Inventor · disambiguated record
Mark G. Bock
Also filed as: BOCK MARK · BOCK MARK G · BOCK MARK GARY
109 granted patents·30 pending applications·1,937 citations·filing 1978–2025
99Inventor score
Top patents by PatentIndex Score
139 records- 0198US5324726ABenzodiazepine analogsMERCK & CO INC·Filed 1992·Granted Jun 28, 1994·137 cites·4 claims
- 0297US4820834ABenzodiazepine analogsMERCK & CO INC·Filed 1987·Granted Apr 11, 1989·161 cites·13 claims
- 0397US4145551APyrazine-2-carbonyloxyguanidinesMERCK & CO INC·Filed 1978·Granted Mar 20, 1979·49 cites·5 claims
- 0496US5756504ATocolytic oxytocin receptor antagonistsMERCK & CO INC·Filed 1995·Granted May 26, 1998·112 cites·11 claims
- 0595US5004741AMethods of antagonizing CCK or gastrin with benzodiazepine analogsMERCK & CO INC·Filed 1988·Granted Apr 2, 1991·59 cites·15 claims
- 0695US4362724AMethod of treating edema and hypertension and pharmaceutical composition therefor in which the active ingredient comprises a novel substituted pyrazinyl-1,2,4-oxadiazole and a kaliuretic diureticMERCK & CO INC·Filed 1981·Granted Dec 7, 1982·40 cites·6 claims
- 0794US5464788ATocolytic oxytocin receptor antagonistsMERCK & CO INC·Filed 1994·Granted Nov 7, 1995·135 cites·11 claims
- 0894US4309430APyrazinyl-1,2,4-oxadiazole-5-ones, for treatment of edema, and processes for preparing sameMERCK & CO INC·Filed 1980·Granted Jan 5, 1982·53 cites·11 claims
- 0992US9938234B2PPAR agonistsSALK INST FOR BIOLOGICAL STUDI·Filed 2015·Granted Apr 10, 2018·13 cites·10 claims
- 1092US5665719ABenzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonistsMERCK & CO INC·Filed 1995·Granted Sep 9, 1997·74 cites·20 claims
- 1191US9624192B2Carbamate/urea derivativesAUBERSON YVES·Filed 2016·Granted Apr 18, 2017·11 cites·20 claims
- 1291US6436962B1Arylhydantoin derivatives and uses thereofMERCK & CO INC·Filed 2000·Granted Aug 20, 2002·34 cites·31 claims
- 1390US12012397B2Sulphonyl urea derivatives as NLRP3 inflammasome modulatorsNODTHERA LTD·Filed 2022·Granted Jun 18, 2024·1 cites·20 claims
- 1490US8163704B2Glycoside derivatives and uses thereofBEBERNITZ GREGORY RAYMOND·Filed 2010·Granted Apr 24, 2012·15 cites·72 claims
- 1590US4454132APharmaceutical compositions of novel substituted pyrazinyl-1,2,4-oxadiazoles useful in the treatment of edema and hypertensionMERCK & CO INC·Filed 1982·Granted Jun 12, 1984·22 cites·4 claims
- 1689US8263635B2Inhibitors of CYP 17BOCK MARK G·Filed 2010·Granted Sep 11, 2012·17 cites·16 claims
- 1789US5166151A2-Benzazepines with 5- and 6-membered heterocyclic rings, compositions and medical methods of use thereofMERCK & CO INC·Filed 1991·Granted Nov 24, 1992·41 cites·16 claims
- 1889US4628084AProcess for 3-acylamino benzodiazepinesMERCK & CO INC·Filed 1986·Granted Dec 9, 1986·28 cites·5 claims
- 1988US11518757B2Sulphonyl urea derivatives as NLRP3 inflammasome modulatorsNODTHERA LTD·Filed 2018·Granted Dec 6, 2022·4 cites·21 claims
- 2088US4755508ABenzodiazepine analogs and use as antogonists of gastrin and cholecystokininMERCK & CO INC·Filed 1987·Granted Jul 5, 1988·49 cites·9 claims
- 2187US9034874B2Carbamate/urea derivativesAUBERSON YVES·Filed 2013·Granted May 19, 2015·12 cites·20 claims
- 2287US5175159A3-substituted-1,4-benzodiazepines as oxytocin antagonistsMERCK & CO INC·Filed 1990·Granted Dec 29, 1992·36 cites·7 claims
- 2386US8722633B2Glycoside derivatives and uses thereofBEBERNITZ GREGORY RAYMOND·Filed 2012·Granted May 13, 2014·9 cites·18 claims
- 2486US5834464AImidazolinobenzodiazepinesMERCK & CO INC·Filed 1994·Granted Nov 10, 1998·29 cites·6 claims
- 2586US5206234ABenzolactam analogs as antagonists of cckMERCK & CO INC·Filed 1991·Granted Apr 27, 1993·61 cites·34 claims
- 2686US4309540ASubstituted pyrazinyl-1,2,4-oxadiazolesMERCK & CO INC·Filed 1980·Granted Jan 5, 1982·28 cites·8 claims
- 2785US9796683B2Tetrasubstituted alkene compounds and their useEISAI R&D MAN CO LTD·Filed 2016·Granted Oct 24, 2017·6 cites·32 claims
- 2885US8828951B2Glycoside derivatives and uses thereofBEBERNITZ GREGORY RAYMOND·Filed 2012·Granted Sep 9, 2014·7 cites·22 claims
- 2985US5220018ACholecystokinin antagonistsMERCK & CO INC·Filed 1992·Granted Jun 15, 1993·29 cites·8 claims
- 3085US4554272ASubstituted quinazolino-1,4-benzodiazepin-6,9-diones and their preparationMERCK & CO INC·Filed 1985·Granted Nov 19, 1985·20 cites·11 claims
- 3184US8466114B2Glycoside derivatives and uses thereofBEBERNITZ GREGORY RAYMOND·Filed 2012·Granted Jun 18, 2013·6 cites·22 claims
- 3284US5597915ABenzodiazepine derivatives, compositions containing them and their use in therapyMERCK SHARP & DOHME·Filed 1993·Granted Jan 28, 1997·51 cites·4 claims
- 3383US5177071A1,4-benzodiazepines with 6-membered heterocyclic rings to treat panic and anxiety disorderMERCK & CO INC·Filed 1991·Granted Jan 5, 1993·47 cites·3 claims
- 3483US4847248A1,4-Benzodiazepines with 5- and 6-membered heterocyclic rings and their use as cholecystokinins and gastrin antagonistsMERCK & CO INC·Filed 1988·Granted Jul 11, 1989·19 cites·12 claims
- 3583US4636491ARenin inhibitory peptides having improved solubilityMERCK & CO INC·Filed 1984·Granted Jan 13, 1987·26 cites·4 claims
- 3682US12459925B2Sulphonyl urea derivatives as NLRP3 inflammasome modulatorsNODTHERA LTD·Filed 2024·Granted Nov 4, 2025·0 cites·20 claims
- 3782US9273026B2Carbamate/urea derivativesAUBERSON YVES·Filed 2015·Granted Mar 1, 2016·4 cites·24 claims
- 3881US6919343B2N-biphenyl(substituted methyl) aminocycloalkane-carboxamide derivativesMERCK & CO INC·Filed 2003·Granted Jul 19, 2005·14 cites·40 claims
- 3981US4663321ATriazolobenzodiazepines and pharmaceutical useMERCK & CO INC·Filed 1985·Granted May 5, 1987·17 cites·12 claims
- 4079US5220017ACholecystokinin antagonistsMERCK & CO INC·Filed 1992·Granted Jun 15, 1993·36 cites·2 claims
- 4178US9029399B217α-hydroxylase/C17,20-lyase inhibitorsBOCK MARK GARY·Filed 2012·Granted May 12, 2015·4 cites·17 claims
- 4277US8946260B217α-hydroxylase/C17,20-lyase inhibitorsBOCK MARK GARY·Filed 2011·Granted Feb 3, 2015·2 cites·9 claims
- 4376US4479941ARenin inhibitory peptides having PHE13 delectionMERCK & CO INC·Filed 1982·Granted Oct 30, 1984·33 cites·8 claims
- 4475US9227969B2Compounds and compositions as inhibitors of MEKBOCK MARK GARY·Filed 2014·Granted Jan 5, 2016·2 cites·16 claims
- 4574US10550071B2PPAR agonistsSALK INST FOR BIOLOGICAL STUDI·Filed 2018·Granted Feb 4, 2020·1 cites·18 claims
- 4674US6908921B2Quinoxalinone derivatives as bradykinin B1 antagonistsMERCK & CO INC·Filed 2003·Granted Jun 21, 2005·7 cites·19 claims
- 4774US4724237A2-substituted-aminomethyl-1,4-benzodiazepinesMERCK & CO INC·Filed 1984·Granted Feb 9, 1988·8 cites·9 claims
- 4871USRE45173EInhibitors of CYP 17NOVARTIS AG·Filed 2013·Granted Sep 30, 2014·2 cites·21 claims
- 4971US5204349AAmide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonistsMERCK & CO INC·Filed 1991·Granted Apr 20, 1993·14 cites·6 claims
- 5071US4487963AEnantioselective synthesis of 4-amino-3-hydroxy-2,4-(disubstituted)pentanoic acidMERCK & CO INC·Filed 1983·Granted Dec 11, 1984·7 cites·1 claims
Showing the top 50 of 139 patent records by PatentIndex Score.
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