Inventor · disambiguated record
Philippe Yaiche
Also filed as: YAICHE PHILIPPE
43 granted patents·5 pending applications·64 citations·filing 2001–2013
96Inventor score
Technology areasA61P
Top patents by PatentIndex Score
48 records- 0189US8697883B2Cyclopenta[C]pyrrole-2-carboxylate derivatives, preparation thereof and therapeutic use thereofABOUABDELLAH AHMED·Filed 2010·Granted Apr 15, 2014·19 cites·10 claims
- 0282US8592437B2Heteroarylamide pyrimidone compoundsLOCHEAD ALISTAIR·Filed 2009·Granted Nov 26, 2013·6 cites·20 claims
- 0381US8394787B27-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereofABOUABDELLAH AHMED·Filed 2010·Granted Mar 12, 2013·6 cites·13 claims
- 0476US7247638B28-Substituted-6,7,8,9-tetrahydropyrimido [1,2-a] pyrimidin-4-one derivatives.MITSUBISHI PHARMA CORP·Filed 2005·Granted Jul 24, 2007·2 cites·17 claims
- 0576US7217715B2Substituted 8-perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivativesMITSUBISHI PHARMA CORP·Filed 2005·Granted May 15, 2007·2 cites·18 claims
- 0674US8865738B25-membered heterocyclic compound cyclopenta[C]pyrrolylalkylcarbamate derivatives, preparation thereof, and therapeutic use thereofABOUABDELLAH AHMED·Filed 2010·Granted Oct 21, 2014·3 cites·15 claims
- 0773US7566720B22-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivativesSANOFI AVENTIS·Filed 2007·Granted Jul 28, 2009·1 cites·5 claims
- 0873US7507743B2Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one derivativesSANOFI AVENTIS·Filed 2007·Granted Mar 24, 2009·1 cites·4 claims
- 0973US7465737B2Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl -6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivativesSANOFI AVENTIS·Filed 2007·Granted Dec 16, 2008·1 cites·12 claims
- 1072US8592580B2Substituted triazinone derivativesLOCHEAD ALISTAIR·Filed 2010·Granted Nov 26, 2013·2 cites·9 claims
- 1172US7781440B2Use of substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivativesSANOFI AVENTIS·Filed 2008·Granted Aug 24, 2010·1 cites·10 claims
- 1272US7547705B2Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivativesSANOFI AVENTIS·Filed 2007·Granted Jun 16, 2009·1 cites·5 claims
- 1372US7462621B2Use of substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives as therapeutic agentsSANOFI AVENTIS·Filed 2007·Granted Dec 9, 2008·1 cites·8 claims
- 1472US7232827B2Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one derivativesMITSUBISHI PHARMA CORP·Filed 2003·Granted Jun 19, 2007·5 cites·12 claims
- 1571US8598187B2Arylamide pyrimidone compoundsLOCHEAD ALISTAIR·Filed 2009·Granted Dec 3, 2013·1 cites·22 claims
- 1670US8889702B2Derivatives of azaspiranyl-alkylcarbamates of 5-member heterocyclic compounds, preparation thereof and therapeutic use thereofABOUABDELLAH AHMED·Filed 2010·Granted Nov 18, 2014·2 cites·12 claims
- 1770US8716289B2Carbamate derivatives of alkyl-heterocycles, preparation thereof and therapeutic use thereofABOUABDELLAH AHMED·Filed 2009·Granted May 6, 2014·1 cites·12 claims
- 1869US8598175B2Heteroarylamide pyrimidone derivativesCHEREZE NATHALIE·Filed 2009·Granted Dec 3, 2013·1 cites·20 claims
- 1969US8592436B2Arylamide pyrimidone derivativesCHEREZE NATHALIE·Filed 2009·Granted Nov 26, 2013·1 cites·20 claims
- 2065US8507476B2Substituted arylamide diazepinopyrimidone derivativesFAYOL AUDE·Filed 2010·Granted Aug 13, 2013·1 cites·12 claims
- 2165US7214682B2Substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo{1,2-a}pyrimidin-5(1h)one derivativesMITSUBISHI PHARMA CORP·Filed 2002·Granted May 8, 2007·2 cites·10 claims
- 2265US7067521B21-[alkyl], 1-[(heteroaryl)alkyl] and 1-[(aryl)alkyl]-7pyridinyl-imidazo[1,2-alpha]pyrimidin-5(1H)-one derivativesSANOFI AVENTIS·Filed 2001·Granted Jun 27, 2006·2 cites·10 claims
- 2365US6974819B22-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydoimidazo{1,2-a}pyrimidin-5(1H)one derivativesMITSUBISHI PHARMA CORP·Filed 2001·Granted Dec 13, 2005·2 cites·16 claims
- 2458US2008318980A1USE OF 7-(PYRIMIDIN-4 YL)-IMIDAZO[1,2-a]PYRIMIDIN-5(1H)-ONES AS GSK-3BETA INHIBITORSSANOFI AVENTIS·Filed 2008·Application pending·0 cites
- 2555US8148364B2Substituted bicyclic pyrimidone derivativesCHEREZE NATHALIE·Filed 2008·Granted Apr 3, 2012·0 cites·10 claims
- 2655US8093256B2Use of 8-substituted-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivativesLOCHEAD ALISTAIR·Filed 2007·Granted Jan 10, 2012·0 cites·18 claims
- 2755US7452897B2Use of substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives for the treatment of neurodegenerative diseasesSANOFI AVENTIS·Filed 2007·Granted Nov 18, 2008·0 cites·8 claims
- 2855US7393853B2Use of substituted 8-Perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives as therapeutic agentsSANOFI AVENTIS·Filed 2007·Granted Jul 1, 2008·0 cites·20 claims
- 2954US2006014762A12-Pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-A]pyrimidin-4-one and 7-pyridinyl-2,3-dihydoimidazo[1,2-A]pyrimidin-5(1H)one derivativesMITSUBISHI PHARMA CORP·Filed 2005·Application pending·0 cites
- 3053US7608624B21-[alkyl], 1-[(heteroaryl)alkyl] and 1-[(aryl)alkyl]-7-pyridinyl-imidazo[1,2-a]pyrimidin-5(1h)-one derivativesSANOFI AVENTIS·Filed 2006·Granted Oct 27, 2009·0 cites·7 claims
- 3153US7294631B2Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivativesSANOFI AVENTIS·Filed 2006·Granted Nov 13, 2007·0 cites·13 claims
- 3252US7294632B2Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one derivativesSANOFI AVENTIS·Filed 2005·Granted Nov 13, 2007·0 cites·11 claims
- 3351US8198287B2Substituted heteroaryl pyridopyrimidone derivativesFAYOL AUDE·Filed 2009·Granted Jun 12, 2012·0 cites·10 claims
- 3451US7429663B27-(Pyrimidin-4-yl)-Imidazo[1,2-a]Pyrimidin-5(1H)-ones as GSK3β inhibitorsSANOFI AVENTIS·Filed 2003·Granted Sep 30, 2008·0 cites·6 claims
- 3551US7211581B2Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivativesMITSUBISHI PHARMA CORP·Filed 2005·Granted May 1, 2007·0 cites·7 claims
- 3651US2009281121A1SUBSTITUTED 8-PIPERIDINYL-2-PYRIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE AND 8-PIPERIDINYL-2-PYRIMIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE DERIVATIVESSANOFI AVENTIS·Filed 2009·Application pending·0 cites
- 3748US7388005B2Substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo [1,2-a]pyrimidin-5(1H)one derivatives for neurodegenerative disordersSANOFI AVENTIS·Filed 2002·Granted Jun 17, 2008·0 cites·15 claims
- 3848US2013211087A17-aza-spiro[3,5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereofABOUABDELLAH AHMED·Filed 2013·Application pending·0 cites
- 3943US2011294786A1Substituted bicyclic pyrimidone derivativesCHEREZE NATHALIE·Filed 2011·Application pending·0 cites
- 4039US8211903B2Substituted pyrimido isoquinoline derivativesLOCHEAD ALISTAIR·Filed 2010·Granted Jul 3, 2012·0 cites·6 claims
- 4139US8202874B2Substituted N-oxide pyrazine derivativesLOCHEAD ALISTAIR·Filed 2010·Granted Jun 19, 2012·0 cites·6 claims
- 4238US9073915B2Substituted pyrimidone derivativesLOCHEAD ALISTAIR·Filed 2010·Granted Jul 7, 2015·0 cites·9 claims
- 4337US9073914B2Substituted alkyl pyrimidin-4-one derivativesFAYOL AUDE·Filed 2010·Granted Jul 7, 2015·0 cites·11 claims
- 4437US8614219B2Substituted pyrimidin-4-one derivativesFAYOL AUDE·Filed 2010·Granted Dec 24, 2013·0 cites·13 claims
- 4536US8507470B2Substituted arylamide oxazepinopyrimidone derivativesFAYOL AUDE·Filed 2010·Granted Aug 13, 2013·0 cites·12 claims
- 4636US8501728B2Substituted heteroarylamide oxazepinopyrimidone derivativesFAYOL AUDE·Filed 2010·Granted Aug 6, 2013·0 cites·12 claims
- 4735US8507475B2Substituted heteroarylamide diazepinopyrimidone derivativesFAYOL AUDE·Filed 2010·Granted Aug 13, 2013·0 cites·12 claims
- 4833US8273758B2Substituted tricyclic derivativesALMARIO GARCIA ANTONIO·Filed 2010·Granted Sep 25, 2012·0 cites·9 claims
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