Inventor · disambiguated record
Jefferson Wright Tilley
Also filed as: TILLEY JEFFERSON · TILLEY JEFFERSON W · TILLEY JEFFERSON WRIGHT
78 granted patents·14 pending applications·1,122 citations·filing 1977–2017
99Inventor score
Top patents by PatentIndex Score
92 records- 0197US4927838APyridine compounds which are useful in treating a disease state characterized by an excess of platelet activating factorsHOFFMANN LA ROCHE·Filed 1988·Granted May 22, 1990·101 cites·40 claims
- 0297US4916145ASubstituted n-[(pyridyl)alkyl]aryl-carboxamideHOFFMANN LA ROCHE·Filed 1987·Granted Apr 10, 1990·74 cites·19 claims
- 0395US7807674B2Thyroid hormone analogsHOFFMANN LA ROCHE·Filed 2008·Granted Oct 5, 2010·35 cites·19 claims
- 0495US6388084B14-pyridinyl-n-acyl-l-phenylalaninesHOFFMANN LA ROCHE·Filed 2000·Granted May 14, 2002·61 cites·8 claims
- 0595US6380387B14-Pyrimidinyl-n-acyl-l phenylalaninesHOFFMANN LA ROCHE·Filed 2000·Granted Apr 30, 2002·55 cites·61 claims
- 0694US6455550B1N-alkanoylphenylalanine derivativesHOFFMANN LA ROCHE·Filed 1998·Granted Sep 24, 2002·60 cites·150 claims
- 0794US6229011B1N-aroylphenylalanine derivative VCAM-1 inhibitorsHOFFMANN LA ROCHE·Filed 1998·Granted May 8, 2001·89 cites·308 claims
- 0894US4169154AMethod of treating depression with thiourea derivativesHOFFMANN LA ROCHE·Filed 1978·Granted Sep 25, 1979·43 cites·2 claims
- 0993US7553833B23,3-spiroindolinone derivativesHOFFMANN LA ROCHE·Filed 2008·Granted Jun 30, 2009·25 cites·8 claims
- 1093US7452882B2Thyroid hormone analogsHOFFMANN LA ROCHE·Filed 2006·Granted Nov 18, 2008·24 cites·11 claims
- 1193US4786646ACyclopropylpropenamidesHOFFMANN LA ROCHE·Filed 1987·Granted Nov 22, 1988·42 cites·27 claims
- 1289US6916933B24-pyridinyl-n-acyl-l-phenylalaninesHOFFMANN LA ROCHE·Filed 2003·Granted Jul 12, 2005·23 cites·61 claims
- 1388US6806365B2N-alkanoylphenylalamine derivativesHOFFMANN LA ROCHE·Filed 2002·Granted Oct 19, 2004·17 cites·305 claims
- 1488US6288267B1Thioamide derivativesHOFFMANN LA ROCHE·Filed 2000·Granted Sep 11, 2001·23 cites·23 claims
- 1587US7947692B2Substituted thiazolo[5,4-d]pyrimidine urea derivativesHOFFMANN LA ROCHE·Filed 2007·Granted May 24, 2011·17 cites·41 claims
- 1687US6423728B1Heterocyclic thioamide derivativesHOFFMANN LA ROCHE·Filed 2001·Granted Jul 23, 2002·21 cites·26 claims
- 1786US6426348B1Diphenyl heterocyclic thioamide derivativesHOFFMANN LA ROCHE·Filed 2001·Granted Jul 30, 2002·17 cites·9 claims
- 1885US6479666B2Phenyl-keto-imidazolidine thioamide derivativesHOFFMANN LA ROCHE·Filed 2001·Granted Nov 12, 2002·16 cites·21 claims
- 1984US8076334B2Prodrugs of thyroid hormone analogsHAYNES NANCY-ELLEN·Filed 2008·Granted Dec 13, 2011·15 cites·18 claims
- 2084US7728029B2Adamantyl-pyrazole carboxamides as inhibitors of 11β-hdroxysteroid dehydrogenaseHOFFMANN LA ROCHE·Filed 2007·Granted Jun 1, 2010·8 cites·19 claims
- 2184US6458844B2Diphenyl carbocyclic thioamide derivativesHOFFMANN LA ROCHE·Filed 2001·Granted Oct 1, 2002·15 cites·25 claims
- 2283US7524870B2Biaryloxymethylarenecarboxylic acids as glycogen synthase activatorsHOFFMANN LA ROCHE·Filed 2005·Granted Apr 28, 2009·4 cites·13 claims
- 2383US4788206APentadieneamidesHOFFMANN LA ROCHE·Filed 1987·Granted Nov 29, 1988·32 cites·30 claims
- 2482US5344843ACat-1 inhibitors, pharmaceutical compositions and methods of useHOFFMANN LA ROCHE·Filed 1992·Granted Sep 6, 1994·28 cites·38 claims
- 2582US4202978A(S)-1-[2-(4-(2-Hydroxy-s-(1-alkylaminopropoxy)phenylalkyl]-4-phenylpiperazinesHOFFMANN LA ROCHE·Filed 1978·Granted May 13, 1980·18 cites·26 claims
- 2679USRE46024EThyroid hormone analogsHOFFMANN LA ROCHE·Filed 2015·Granted Jun 7, 2016·2 cites·19 claims
- 2779US4329289AAdrenergic blocking agentsHOFFMANN LA ROCHE·Filed 1981·Granted May 11, 1982·10 cites·2 claims
- 2878US4551460APyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosisHOFFMANN LA ROCHE·Filed 1983·Granted Nov 5, 1985·10 cites·58 claims
- 2977US7741327B2Pyrrolidinone glucokinase activatorsHOFFMANN LA ROCHE·Filed 2009·Granted Jun 22, 2010·3 cites·31 claims
- 3077US7642244B2Neuropeptide-2 receptor (Y-2R) agonists and uses thereofHOFFMANN LA ROCHE·Filed 2006·Granted Jan 5, 2010·4 cites·18 claims
- 3177US6265572B1Pyrrolidincarbonylamino cyclic disulfide anti-inflammatory agentsHOFFMANN LA ROCHE·Filed 2000·Granted Jul 24, 2001·10 cites·26 claims
- 3277US4285873AAdrenergic blocking agentsHOFFMANN LA ROCHE·Filed 1980·Granted Aug 25, 1981·9 cites·1 claims
- 3377US4281189ASulfonamide intermediates for adrenergic blocking agentsHOFFMANN LA ROCHE·Filed 1980·Granted Jul 28, 1981·9 cites·2 claims
- 3476US7652053B2Diaminocycloalkane MCH receptor antagonistsHOFFMANN LA ROCHE·Filed 2007·Granted Jan 26, 2010·2 cites·19 claims
- 3576US7355049B2Biaryloxymethylarenecarboxylic acids as glycogen synthase activatorHOFFMANN LA ROCHE·Filed 2004·Granted Apr 8, 2008·8 cites·18 claims
- 3676US4066695AThiourea derivativesHOFFMANN LA ROCHE·Filed 1977·Granted Jan 3, 1978·11 cites·3 claims
- 3775US8344027B24-dimethylaminobutyric acid derivativesHOFFMANN LA ROCHE·Filed 2009·Granted Jan 1, 2013·2 cites·30 claims
- 3875US8188098B2GPR119 receptor agonistsERICKSON SHAWN DAVID·Filed 2009·Granted May 29, 2012·5 cites·2 claims
- 3974US4348396ASubstituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with themHOFFMANN LA ROCHE·Filed 1980·Granted Sep 7, 1982·8 cites·35 claims
- 4073US8258134B2Pyridazinone glucokinase activatorsBERTHEL STEVEN JOSEPH·Filed 2009·Granted Sep 4, 2012·2 cites·2 claims
- 4173US4927826ACycloproylpropenamides useful as platelet activing factor (PAF) antagonistsHOFFMANN LA ROCHE·Filed 1988·Granted May 22, 1990·10 cites·18 claims
- 4272US7842825B2Biaryloxymethylarenecarboxylic acids as glycogen synthase activatorHOFFMANN LA ROCHE·Filed 2008·Granted Nov 30, 2010·1 cites·9 claims
- 4371US5128448ACCK analogs with appetite regulating activityHOFFMANN LA ROCHE·Filed 1990·Granted Jul 7, 1992·30 cites·47 claims
- 4469US9321750B2ROR modulators and their usesINNOV17 LLC·Filed 2013·Granted Apr 26, 2016·1 cites·7 claims
- 4569US6420600B1Phenylalaninol derivativesHOFFMANN LA ROCHE·Filed 2000·Granted Jul 16, 2002·4 cites·15 claims
- 4668US5182263AAnalogs of tyrosine sulfate or tyrosine phosphate containing peptidesHOFFMANN LA ROCHE·Filed 1991·Granted Jan 26, 1993·23 cites·30 claims
- 4768US4599336ADerivatives of (E)-3-(4-oxo-4H-quinazolin-3-yl)-2-propenamideHOFFMANN LA ROCHE·Filed 1983·Granted Jul 8, 1986·7 cites·28 claims
- 4868US4304721AAdrenergic blocking agentsHOFFMANN LA ROCHE·Filed 1980·Granted Dec 8, 1981·25 cites·1 claims
- 4966US4113776A1-(2-Aminoethyl)-3-(2,6-dihalophenyl)guanidinesHOFFMANN LA ROCHE·Filed 1977·Granted Sep 12, 1978·6 cites·3 claims
- 5062US4336382A1,4-Disubstituted piperazine compoundsHOFFMANN LA ROCHE·Filed 1980·Granted Jun 22, 1982·4 cites·11 claims
Showing the top 50 of 92 patent records by PatentIndex Score.
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