Inventor · disambiguated record
Francisco Javier Lopez-Tapia
Also filed as: LOPEZ-TAPIA FRANCISCO · LOPEZ-TAPIA FRANCISCO J · LOPEZ-TAPIA FRANCISCO JAVIER
38 granted patents·9 pending applications·180 citations·filing 1996–2020
96Inventor score
Files withHOFFMANN LA ROCHE17ROCHE PALO ALTO LLC8SYNTEX LLC5BROTHERTON-PLEISS CHRISTINE E4GENENTECH INC3
Top patents by PatentIndex Score
47 records- 0189US5859014APyrimidinedione, pyrimidinetrione, triazinedione and tetrahydroquinazolinedione derivatives as α1 -adrenergic receptor antagonistsSYNTEX INC·Filed 1996·Granted Jan 12, 1999·50 cites·21 claims
- 0288US8871760B2[1,2,4]triazolo[3,4-C][1,4]oxazines as P2X7 modulatorsBROTHERTON-PLEISS CHRISTINE E·Filed 2010·Granted Oct 28, 2014·19 cites·14 claims
- 0388US6184242B12-(substituted-phenyl)amino-imidazoline derivativesSYNTEX USA LLC·Filed 1998·Granted Feb 6, 2001·31 cites·6 claims
- 0483US8889682B2Inhibitors of bruton'S tyrosine kinaseBROTHERTON-PLEISS CHRISTINE E·Filed 2012·Granted Nov 18, 2014·8 cites·10 claims
- 0579US8940741B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Granted Jan 27, 2015·4 cites·19 claims
- 0679US6903086B2Alkoxycarbonylamino benzoic acid or alkoxycarbonylamino tetrazolyl phenyl derivatives as IP antagonistsSYNTEX LLC·Filed 2002·Granted Jun 7, 2005·16 cites·20 claims
- 0776US8481540B2Inhibitors of bruton's tyrosine kinaseBERTHEL STEVEN JOSEPH·Filed 2011·Granted Jul 9, 2013·4 cites·17 claims
- 0875US6569860B2Alkoxycarbonylamino heteroaryl carboxylic acid derivatives as IP antagonistsROCHE PALO ALTO LLC·Filed 2002·Granted May 27, 2003·11 cites·23 claims
- 0974US7776910B2Arylsulfonyl pyrrolidines as 5-HT6 inhibitorsROCHE PALO ALTO LLC·Filed 2007·Granted Aug 17, 2010·3 cites·16 claims
- 1074US6998414B2Substituted arylamides as IP antagonistsROCHE PALO ALTO LLC·Filed 2004·Granted Feb 14, 2006·6 cites·64 claims
- 1173US8742098B2Inhibitors of Bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2012·Granted Jun 3, 2014·2 cites·20 claims
- 1273US7279498B2Substituted aryl amides as IP antagonistsROCHE PALO ALTO LLC·Filed 2005·Granted Oct 9, 2007·1 cites·14 claims
- 1372US7141584B22-(substituted-phenyl)amino-imidazoline derivativesROCHE PALO ALTO LLC·Filed 2003·Granted Nov 28, 2006·3 cites·9 claims
- 1472US6596876B22-(substituted-phenyl)amino-imidazoline derivativesSYNTEX LLC·Filed 2002·Granted Jul 22, 2003·3 cites·20 claims
- 1572US6472536B12-(substituted-phenyl)amino-imidazoline derivativesSYNTEX LLC·Filed 2000·Granted Oct 29, 2002·3 cites·9 claims
- 1669US11104668B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Aug 31, 2021·0 cites·14 claims
- 1769US9469644B2Inhibitors of Bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Oct 18, 2016·1 cites·17 claims
- 1869US9458105B2Inhibitors of Bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Granted Oct 4, 2016·1 cites·5 claims
- 1968US8729078B2Inhibitors of bruton's tyrosine kinaseBILLEDEAU ROLAND JOSEPH·Filed 2012·Granted May 20, 2014·2 cites·18 claims
- 2068US2020207741A1Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2020·Application pending·0 cites
- 2165US9624201B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Apr 18, 2017·0 cites·22 claims
- 2265US9359345B2Thiazole derivatives as inhibitors of Bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Granted Jun 7, 2016·1 cites·20 claims
- 2364US10640491B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2018·Granted May 5, 2020·0 cites·6 claims
- 2464US2020181154A1Pyrazole carboxamide compounds and methods of useGENENTECH INC·Filed 2020·Application pending·0 cites
- 2563US6693200B22-(substituted-phenyl)amino-imidazoline derivativesSYNTEX LLC·Filed 2003·Granted Feb 17, 2004·1 cites·10 claims
- 2661US10093657B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2017·Granted Oct 9, 2018·0 cites·2 claims
- 2761US7244738B2Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonistsROCHE PALO ALTO LLC·Filed 2004·Granted Jul 17, 2007·1 cites·11 claims
- 2858US2019194209A1Pyrazole carboxamide compounds and methods of useGENENTECH INC·Filed 2019·Application pending·0 cites
- 2955US8372865B2Dihydropyridone amides as P2X7 modulatorsROCHE PALO ALTO LLC·Filed 2009·Granted Feb 12, 2013·0 cites·13 claims
- 3054US2018057500A1Pyrazole carboxamide compounds and methods of useGENENTECH INC·Filed 2017·Application pending·0 cites
- 3153US8153809B2Dihydropyridone ureas as P2X7 modulatorsBROTHERTON-PLEISS CHRISTINE E·Filed 2009·Granted Apr 10, 2012·0 cites·30 claims
- 3252US2007265446A1Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonistsCONNOLLY TERRENCE J·Filed 2007·Application pending·0 cites
- 3350US6335459B1Aryl carboxylic acid and aryl tetrazole derivatives as IP receptor modulatorsSYNTEX LLC·Filed 1999·Granted Jan 1, 2002·9 cites·32 claims
- 3449US9802920B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Oct 31, 2017·0 cites·23 claims
- 3549US8288552B2Dihydropyridone amidesas P2X7 modulatorsBERGER JACOB·Filed 2009·Granted Oct 16, 2012·0 cites·28 claims
- 3649US8163929B2Dihydropyridone amides as P2X7 modulatorsBERGER JACOB·Filed 2009·Granted Apr 24, 2012·0 cites·25 claims
- 3749US2022289720A1Aryl sulfonamides as small molecule stat3 inhibitorsUNIV HAWAII·Filed 2020·Application pending·0 cites
- 3848US9556150B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Jan 31, 2017·0 cites·18 claims
- 3947US9663494B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted May 30, 2017·0 cites·13 claims
- 4047US9556147B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2014·Granted Jan 31, 2017·0 cites·16 claims
- 4145US2005124607A15-Substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonistsFiled 2004·Application pending·0 cites
- 4244US7754759B2Arylsulfonyl chromans as 5-HT6 inhibitorsROCHE PALO ALTO LLC·Filed 2006·Granted Jul 13, 2010·0 cites·27 claims
- 4343US8153808B2Dihydropyridone amides as P2X7 modulatorsLOPEZ-TAPIA FRANCISCO JAVIER·Filed 2009·Granted Apr 10, 2012·0 cites·30 claims
- 4442US9499548B2Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Granted Nov 22, 2016·0 cites·17 claims
- 4542US2015290192A1Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Application pending·0 cites
- 4641US2015284394A1Inhibitors of bruton's tyrosine kinaseHOFFMANN LA ROCHE·Filed 2013·Application pending·0 cites
- 4736US8435990B2Dihydropyrimidone amides as P2X7 modulatorsBROTHERTON-PLEISS CHRISTINE E·Filed 2010·Granted May 7, 2013·0 cites·21 claims
Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →