Inventor · disambiguated record
Arlindo L. Castelhano
Also filed as: CASTELHANO ARLINDO · CASTELHANO ARLINDO L · CASTELHANO ARLINDO LUCAS
49 granted patents·9 pending applications·1,050 citations·filing 1985–2022
98Inventor score
Top patents by PatentIndex Score
58 records- 0195US6680324B2Compounds specific to adenosine A1 receptors and uses thereofOSI PHARM INC·Filed 2001·Granted Jan 20, 2004·68 cites·37 claims
- 0295US6680322B2Compounds specific to adenosine A1 receptors and uses thereofOSI PHARM INC·Filed 2000·Granted Jan 20, 2004·67 cites·37 claims
- 0392US7485658B2N-substituted pyrazolyl-amidyl-benzimidazolyl c-Kit inhibitorsOSI PHARM INC·Filed 2004·Granted Feb 3, 2009·39 cites·5 claims
- 0492US6916804B2Pyrimidine A2b selective antagonist compounds, their synthesis and useOSI PHARM INC·Filed 2002·Granted Jul 12, 2005·45 cites·22 claims
- 0592US6143744ASulfamide-metalloprotease inhibitorsSYNTEX INC·Filed 1999·Granted Nov 7, 2000·55 cites·46 claims
- 0691US5998412ASulfamide-metalloprotease inhibitorsSYNTEX INC·Filed 1998·Granted Dec 7, 1999·52 cites·15 claims
- 0790US6376506B1Sulfamide-metalloprotease inhibitorsSYNTEX LLC·Filed 1999·Granted Apr 23, 2002·47 cites·5 claims
- 0889US6800633B2Pyrrolo[2,3d]pyrimidine compositions and their useOSI PHARM INC·Filed 2000·Granted Oct 5, 2004·29 cites·16 claims
- 0989US6673802B2Compounds specific to adenosine A3 receptor and uses thereofOSI PHARM INC·Filed 2001·Granted Jan 6, 2004·26 cites·16 claims
- 1088US7504407B2Compounds specific to adenosine A1 and A3 receptors and uses thereofOSI PHARM INC·Filed 2002·Granted Mar 17, 2009·29 cites·12 claims
- 1188US5932595AMatrix metalloprotease inhibitorsSYNTEX INC·Filed 1996·Granted Aug 3, 1999·88 cites·60 claims
- 1286US6664252B24-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereofOSI PHARM INC·Filed 2000·Granted Dec 16, 2003·28 cites·34 claims
- 1385US7160890B2Compounds specific to adenosine A3 receptor and uses thereofOSI PHARM INC·Filed 2000·Granted Jan 9, 2007·16 cites·46 claims
- 1485US6008243AMetalloproteinase inhibitors, pharmaceutical compositions containing them, and their useAGOURON PHARMA·Filed 1997·Granted Dec 28, 1999·70 cites·15 claims
- 1585US4970297ATransglutaminase inhibitorsSYNTEX INC·Filed 1987·Granted Nov 13, 1990·22 cites·22 claims
- 1683US7429574B24-heterocyclo-pyrrolo[2,3d] pyrimidine compositions and their useOSI PHARM INC·Filed 2004·Granted Sep 30, 2008·14 cites·8 claims
- 1783US6495699B2Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their useAGOURON PHARMA·Filed 2001·Granted Dec 17, 2002·11 cites·1 claims
- 1883US6130220ASulfamide-metalloprotease inhibitorsSYNTEX INC·Filed 1999·Granted Oct 10, 2000·30 cites·44 claims
- 1982US6949563B2(2-carboxamido)(3-amino)thiophene compoundsWYNNE GRAHAM MICHAEL·Filed 2004·Granted Sep 27, 2005·19 cites·16 claims
- 2082US4912120A3,5-substituted 4,5-dihydroisoxazoles as transglutaminase inhibitorsSYNTEX INC·Filed 1987·Granted Mar 27, 1990·55 cites·32 claims
- 2181US6878716B1Compounds specific to adenosine A1 receptor and uses thereofOSI PHARM INC·Filed 1999·Granted Apr 12, 2005·27 cites·35 claims
- 2281US4929630ATransglutaminase inhibitorsSYNTEX INC·Filed 1989·Granted May 29, 1990·49 cites·13 claims
- 2378US7262196B2Tri(cyclo) substituted amide glucokinase activator compoundsPROSIDION LTD·Filed 2004·Granted Aug 28, 2007·11 cites·17 claims
- 2476US7501407B2Pyrimidine A2B selective antagonist compounds, their synthesis and useOSI PHARM INC·Filed 2004·Granted Mar 10, 2009·8 cites·7 claims
- 2575US8557814B2mTOR inhibitor salt formsCASTELHANO ARLINDO L·Filed 2009·Granted Oct 15, 2013·4 cites·18 claims
- 2674US7521448B2N-substituted benzimidazolyl c-Kit inhibitorsOSI PHARM INC·Filed 2004·Granted Apr 21, 2009·9 cites·6 claims
- 2774US7439256B2(Arylamidoaryl) cyanoguanidine compoundsCASTELHANO ARLINDO·Filed 2005·Granted Oct 21, 2008·5 cites·8 claims
- 2873US7645754B2Pyrrolopyrimidine A2B selective antagonist compounds, their synthesis and useOSI PHARM INC·Filed 2007·Granted Jan 12, 2010·1 cites·10 claims
- 2973US7598252B2Compounds specific to adenosine A, receptors and uses thereofOSI PHARM INC·Filed 2003·Granted Oct 6, 2009·4 cites·6 claims
- 3073US6037472AMatrix metalloprotease inhibitorsSYNTEX INC·Filed 1994·Granted Mar 14, 2000·23 cites·15 claims
- 3170US12116359B2EBNA1 inhibitor crystalline forms, and methods of preparing and using sameTHE WISTAR INST·Filed 2022·Granted Oct 15, 2024·0 cites·10 claims
- 3269US6686366B1Compounds specific to adenosine A3 receptor and uses thereofOSI PHARM INC·Filed 1999·Granted Feb 3, 2004·32 cites·50 claims
- 3367US7662844B2Naphthylene derivatives as cytochrome P450 inhibitorsOSI PHARM INC·Filed 2004·Granted Feb 16, 2010·6 cites·33 claims
- 3467US7064122B2Pancreatic lipase inhibitor compounds, their synthesis and useOSI PHARM INC·Filed 2002·Granted Jun 20, 2006·3 cites·27 claims
- 3564US7442709B2N3-substituted imidazopyridine c-Kit inhibitorsOSI PHARM INC·Filed 2004·Granted Oct 28, 2008·2 cites·4 claims
- 3663US11242338B2EBNA1 inhibitor crystalline forms, and methods of preparing and using sameTHE WISTAR INST·Filed 2019·Granted Feb 8, 2022·0 cites·25 claims
- 3763US7767673B2N-substituted imidazopyridine c-Kit inhibitorsOSI PHARM INC·Filed 2008·Granted Aug 3, 2010·0 cites·8 claims
- 3862US2009082369A1Pyrrolo[2,3d]pyrimidine compositions and their useOSI PHARM INC·Filed 2008·Application pending·0 cites
- 3960US6376667B1Solid phase synthesis of heterocyclesOSI PHARM INC·Filed 1998·Granted Apr 23, 2002·7 cites·4 claims
- 4060US2008070936A1Compounds specific to adenosine A1 receptors and uses thereofOSI PHARM INC·Filed 2007·Application pending·0 cites
- 4159US6037340ASynthesis and use of thiophene- and pyrrole-based heteroaromatic compoundsOSI PHARM·Filed 1997·Granted Mar 14, 2000·9 cites·64 claims
- 4258US2009192177A12-ARYL pyrrologpyrimidines for A1 and A3 receptorsOSI PHARM INC·Filed 2008·Application pending·0 cites
- 4357US6638941B1Conformationallly constrained peptidomimetics as β-turn templates and modulators of SH3 domainsOSI PHARM INC·Filed 1998·Granted Oct 28, 2003·9 cites·24 claims
- 4456US4668703Aγ-allenyl-γ-aminobutyric acidsSYNTEX INC·Filed 1985·Granted May 26, 1987·4 cites·20 claims
- 4555US6013792AMatrix metalloprotease inhibitorsSYNTEX INC·Filed 1995·Granted Jan 11, 2000·12 cites·22 claims
- 4651US2003212067A1Matrix metalloprotease inhibitorsFiled 2003·Application pending·0 cites
- 4749US2003229067A1Pyrrolopyrimidine A2b selective antagonist compounds, their synthesis and useFiled 2002·Application pending·0 cites
- 4848US2007129547A1Process to prepare substituted imidazopyrazine compoundsMULVIHILL KRISTEN M·Filed 2006·Application pending·0 cites
- 4947US6306892B1Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their useAGOURON PHARMA·Filed 2000·Granted Oct 23, 2001·0 cites·20 claims
- 5044USH1992HMetalloproteinase inhibitors, pharmaceutical compositions containing them, and their pharmaceutical usesAGOURON PHARMA·Filed 1999·Granted Sep 4, 2001·2 cites·26 claims
Showing the top 50 of 58 patent records by PatentIndex Score.
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