl-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1982·Granted May 8, 1984·4 cites·52 claims
- 4454US7329653B2Cyclohexylphenyl vasopressin agonistsWYETH CORP·Filed 2006·Granted Feb 12, 2008·0 cites·8 claims
- 4554US4267191AProcess for enhancing growth promotion in animalsAMERICAN CYANAMID CO·Filed 1980·Granted May 12, 1981·3 cites·10 claims
- 4651US4448973ATherapeutically active 3-substituted amino-1-phenyl and substituted phenyl-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1982·Granted May 15, 1984·3 cites·4 claims
- 4748US5037980APhenyl imidazo[1,2-a]pyrimidinesAMERICAN CYANAMID CO·Filed 1988·Granted Aug 6, 1991·2 cites·10 claims
- 4848US4888345A4,8-disubstituted-1,2-dihydro and 1,2,3,4-tetrahydroimidazo-[1,5-a] pyrimidinesAMERICAN CYANAMID CO·Filed 1988·Granted Dec 19, 1989·2 cites·16 claims
- 4945US2002198221A1N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-alpha]-pyrimidin-7-yl}phenyl)acetamide and compositions and, methods related theretoAMERICAN CYANAMID CO·Filed 2001·Application pending·0 cites
- 5042US4348527A3-Trifluoroacetyl amino-1-aryl-2-pyrazolinesAMERICAN CYANAMID CO·Filed 1981·Granted Sep 7, 1982·1 cites·15 claims
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