Inventor · disambiguated record
Benjamin Littler
Also filed as: LITTLER BENJAMIN · LITTLER BENJAMIN J · LITTLER BENJAMIN JOSEPH
37 granted patents·7 pending applications·758 citations·filing 2004–2024
98Inventor score
Files withVERTEX PHARMA27BIOMED VALLEY DISCOVERIES INC6ALBANY MOLECULAR RES INC2AMBHAIKAR NARENDRA BHALCHANDRA2LORIMER KEITH2
Top patents by PatentIndex Score
44 records- 0198US10787472B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2019·Granted Sep 29, 2020·12 cites·40 claims
- 0297US11584761B2Process of making CFTR modulatorsVERTEX PHARMA·Filed 2020·Granted Feb 21, 2023·9 cites·37 claims
- 0397US9862709B2Processes for making compounds useful as inhibitors of ATR kinaseVERTEX PHARMA·Filed 2015·Granted Jan 9, 2018·16 cites·36 claims
- 0497US9828397B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2016·Granted Nov 28, 2017·23 cites·109 claims
- 0597US9035053B2Processes for making compounds useful as inhibitors of ATR kinaseVERTEX PHARMA·Filed 2012·Granted May 19, 2015·21 cites·24 claims
- 0697US8884018B2Process for preparing modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2014·Granted Nov 11, 2014·62 cites·7 claims
- 0797US8754222B2Process for preparing modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2012·Granted Jun 17, 2014·66 cites·14 claims
- 0897US8461352B2Process for preparing azabicyclic compoundsAMBHAIKAR NARENDRA BHALCHANDRA·Filed 2012·Granted Jun 11, 2013·77 cites·1 claims
- 0997US8404865B2Process for preparing azabicyclic compoundsAMBHAIKAR NARENDRA BHALCHANDRA·Filed 2010·Granted Mar 26, 2013·81 cites·20 claims
- 1097US8344147B2Process for preparing modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2010·Granted Jan 1, 2013·90 cites·24 claims
- 1196US10253054B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2017·Granted Apr 9, 2019·17 cites·38 claims
- 1296US10071979B2Process of producing cycloalkylcarboxamido-indole compoundsVERTEX PHARMA·Filed 2015·Granted Sep 11, 2018·29 cites·28 claims
- 1396US9464102B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2015·Granted Oct 11, 2016·23 cites·21 claims
- 1496US9163042B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2014·Granted Oct 20, 2015·46 cites·20 claims
- 1594US11773119B2Prodrugs of pyridone amides useful as modulators of sodium channelsVERTEX PHARMA·Filed 2020·Granted Oct 3, 2023·2 cites·20 claims
- 1694US9035072B2Process of producing cycloalkylcarboxamido-indole compoundsBELMONT DANIEL T·Filed 2011·Granted May 19, 2015·62 cites·26 claims
- 1793US12122788B2Process of making CFTR modulatorsVERTEX PHARMA·Filed 2023·Granted Oct 22, 2024·1 cites·21 claims
- 1893US9676746B2Crystalline forms of C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2016·Granted Jun 13, 2017·6 cites·82 claims
- 1993US9254291B2Modulators of ATP-binding cassette transportersVERTEX PHARMA·Filed 2012·Granted Feb 9, 2016·52 cites·11 claims
- 2093US8846686B2Compounds useful as inhibitors of ATR kinaseVERTEX PHARMA·Filed 2012·Granted Sep 30, 2014·16 cites·47 claims
- 2192US11434201B2Processes for preparing pyrrolidine compoundsVERTEX PHARMA·Filed 2018·Granted Sep 6, 2022·6 cites·22 claims
- 2290US10208027B2Processes for preparing ATR inhibitorsVERTEX PHARMA·Filed 2017·Granted Feb 19, 2019·3 cites·20 claims
- 2387US11465985B2Processes for making modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2018·Granted Oct 11, 2022·6 cites·8 claims
- 2487US10822331B2Processes for preparing ATR inhibitorsVERTEX PHARMA·Filed 2018·Granted Nov 3, 2020·2 cites·35 claims
- 2587US7825138B2Crystal forms of (3R)-1-(2-methylalanyl-D-tryptophyl)-3-(phenylmethyl)-3-piperidinecarboxylic acid 1,2,2-trimethylhydrazideHELSINN THERAPEUTICS US INC·Filed 2005·Granted Nov 2, 2010·13 cites·1 claims
- 2686US2025084059A1CRYSTALLINE FORMS OF C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2024·Application pending·0 cites
- 2782US10183927B2Crystalline forms of C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2017·Granted Jan 22, 2019·2 cites·26 claims
- 2880US12187698B2Crystalline forms of C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2022·Granted Jan 7, 2025·0 cites·10 claims
- 2980US8466173B2Crystal forms of (3R)-1-(2-methylalanyl-D-tryptophyl)-3-(phenylmethyl)-3-piperidinecarboxylic acid 1,2,2-trimethylhydrazideLORIMER KEITH·Filed 2010·Granted Jun 18, 2013·5 cites·17 claims
- 3076US12415798B2Processes for making modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2022·Granted Sep 16, 2025·0 cites·5 claims
- 3176US7498345B2Process for production of piperidine derivativesALBANY MOLECULAR RES INC·Filed 2004·Granted Mar 3, 2009·6 cites·14 claims
- 3275US7777048B2Processes for preparing biaryl ureas and analogs thereofVERTEX PHARMA·Filed 2009·Granted Aug 17, 2010·1 cites·16 claims
- 3373US10738027B2Crystalline forms of C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2018·Granted Aug 11, 2020·0 cites·10 claims
- 3472US11390600B2Crystalline forms of C21H22Cl2N4O2BIOMED VALLEY DISCOVERIES INC·Filed 2020·Granted Jul 19, 2022·0 cites·10 claims
- 3568US7498443B2Process for production of carebastineALBANY MOLECULAR RES INC·Filed 2004·Granted Mar 3, 2009·3 cites·5 claims
- 3668US2021238158A1Process of producing cycloalkylcarboxamido-indole compoundsVERTEX PHARMA·Filed 2020·Application pending·0 cites
- 3761US2014336393A1Process for preparing modulators of cystic fibrosis transmembrane conductance regulatorVERTEX PHARMA·Filed 2014·Application pending·0 cites
- 3860US2019210991A1Process of producing cycloalkylcarboxamido-indole compoundsVERTEX PHARMA·Filed 2018·Application pending·0 cites
- 3957US7544810B2Processes for preparing biaryl ureas and analogs thereofVERTEX PHARMA·Filed 2006·Granted Jun 9, 2009·0 cites·17 claims
- 4056US9975921B2Crystal forms of anamorelinHELSINN HEALTHCARE SA·Filed 2015·Granted May 22, 2018·0 cites·12 claims
- 4154US2013281701A1Crystal forms of anamorelinLORIMER KEITH·Filed 2013·Application pending·0 cites
- 4250US8067605B2Process for production of piperidine derivativesMECKLER HAROLD·Filed 2010·Granted Nov 29, 2011·0 cites·7 claims
- 4341US2016166540A1Modulators for atp-binding cassette transportersVERTEX PHARMA·Filed 2016·Application pending·0 cites
- 4434US2006047171A1Catalytic hydrogenation of nitriles to produce capsaicinoid derivatives and amine compounds, and methods for purifying and obtaining the polymorphs thereofMECKLER HAROLD·Filed 2004·Application pending·0 cites
Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →