Inventor · disambiguated record
Timothy Paul Burkholder
Also filed as: BURKHOLDER TIMOTHY P · BURKHOLDER TIMOTHY PAUL · BURKHOLDER TIMOTHY R
34 granted patents·2 pending applications·307 citations·filing 1993–2021
97Inventor score
Files withLILLY CO ELI15HOECHST MARION ROUSSEL INC6MERRELL PHARMA INC6AVENTIS PHARMA INC4ENGLER THOMAS ALBERT2
Top patents by PatentIndex Score
36 records- 0190US5635510ASubstituted pyrrolidin-3-yl-alkyl-piperidinesMERRELL PHARMA INC·Filed 1994·Granted Jun 3, 1997·32 cites·57 claims
- 0283US7666879B2Imidazo[1,2-A]pyridine compounds as VEGF-R2 inhibitorsLILLY CO ELI·Filed 2006·Granted Feb 23, 2010·10 cites·7 claims
- 0382US6194406B1Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseaseAVENTIS PHARMA INC·Filed 1997·Granted Feb 27, 2001·33 cites·161 claims
- 0481US7045545B1Aminoalkylbenzofurans as serotonin (5-HT(2c)) agonistsLILLY CO ELI·Filed 2000·Granted May 16, 2006·12 cites·6 claims
- 0581US6638936B1Benzofurylpiperazine serotonin agonistsLILLY CO ELI·Filed 2000·Granted Oct 28, 2003·15 cites·18 claims
- 0680US6211199B1Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseasesAVENTIS PHARMA INC·Filed 1997·Granted Apr 3, 2001·29 cites·119 claims
- 0779US7897600B2Amino pyrazole compoundLILLY CO ELI·Filed 2009·Granted Mar 1, 2011·6 cites·9 claims
- 0879US6967201B1Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agonistsLILLY CO ELI·Filed 2000·Granted Nov 22, 2005·15 cites·9 claims
- 0977US7405299B2Compounds as pharmaceutical agentsLILLY CO ELI·Filed 2003·Granted Jul 29, 2008·15 cites·1 claims
- 1075US8058425B2Purine derivatives as kinase inhibitorsENGLER THOMAS ALBERT·Filed 2011·Granted Nov 15, 2011·5 cites·8 claims
- 1173US5861416ASubstituted pyrrolidin-3-yl-alkyl-piperidinesMERRELL PHARMA INC·Filed 1997·Granted Jan 19, 1999·12 cites·11 claims
- 1272US10253041B27-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds and their use as mutant IDH1 inhibitorsLILLY CO ELI·Filed 2016·Granted Apr 9, 2019·2 cites·10 claims
- 1371US11649247B27-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitorsLILLY CO ELI·Filed 2021·Granted May 16, 2023·0 cites·3 claims
- 1471US8436002B2AKT inhibitorsBEIGHT DOUGLAS WADE·Filed 2010·Granted May 7, 2013·3 cites·10 claims
- 1569US7405305B2Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitorsLILLY CO ELI·Filed 2003·Granted Jul 29, 2008·6 cites·9 claims
- 1668US11629156B27-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitorsLILLY CO ELI·Filed 2021·Granted Apr 18, 2023·0 cites·6 claims
- 1768US5430145AMercaptoacetylamide derivatives useful as inhibitors of enkephalinase and aceMERRELL DOW PHARMA·Filed 1993·Granted Jul 4, 1995·34 cites·27 claims
- 1863US5861417AHeterocyclic substituted pyrrolidine amide derivativesHOECHST MARION ROUSSEL INC·Filed 1997·Granted Jan 19, 1999·9 cites·16 claims
- 1963US5824690ASubstituted pyrrolidin-3-yl-alkyl-piperidinesHOECHST MARION ROUSSEL INC·Filed 1997·Granted Oct 20, 1998·10 cites·69 claims
- 2062US11001596B27-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitorsLILLY CO ELI·Filed 2017·Granted May 11, 2021·0 cites·8 claims
- 2161US5648366ASubstituted pyrrolidin-3-yl-alkyl-piperidinesMERRELL PHARMA INC·Filed 1995·Granted Jul 15, 1997·6 cites·15 claims
- 2260US5864045AHeterocyclic substituted piperazinone derivativesHOECHST MARION ROUSSEL INC·Filed 1998·Granted Jan 26, 1999·14 cites·14 claims
- 2358US5672602ASubstituted piperazine derivativesHOECHST MARION ROUSSEL INC·Filed 1996·Granted Sep 30, 1997·15 cites·17 claims
- 2453US5491143AMercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ACEMERRELL DOW PHARMA·Filed 1995·Granted Feb 13, 1996·4 cites·2 claims
- 2552US9062050B2Inhibitor of JAK1 and JAK2LILLY CO ELI·Filed 2013·Granted Jun 23, 2015·0 cites·6 claims
- 2651US5977139ACarboxysubstituted cyclic carboxamide derivativesHOECHST MARION ROUSSEL INC·Filed 1997·Granted Nov 2, 1999·4 cites·64 claims
- 2751US5661160ASubstituted pyrrolidin-3-yl-alkyl-piperidinesMERRELL PHARMA INC·Filed 1995·Granted Aug 26, 1997·3 cites·15 claims
- 2847US10696665B2Mutant IDH1 inhibitorsLILLY CO ELI·Filed 2017·Granted Jun 30, 2020·0 cites·15 claims
- 2947US6316445B1Carboxy substituted acylic carboxamide derivativesAVENTIS PHARMA INC·Filed 1999·Granted Nov 13, 2001·3 cites·21 claims
- 3047US2011294792A1Purine derivatives as kinase inhibitorsENGLER THOMAS ALBERT·Filed 2011·Application pending·0 cites
- 3145US6329392B1Substituted piperidines useful for the treatment of allergic diseasesAVENTIS PHARMA INC·Filed 1998·Granted Dec 11, 2001·7 cites·77 claims
- 3244US2016229835A1Novel pyridyloxyacetyl tetrahydroisoquinoline compounds useful as nampt inhibitorsLILLY CO ELI·Filed 2014·Application pending·0 cites
- 3339US5527795AMercaptoacetylamide derivatives useful as inhibitors of enkephalinase and aceMERRELL PHARMA INC·Filed 1995·Granted Jun 18, 1996·1 cites·13 claims
- 3437US6881733B1Serotonergic benzofuransLILLY CO ELI·Filed 2000·Granted Apr 19, 2005·0 cites·18 claims
- 3535US5840726AHeterocyclic substituted piperazinone derivativesHOECHST MARION ROUSSEL INC·Filed 1997·Granted Nov 24, 1998·1 cites·18 claims
- 3633US5597845ASubstituted alkyldiamine derivativesMERRELL PHARMA INC·Filed 1994·Granted Jan 28, 1997·1 cites·40 claims
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