Inventor · disambiguated record
Bruce E. Tomczuk
Also filed as: TOMCZUK BRUCE · TOMCZUK BRUCE E · TOMCZUK BRUCE EDWARD
51 granted patents·8 pending applications·663 citations·filing 1986–2019
99Inventor score
Files withDIMENSIONAL PHARM INC33ROBINS CO INC A H7ASTRAZENECA AB4ORTHO MCNEIL PHARM INC43-DIMENSIONAL PHARM INC1
Top patents by PatentIndex Score
59 records- 0196US6037356AHeteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 1998·Granted Mar 14, 2000·67 cites·37 claims
- 0289US8894970B2Arginase inhibitors and methods of use thereofTOMCZUK BRUCE EDWARD·Filed 2011·Granted Nov 25, 2014·25 cites·2 claims
- 0388US6706021B2Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2003·Granted Mar 16, 2004·18 cites·42 claims
- 0488US6566379B1Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2002·Granted May 20, 2003·13 cites·42 claims
- 0588US6245763B1Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted Jun 12, 2001·13 cites·35 claims
- 0686US7402586B2Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsORTHO MCNEIL PHARM INC·Filed 2005·Granted Jul 22, 2008·4 cites·64 claims
- 0786US6350764B2Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Feb 26, 2002·15 cites·37 claims
- 0885US6326492B1Heterocyclic protease inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted Dec 4, 2001·25 cites·41 claims
- 0984US8859602B2Inhibitors of c-fms kinaseILLIG CARL R·Filed 2007·Granted Oct 14, 2014·4 cites·11 claims
- 1084US6521663B2Aminoguanidinyl- and Alkoxyguanidinyl-substituted phenyl acetamides as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Feb 18, 2003·18 cites·30 claims
- 1184US6472399B2Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Oct 29, 2002·13 cites·26 claims
- 1284US6420397B1Heteroaryl protease inhibitors and diagnostic imaging agentsDIMENSIONAL PHARM INC·Filed 2000·Granted Jul 16, 2002·15 cites·35 claims
- 1383US6900231B2Aminopyridyl-substituted phenyl acetamides as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2002·Granted May 31, 2005·15 cites·30 claims
- 1482US6706765B2Aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2003·Granted Mar 16, 2004·12 cites·34 claims
- 1582US5741819AArylsulfonylaminobenzene derivatives and the use thereof as factor Xa inhibitorsDIMENSIONAL PHARM INC·Filed 1995·Granted Apr 21, 1998·57 cites·27 claims
- 1681US7029654B2Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitorsORTHO MCNEIL PHARM INC·Filed 2003·Granted Apr 18, 2006·9 cites·53 claims
- 1781US6638931B1Aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted Oct 28, 2003·11 cites·39 claims
- 1881US5792769AGuanidino protease inhibitors3-DIMENSIONAL PHARM INC·Filed 1996·Granted Aug 11, 1998·34 cites·49 claims
- 1980US7030110B2Cyclic oxyguanidine pyrazinones as protease inhibitorsORTHO MCNEIL PHARM INC·Filed 2002·Granted Apr 18, 2006·8 cites·28 claims
- 2080US6730783B2Process for preparing aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2003·Granted May 4, 2004·9 cites·39 claims
- 2180US6476016B2Cyclic oxyguanidine pyrazinones as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Nov 5, 2002·12 cites·25 claims
- 2280US6344466B2Benzamide and sulfonamide substitued aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Feb 5, 2002·13 cites·42 claims
- 2379US6518310B2Aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Feb 11, 2003·9 cites·36 claims
- 2479US6514978B2Thromboresistant materials incorporating pyrazinone protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Feb 4, 2003·11 cites·25 claims
- 2579US6281206B1Amidino protease inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted Aug 28, 2001·8 cites·28 claims
- 2676US6855722B2Substituted indoles and their use as integrin antagonistsDIMENSIONAL PHARM INC·Filed 2002·Granted Feb 15, 2005·10 cites·56 claims
- 2776US6635637B2Cyclic oxyguanidine protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Oct 21, 2003·9 cites·50 claims
- 2875US5891909AAmidinohydrazones as protease inhibitorsDIMENSIONAL PHARM INC·Filed 1997·Granted Apr 6, 1999·39 cites·76 claims
- 2974US6414020B2Amidino protease inhibitorsDIMENSIONAL PHARM INC·Filed 2001·Granted Jul 2, 2002·4 cites·27 claims
- 3073US6225302B1Amidino protease inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted May 1, 2001·4 cites·26 claims
- 3173US5514716AHydroxamic acid and carboxylic acid derivatives, process for their preparation and use thereofSTERLING WINTHROP INC·Filed 1994·Granted May 7, 1996·26 cites·15 claims
- 3271US6344484B1Tyrosine alkoxyguanidines as integrin inhibitorsDIMENSIONAL PHARM INC·Filed 2000·Granted Feb 5, 2002·6 cites·33 claims
- 3367US9394289B2Inhibitors of c-fms kinaseJANSSEN PHARMACEUTICA NV·Filed 2014·Granted Jul 19, 2016·0 cites·9 claims
- 3467US6235778B1Aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 1997·Granted May 22, 2001·17 cites·42 claims
- 3567US6204263B1Pyrazinone protease inhibitorsDIMENSIONAL PHARM INC·Filed 1999·Granted Mar 20, 2001·21 cites·34 claims
- 3665US7241789B2Substituted indoles and their use as integrin antagonistsDIMENSIONAL PHARMACEUTICAL INC·Filed 2004·Granted Jul 10, 2007·5 cites·21 claims
- 3764US5618844AHydroxamic acid and carboxylic acid derivatives, process for their preparation and use thereofSANOFI SA·Filed 1995·Granted Apr 8, 1997·20 cites·15 claims
- 3863US6034127AAmidino protease inhibitorsDIMENSIONAL PHARM INC·Filed 1996·Granted Mar 7, 2000·13 cites·32 claims
- 3962US6133315AAmidino protease inhibitorsDIMENSIONAL PHARM INC·Filed 1999·Granted Oct 17, 2000·12 cites·28 claims
- 4060US4772600AFused imidazoheterocyclic compounds and pharmaceutical compositionsROBINS CO INC A H·Filed 1986·Granted Sep 20, 1988·11 cites·160 claims
- 4160US2020223871A1Arginase Inhibitors and Methods of UseASTRAZENECA AB·Filed 2019·Application pending·0 cites
- 4259US2006058291A1Cyclic oxyguanidine pyrazinones as protease inhibitorsORTHO MCNEIL PHARM INC·Filed 2005·Application pending·0 cites
- 4357US2019127395A1Arginase Inhibitors and Methods of UseASTRAZENECA AB·Filed 2018·Application pending·0 cites
- 4456US6417161B1Amino acid amidinohydrazones, alkoxyguanidines and aminoguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 1999·Granted Jul 9, 2002·9 cites·39 claims
- 4556US5114944A2-phenylpyrazolo[1,5-a]pyrimidine-3-acetic acid derivatives exhibiting therapeutic effectsROBINS CO INC A H·Filed 1991·Granted May 19, 1992·5 cites·23 claims
- 4654US2007219233A1Substituted Indoles and Their Use as Integrin AntagonistsLU TIANBO·Filed 2007·Application pending·0 cites
- 4753US10118936B2Arginase inhibitors and methods of useASTRAZENECA AB·Filed 2015·Granted Nov 6, 2018·0 cites·22 claims
- 4853US2005159457A1Aminopyridinyl-, aminoguanidinyl- and alkoxyguanidinyl-substituted phenyl acetamides as protease inhibitorsFiled 2005·Application pending·0 cites
- 4953US2005228011A1Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonistsDIMENSIONAL PHARM INC·Filed 2004·Application pending·0 cites
- 5052US6344486B1Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitorsDIMENSIONAL PHARM INC·Filed 1999·Granted Feb 5, 2002·9 cites·64 claims
Showing the top 50 of 59 patent records by PatentIndex Score.
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