Inventor · disambiguated record
Angus Murray Macleod
Also filed as: MACLEOD ANGUS · MACLEOD ANGUS M · MACLEOD ANGUS MURRAY
81 granted patents·21 pending applications·1,485 citations·filing 1987–2024
99Inventor score
Files withMERCK SHARP & DOHME52INFLAZOME LTD28MERCK SHARPE & DOHME LTD5ANDREWS MARTIN JAMES INGLIS3SHIRE LLC3
Top patents by PatentIndex Score
102 records- 0198US5514718AHeterocyclic compounds, processes for their preparation and pharmaceutical compositions containing themMERCK SHARP & DOHME·Filed 1994·Granted May 7, 1996·551 cites·12 claims
- 0296US5885999ASerine derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 1997·Granted Mar 23, 1999·103 cites·19 claims
- 0393US6136824A1-piperidinyl-propan-2-derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 2000·Granted Oct 24, 2000·61 cites·28 claims
- 0491US11981667B2Sulfonamide carboxamide compoundsINFLAZOME LTD·Filed 2022·Granted May 14, 2024·1 cites·8 claims
- 0590US11370776B2Sulfonylureas and sulfonylthioureas as NLRP3 inhibitorsINFLAZOME LTD·Filed 2018·Granted Jun 28, 2022·6 cites·19 claims
- 0689US7915256B2Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseasesGALAPAGOS NV·Filed 2009·Granted Mar 29, 2011·12 cites·50 claims
- 0789US7501411B2Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseasesGALAPAGOS NV·Filed 2007·Granted Mar 10, 2009·12 cites·54 claims
- 0888US6310203B1Precursor compounds to substituted 1,2,4-triazolo[3,4,-a]phathalazine GABA alpha 5 ligandsMERCK SHARPE & DOHME LTD·Filed 2000·Granted Oct 30, 2001·28 cites·2 claims
- 0988US5334606AOxazolidindione substituted indole derivativesMERCK SHARPE & DOHME LTD·Filed 1992·Granted Aug 2, 1994·68 cites·5 claims
- 1086US7381725B2Pyridazine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2003·Granted Jun 3, 2008·17 cites·4 claims
- 1186US5620989A4-Arylmethyloxymethyl piperidines as tachykinin antagonsitsMERCK SHARP & DOHME·Filed 1993·Granted Apr 15, 1997·61 cites·12 claims
- 1283US11465992B2Sulfonamide carboxamide compoundsINFLAZOME LTD·Filed 2018·Granted Oct 11, 2022·1 cites·37 claims
- 1383US10973803B2Sodium salt of N-((1,2,3,5,6,7-hexahydro-s-indacen-4-yl)carbamoyl)-1-isopropyl-1H-pyrazole-3-sulfonamideINFLAZOME LTD·Filed 2020·Granted Apr 13, 2021·1 cites·32 claims
- 1483US5472978AAromatic compounds, pharmaceutical compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1992·Granted Dec 5, 1995·26 cites·9 claims
- 1583US5242927AProdrugs for oxadiazole muscarinic agonistsMERCK SHARP & DOHME·Filed 1988·Granted Sep 7, 1993·33 cites·7 claims
- 1682US5760018AGem-disubstituted azacyclic tachykinin antagonistsMERCK SHARP & DOHME·Filed 1995·Granted Jun 2, 1998·59 cites·11 claims
- 1782US5405853AThiadiazoles useful in the treatment of senile dementiaMERCK SHARPE & DOHME LTD·Filed 1993·Granted Apr 11, 1995·23 cites·8 claims
- 1881US11613542B2Sulfonylureas and sulfonylthioureas as NLRP3 inhibitorsINFLAZOME LTD·Filed 2018·Granted Mar 28, 2023·2 cites·32 claims
- 1981US5612337ASubstituted morpholine derivatives and their use as therapeutic agentsMERCK SHARP & DOHME·Filed 1994·Granted Mar 18, 1997·46 cites·24 claims
- 2080US11542255B2Sulfonylureas and sulfonylthioureas as NLRP3 inhibitorsINFLAZOME LTD·Filed 2018·Granted Jan 3, 2023·2 cites·24 claims
- 2180US11518739B2Sulfonamide carboxamide compoundsINFLAZOME LTD·Filed 2018·Granted Dec 6, 2022·2 cites·22 claims
- 2279US11858922B2Sulfonylureas and related compounds and use of sameUNIV QUEENSLAND·Filed 2017·Granted Jan 2, 2024·2 cites·36 claims
- 2379US6559166B1Phenylsulphonyl derivatives as 5-HT receptor ligandsMERCK SHARP & DOHME·Filed 2000·Granted May 6, 2003·14 cites·7 claims
- 2479US6200975B1Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligandsMERCK SHARP & DOHME·Filed 1998·Granted Mar 13, 2001·42 cites·24 claims
- 2579US2025115591A1Novel sulfonamide carboxamide compoundsINFLAZOME LTD·Filed 2024·Application pending·0 cites
- 2678US7030128B2Imidazo-pyrimidine derivatives as ligands for GABA receptorsMERCK SHARP & DOHME·Filed 2002·Granted Apr 18, 2006·11 cites·10 claims
- 2777US7893058B2Imidazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseasesJANSSEN PHARMACEUTICA NV·Filed 2007·Granted Feb 22, 2011·2 cites·55 claims
- 2876US11926600B2Sulfonylureas and sulfonylthioureas as NLRP3 inhibitorsINFLAZOME LTD·Filed 2018·Granted Mar 12, 2024·1 cites·12 claims
- 2976US6900209B2Nitrogen substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives for enhancing cognitionMERCK SHARP & DOHME·Filed 2001·Granted May 31, 2005·8 cites·10 claims
- 3076US5973156APiperidine and tetrahydropyridine derivativesMERCK SHARP & DOME LTD·Filed 1996·Granted Oct 26, 1999·25 cites·12 claims
- 3175US5977116APiperazine, piperidine and tetrahydropyridine derivativesMERCK SHARP & DOHME·Filed 1996·Granted Nov 2, 1999·19 cites·10 claims
- 3275US2025019355A1CompoundsINFLAZOME LTD·Filed 2024·Application pending·0 cites
- 3374US8362018B2Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infectionsBIOFOCUS DPI LTD·Filed 2008·Granted Jan 29, 2013·5 cites·17 claims
- 3474US6211219B1Aminocyclohexane derivatives as 5-HT receptor agonistsMERCK SHARP & DOHME·Filed 1997·Granted Apr 3, 2001·18 cites·10 claims
- 3572US7468393B2Diarylsulfones as 5-HT2A antagonistsMERCK SHARP & DOHME·Filed 2007·Granted Dec 23, 2008·1 cites·17 claims
- 3671US5519163AInhibitors of phosphoinositide-specific phospholipase CMERCK & CO INC·Filed 1993·Granted May 21, 1996·25 cites·6 claims
- 3768US6355638B1Pyrazolo[1,5-d][1,2,4] triazines for enhancing cognitionMERCK SHARP & DOHME·Filed 2000·Granted Mar 12, 2002·4 cites·9 claims
- 3866US7482457B2Substituted quinoline-4-carboxylic hydrazides as NK-2/NK-3 receptor ligandsMERCK SHARP & DOHME·Filed 2004·Granted Jan 27, 2009·2 cites·12 claims
- 3966US7144887B2Substituted 1,2,3-triazolo[1,5-a]quinazolines for enhancing cognitionMERCK SHARP & DOHME·Filed 2000·Granted Dec 5, 2006·3 cites·7 claims
- 4065US7094777B25-HT2A receptor ligandsMERK SHARP & DOHME LTD·Filed 2004·Granted Aug 22, 2006·5 cites·24 claims
- 4165US5612336AHeterocyclic amide derivatives as tachykinin antagonistsMERCK SHARP & DOHME·Filed 1993·Granted Mar 18, 1997·9 cites·13 claims
- 4265US5328927AHetercyclic compounds, processes for their preparation and pharmaceutical compositions containing themMERCK SHARPE & DOHME LTD·Filed 1993·Granted Jul 12, 1994·16 cites·13 claims
- 4364US6777430B2Phenylsulphonyl derivatives as 5-HT receptor ligandsMERCK SHARP & DOHME·Filed 2003·Granted Aug 17, 2004·2 cites·9 claims
- 4464US5554627ATachykinin antagonistsMERCK SHARP & DOHME·Filed 1993·Granted Sep 10, 1996·8 cites·11 claims
- 4564US2021332020A1Phenylsulfonylurea derivatives useful as nlrp3 inhibitorsINFLAZOME LTD·Filed 2019·Application pending·0 cites
- 4663US5661162A4-aminomethyl/thiomethyl/sulfonylmethyl-4-phenylpiperdines as tachykinin receptor antagonistsMERCK SHARP & DOHME·Filed 1993·Granted Aug 26, 1997·17 cites·13 claims
- 4762US6949549B2Imidazolophthalazine derivatives as ligands for GABAA receptorsMERCK SHARP & DOHME·Filed 2001·Granted Sep 27, 2005·2 cites·6 claims
- 4862US5580877APyrazolo-quinoline derivatives for treating cerebral ischemiaMERCK SHARP & DOHME·Filed 1995·Granted Dec 3, 1996·8 cites·11 claims
- 4960US5998440AAzetidine, pyrrolidine and piperidine derivativesMERCK SHARPE & DOHME LTD·Filed 1996·Granted Dec 7, 1999·8 cites·11 claims
- 5060US5849746ASubstituted 1,4-piperazine-heteroaryl derivatives as 5-HT1D receptor agonistsMERCK SHARP & DOHME·Filed 1996·Granted Dec 15, 1998·16 cites·7 claims
Showing the top 50 of 102 patent records by PatentIndex Score.
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