Inventor · disambiguated record
Michael Hale
Also filed as: HALE MICHAEL · HALE MICHAEL R · HALE MICHAEL ROBIN
48 granted patents·19 pending applications·1,686 citations·filing 1997–2025
99Inventor score
Top patents by PatentIndex Score
67 records- 0198US6784195B2Pyrazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2001·Granted Aug 31, 2004·182 cites·21 claims
- 0297US7345054B2Heterocyclic inhibitors of ERK2 and uses thereofVERTEX PHARMA·Filed 2005·Granted Mar 18, 2008·57 cites·9 claims
- 0397US6319946B1Inhibitors of aspartyl proteaseVERTEX PHARMA·Filed 2000·Granted Nov 20, 2001·88 cites·22 claims
- 0496US7354939B2Pyrrole inhibitors of ERK protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2005·Granted Apr 8, 2008·52 cites·9 claims
- 0596US7304061B2Heterocyclic inhibitors of ERK2 and uses thereofVERTEX PHARMA·Filed 2003·Granted Dec 4, 2007·65 cites·22 claims
- 0696US6743791B2Heterocyclic inhibitors of ERK2 and uses thereofVERTEX PHARMA·Filed 2002·Granted Jun 1, 2004·123 cites·57 claims
- 0796US6495582B1Isoxazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2001·Granted Dec 17, 2002·104 cites·25 claims
- 0895US7253187B2Heterocyclic inhibitors of ERK2 and uses thereofVERTEX PHARMA·Filed 2004·Granted Aug 7, 2007·90 cites·25 claims
- 0995US6699865B2Pyrazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2003·Granted Mar 2, 2004·71 cites·21 claims
- 1095US6593357B1Pyrazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2002·Granted Jul 15, 2003·81 cites·21 claims
- 1195US6528509B1Pyrazole compositions useful as inhibitors of ERKVERTEX PHARMACUTICALS INC·Filed 2001·Granted Mar 4, 2003·177 cites·21 claims
- 1293US7056944B2Pyrazole compositions useful as inhibitors of erkVERTEX PHARMA·Filed 2003·Granted Jun 6, 2006·56 cites·24 claims
- 1393US6949580B2Pyrazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2003·Granted Sep 27, 2005·58 cites·8 claims
- 1492US7501415B2Selective inhibitors of ERK protein kinase and uses thereofVERTEX PHARMA·Filed 2005·Granted Mar 10, 2009·25 cites·7 claims
- 1592US7358258B2Prodrugs of an ERK protein kinase inhibitorVERTEX PHARMA·Filed 2005·Granted Apr 15, 2008·23 cites·6 claims
- 1691US12006330B2Substituted macrocyclic compounds and related methods of treatmentALKERMES INC·Filed 2021·Granted Jun 11, 2024·2 cites·113 claims
- 1791US6613743B2Sulfonamide inhibitors of aspartyl proteaseVERTEX PHARMA·Filed 2000·Granted Sep 2, 2003·24 cites·25 claims
- 1891US6436989B1Prodrugs of aspartyl protease inhibitorsVERTEX PHARMA·Filed 1997·Granted Aug 20, 2002·62 cites·12 claims
- 1990US12054495B2Substituted macrocyclic compounds and related methods of treatmentALKERMES INC·Filed 2022·Granted Aug 6, 2024·1 cites·51 claims
- 2090US7244735B2Heterocyclic protein kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2004·Granted Jul 17, 2007·39 cites·13 claims
- 2188US7304071B2Protein kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2003·Granted Dec 4, 2007·35 cites·20 claims
- 2288US6649640B2Isoxazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2002·Granted Nov 18, 2003·25 cites·10 claims
- 2387USRE49500EPyrrole inhibitors of ERK protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2020·Granted Apr 25, 2023·1 cites·17 claims
- 2487US7407962B2Heteroaryl compounds useful as inhibitors or protein kinasesVERTEX PHARMA·Filed 2004·Granted Aug 5, 2008·29 cites·16 claims
- 2586US7456190B2Compositions useful as protein kinase inhibitorsVERTEX PHARMA·Filed 2004·Granted Nov 25, 2008·24 cites·9 claims
- 2686US7279476B2Pyrazole-derived kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2005·Granted Oct 9, 2007·14 cites·18 claims
- 2785US6875789B2Pyrazole-derived kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2002·Granted Apr 5, 2005·24 cites·5 claims
- 2884US11542276B2Substituted macrocyclic compounds and related methods of treatmentALKERMES INC·Filed 2020·Granted Jan 3, 2023·1 cites·122 claims
- 2984US6750239B2Pyrazole-derived kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2002·Granted Jun 15, 2004·22 cites·27 claims
- 3084US6693108B2Inhibitors of c-JUN N terminal kinases (JNK) and other protein kinasesVERTEX PHARMA·Filed 2002·Granted Feb 17, 2004·20 cites·11 claims
- 3184US6559137B1Sulphonamide derivatives as prodrugs of aspartyl protease inhibitorsVERTEX PHARMA·Filed 2000·Granted May 6, 2003·17 cites·41 claims
- 3282US7169798B2Inhibitors of c-Jun N terminal kinases (JNK) and other protein kinasesVERTEX PHARMA·Filed 2004·Granted Jan 30, 2007·16 cites·11 claims
- 3382US6706711B2Pyrazole derived kinase inhibitorVERTEX PHARMA·Filed 2002·Granted Mar 16, 2004·17 cites·28 claims
- 3482US2023183276A1Pyrrole inhibitors of erk protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2023·Application pending·0 cites
- 3579US7462612B2Pyridine inhibitors of ERK2 and uses thereofVERTEX PHARMA·Filed 2005·Granted Dec 9, 2008·4 cites·15 claims
- 3679US7419967B2Sulfonamide inhibitors of aspartyl proteaseVERTEX PHARMA·Filed 2005·Granted Sep 2, 2008·2 cites·13 claims
- 3779US6962936B2Triazole-derived kinase inhibitors and uses thereofVERTEX PHARMA·Filed 2002·Granted Nov 8, 2005·10 cites·22 claims
- 3879US2025092063A1Substituted Macrocyclic Compounds and Related Methods of TreatmentALKERMES INC·Filed 2024·Application pending·0 cites
- 3978USRE48266EPyrrole inhibitors of ERK protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2019·Granted Oct 20, 2020·1 cites·17 claims
- 4077US7183307B2Pyrazole-derived kinase inhibitors and uses thereofVERTEX PHARMACEUTICALS INCROPO·Filed 2004·Granted Feb 27, 2007·15 cites·7 claims
- 4176US8455497B2Inhibitors of aspartyl proteaseHALE MICHAEL R·Filed 2009·Granted Jun 4, 2013·2 cites·40 claims
- 4275USRE47318EPyrrole inhibitors of erk protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2016·Granted Mar 26, 2019·1 cites·17 claims
- 4375US7354919B2Isoxazole compositions useful as inhibitors of ERKVERTEX PHARMA·Filed 2003·Granted Apr 8, 2008·6 cites·19 claims
- 4475US6838474B2Sulphonamide derivatives as prodrugs of aspartyl protease inhibitorsVERTEX PHARMA·Filed 2003·Granted Jan 4, 2005·6 cites·12 claims
- 4574US6617350B2Inhibitors of aspartyl proteaseVERTEX PHARMA·Filed 2001·Granted Sep 9, 2003·5 cites·22 claims
- 4674US2024368182A1Substituted Macrocyclic Compounds and Related Methods of TreatmentALKERMES INC·Filed 2024·Application pending·0 cites
- 4773USRE46097EPyrrole inhibitors of ERK protein kinase, synthesis thereof and intermediates theretoVERTEX PHARMA·Filed 2013·Granted Aug 9, 2016·1 cites·13 claims
- 4872US6878728B1Inhibitors of aspartyl proteaseVERTEX PHARMA·Filed 2000·Granted Apr 12, 2005·7 cites·20 claims
- 4967US2010124543A1Sulphonamide derivatives as prodrugs of aspartyl protease inhibitorsVERTEX PHARMA·Filed 2009·Application pending·0 cites
- 5064US7592368B2Sulphonamide derivatives as prodrugs of aspartyl protease inhibitorsVERTEX PHARMA·Filed 2004·Granted Sep 22, 2009·1 cites·20 claims
Showing the top 50 of 67 patent records by PatentIndex Score.
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