Inventor · disambiguated record
Paul F. Jackson
Also filed as: JACKSON PAUL · JACKSON PAUL F · JACKSON PAUL FRANCIS
58 granted patents·23 pending applications·2,690 citations·filing 1993–2022
99Inventor score
Files withGUILFORD PHARM INC46ZENECA LTD7JACKSON PAUL F5JACKSON PAUL FRANCIS3JANSSEN PHARMACEUTICA NV3
Top patents by PatentIndex Score
81 records- 0197US5968915ANaaladase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Oct 19, 1999·102 cites·14 claims
- 0296US6635642B1PARP inhibitors, pharmaceutical compositions comprising same, and methods of using sameGUILFORD PHARM INC·Filed 1998·Granted Oct 21, 2003·157 cites·2 claims
- 0396US6121278ADi-n-heterocyclic compounds, methods, and compositions for inhibiting parp activityGUILFORD PHARM INC·Filed 1998·Granted Sep 19, 2000·109 cites·115 claims
- 0496US5863536APhosphoramidate derivativesGUILFORD PHARM INC·Filed 1996·Granted Jan 26, 1999·121 cites·24 claims
- 0596US5672592ACertain phosphonomethyl-pentanedioic acid derivatives thereofGUILFORD PHARM INC·Filed 1996·Granted Sep 30, 1997·100 cites·11 claims
- 0695US6017903APharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Jan 25, 2000·88 cites·40 claims
- 0795US5880112ANaaladase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Mar 9, 1999·86 cites·9 claims
- 0894US5795877AInhibitors of NAALADase enzyme activityGUILFORD PHARM INC·Filed 1996·Granted Aug 18, 1998·143 cites·24 claims
- 0993US6265609B1Thio-substituted pentanedioic acid derivativesGUILFORD PHARM INC·Filed 1999·Granted Jul 24, 2001·66 cites·35 claims
- 1093US5962521AHydroxamic acid derivativesGUILFORD PHARM INC·Filed 1997·Granted Oct 5, 1999·90 cites·35 claims
- 1192US6426415B1Alkoxy-substituted compounds, methods and compositions for inhibiting parp activityGUILFORD PHARM INC·Filed 1998·Granted Jul 30, 2002·66 cites·16 claims
- 1291US6197785B1Alkoxy-substituted compounds, methods, and compositions for inhibiting PARP activityGUILFORD PHARM INC·Filed 1998·Granted Mar 6, 2001·90 cites·23 claims
- 1391US6011021AMethods of cancer treatment using naaladase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Jan 4, 2000·51 cites·32 claims
- 1491US5902817ACertain sulfoxide and sulfone derivativesGUILFORD PHARM INC·Filed 1997·Granted May 11, 1999·104 cites·17 claims
- 1590US6384022B1Prodrugs of NAALAdase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted May 7, 2002·82 cites·85 claims
- 1690US6346536B1Poly(ADP-ribose) polymerase inhibitors and method for treating neural or cardiovascular tissue damage using the sameGUILFORD PHARM INC·Filed 1997·Granted Feb 12, 2002·44 cites·19 claims
- 1790US6313159B1Metabotropic glutamate receptor ligand derivatives as naaladase inhibitorsGUILFORD PHARM INC·Filed 1999·Granted Nov 6, 2001·39 cites·22 claims
- 1890US6054444APhosphonic acid derivativesGUILFORD PHARM INC·Filed 1997·Granted Apr 25, 2000·83 cites·33 claims
- 1989US6514983B1Compounds, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damageGUILFORD PHARM INC·Filed 1998·Granted Feb 4, 2003·85 cites·21 claims
- 2089US6452044B2Benzenedicarboxylic acid derivativesGUILFORD PHARM INC·Filed 2001·Granted Sep 17, 2002·28 cites·38 claims
- 2189US6025345AInhibitors of NAALADase enzyme activityGUILFORD PHARM INC·Filed 1997·Granted Feb 15, 2000·46 cites·10 claims
- 2289US5824662ATreatment of global and focal ischemia using naaladase inhibitorsGUILFORD PHARM INC·Filed 1996·Granted Oct 20, 1998·74 cites·12 claims
- 2389US5804602AMethods of cancer treatment using naaladase inhibitorsGUILFORD PHARM INC·Filed 1996·Granted Sep 8, 1998·90 cites·9 claims
- 2488US6046180ANAALADase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Apr 4, 2000·79 cites·7 claims
- 2588US5977090APharmaceutical compositions and methods of treating compulsive disorders using NAALADase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Nov 2, 1999·79 cites·44 claims
- 2687US6348464B1Pyrrolecarbonylimino derivatives as naaladase inhibitorsGUILFORD PHARM INC·Filed 1999·Granted Feb 19, 2002·35 cites·23 claims
- 2783US5656626ASubstituted nitrogen heterocyclesZENECA LTD·Filed 1995·Granted Aug 12, 1997·30 cites·11 claims
- 2882US6903109B2Arylindenopyridines and related therapeutic and prophylactic methodsORTHO MUNIEL PHARMACEUTICAL IN·Filed 2002·Granted Jun 7, 2005·19 cites·24 claims
- 2982US6025344ACertain dioic acid derivatives useful as NAALADase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Feb 15, 2000·45 cites·25 claims
- 3081US6306889B1Compounds, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damageGUILFORD PHARM INC·Filed 1998·Granted Oct 23, 2001·19 cites·10 claims
- 3181US6271245B1Hydroxamic acid derivativesGUILFORD PHARM INC·Filed 1999·Granted Aug 7, 2001·37 cites·11 claims
- 3280US6071965APhosphinic alkanoic acid derivativesGUILFORD PHARM INC·Filed 1997·Granted Jun 6, 2000·58 cites·20 claims
- 3379US7803793B2Heterocyclic derived metalloprotease inhibitorsJANSSEN PHARMACEUTICA NV·Filed 2007·Granted Sep 28, 2010·5 cites·32 claims
- 3479US6372726B1Methods of cancer treatment using NAALADase inhibitorsGUILFORD PHARM INC·Filed 1999·Granted Apr 16, 2002·35 cites·12 claims
- 3579US5502048ASubstituted nitrogen heterocyclesZENECA LTD·Filed 1994·Granted Mar 26, 1996·37 cites·18 claims
- 3678US6004946ATreatment of global and focal ischemia using naaladase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Dec 21, 1999·39 cites·5 claims
- 3775US6028216AAsymmetric syntheses and intermediates for preparing enantiomer-enriched hydroxyphosphinyl derivativesGUILFORD PHARM INC·Filed 1997·Granted Feb 22, 2000·24 cites·13 claims
- 3874US6458775B1NAALADase inhibitors useful as pharmaceutical compounds and compositionsGUILFORD PHARM INC·Filed 1999·Granted Oct 1, 2002·30 cites·55 claims
- 3974US6288046B1Phosphonic acid derivativesGUILFORD PHARM INC·Filed 1999·Granted Sep 11, 2001·35 cites·22 claims
- 4073US6413948B1Pharmaceutical compositions and methods of effecting a neuronal activity in an animal using naaladase inhibitorsGUILFORD PHARM INC·Filed 1999·Granted Jul 2, 2002·29 cites·39 claims
- 4172US5985855ATreatment of global and focal ischemia using NAALADase inhibitorsGUILFORD PHARM INC·Filed 1997·Granted Nov 16, 1999·29 cites·9 claims
- 4270US6121252APhosphinic acid derivativesGUILFORD PHARM INC·Filed 1998·Granted Sep 19, 2000·34 cites·108 claims
- 4369US6380211B1Alkoxy-substituted compounds, methods, and compositions for inhibiting PARP activityGUILFORD PHARM INC·Filed 2000·Granted Apr 30, 2002·3 cites·15 claims
- 4468US6479471B1NAALADase inhibitorsGUILFORD PHARM INC·Filed 1999·Granted Nov 12, 2002·21 cites·11 claims
- 4564US6852750B2Benzenedicarboxylic acid derivativesGUILFORD PHARM INC·Filed 2002·Granted Feb 8, 2005·1 cites·14 claims
- 4663US8883473B2Methods of treatment using allosteric processing inhibitors for matrix metalloproteinasesLEONARD KRISTI A·Filed 2012·Granted Nov 11, 2014·1 cites·14 claims
- 4760US8017614B2Arylindenopyrimidines compound and use as an adenosine A2a receptor antagonistsJANSSEN PHARMACEUTICA NV·Filed 2008·Granted Sep 13, 2011·0 cites·10 claims
- 4858US2024376085A1Benzimidazoles as modulators of il-17JANSSEN PHARMACEUTICA NV·Filed 2022·Application pending·0 cites
- 4957US5747523ASubstituted ethyl α,α-diarylmethyl ether derivativesGUILFORD PHARM INC·Filed 1996·Granted May 5, 1998·6 cites·21 claims
- 5055US2006154949A1Arylindenopyridines and related therapeutic and prophylactic methodsHEINTZELMAN GEOFFREY R·Filed 2005·Application pending·0 cites
Showing the top 50 of 81 patent records by PatentIndex Score.
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