Inventor · disambiguated record
Roland E. Dolle
Also filed as: DOLLE III ROLAND E · DOLLE III ROLAND ELLWOOD · DOLLE ROLAND · DOLLE ROLAND E
87 granted patents·33 pending applications·1,258 citations·filing 1992–2025
99Inventor score
Top patents by PatentIndex Score
120 records- 0194US7087749B2Substituted piperidine compounds and methods of their useADOLOR CORP·Filed 2004·Granted Aug 8, 2006·36 cites·34 claims
- 0294US6432947B1N-heterocyclic derivatives as NOS inhibitorsBERLEX LAB·Filed 1999·Granted Aug 13, 2002·89 cites·34 claims
- 0391US7884102B2Substituted piperidine compounds and methods of their useADOLOR CORP·Filed 2008·Granted Feb 8, 2011·15 cites·55 claims
- 0491US6992090B2Substituted piperidine compounds and methods of their useADOLOR CORP·Filed 2003·Granted Jan 31, 2006·37 cites·27 claims
- 0590US5552400AFused-bicyclic lactams as interleukin-1β converting enzyme inhibitorsSTERLING WINTHROP INC·Filed 1994·Granted Sep 3, 1996·70 cites·10 claims
- 0690US5447954APhenylderivate as inhibitors of ATP citrate lyaseSMITHKLINE BEECHAM PLC·Filed 1992·Granted Sep 5, 1995·111 cites·10 claims
- 0789US7767814B2Substituted piperidine compounds and methods of their useADOLOR CORP·Filed 2006·Granted Aug 3, 2010·5 cites·62 claims
- 0889US7338962B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2004·Granted Mar 4, 2008·19 cites·5 claims
- 0989US5462939APeptidic ketones as interleukin-1β-converting enzyme inhibitorsSTERLING WINTHROP INC·Filed 1993·Granted Oct 31, 1995·70 cites·15 claims
- 1088US6794510B2Processes for the preparation of peripheral opioid antagonist compounds and intermediates theretoADOLOR CORP·Filed 2002·Granted Sep 21, 2004·16 cites·14 claims
- 1188US5972719ACombinatorial hydroxy-amino acid amide librariesPHARMACOPEIA INC·Filed 1996·Granted Oct 26, 1999·39 cites·14 claims
- 1287US7638527B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2007·Granted Dec 29, 2009·5 cites·26 claims
- 1387US7544676B2Sulfamoyl benzamides and methods of their useADOLOR CORP·Filed 2006·Granted Jun 9, 2009·18 cites·74 claims
- 1487US5585357AHeteroaryloxymethyl ketones as interleukin-1βconverting enzyme inhibitorsSANOFI WINTHROP INC·Filed 1996·Granted Dec 17, 1996·69 cites·24 claims
- 1586US7598261B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2006·Granted Oct 6, 2009·7 cites·93 claims
- 1686US5976894ACombinatorial amide alcohol librariesPHARMACOPEIA INC·Filed 1997·Granted Nov 2, 1999·46 cites·19 claims
- 1785US5892038AHydroxy-amino acid amidesPHARMACOPEIA INC·Filed 1997·Granted Apr 6, 1999·28 cites·3 claims
- 1884US8278323B2Opioid antagonistsDOLLE ROLAND E·Filed 2009·Granted Oct 2, 2012·2 cites·32 claims
- 1984US7671052B2Phenyl derivatives and methods of useADOLOR CORP·Filed 2005·Granted Mar 2, 2010·12 cites·73 claims
- 2083US8969570B2Beta-lactamase inhibitorsCUBIST PHARM INC·Filed 2013·Granted Mar 3, 2015·3 cites·15 claims
- 2183US7297796B2Sulfamoyl benzamide derivatives and methods of their useADOLOR CORP·Filed 2005·Granted Nov 20, 2007·7 cites·135 claims
- 2283US5872262AHydroxy-amino acid amidesPHARMACOPEIA INC·Filed 1997·Granted Feb 16, 1999·48 cites·7 claims
- 2382US8580788B2Opioid antagonistsDOLLE ROLAND E·Filed 2012·Granted Nov 12, 2013·2 cites·18 claims
- 2482US7538110B2Opioid antagonistsADOLOR CORP·Filed 2006·Granted May 26, 2009·4 cites·90 claims
- 2581US7820827B2Substituted piperidine compounds and methods of their useADOLOR CORP·Filed 2005·Granted Oct 26, 2010·3 cites·18 claims
- 2681US5948696ACombinatorial biaryl amino acid amide librariesPHARMACOPEIA INC·Filed 1997·Granted Sep 7, 1999·42 cites·10 claims
- 2781US5670494AN-(pyrimidinyl)-aspartic acid analogs as interleukin-1β converting enzyme inhibitorsSANOFT·Filed 1995·Granted Sep 23, 1997·49 cites·2 claims
- 2881US5622967AQuinolone carboxamide Calpain inhibitorsSTERLING WINTHROP INC·Filed 1995·Granted Apr 22, 1997·34 cites·16 claims
- 2981US5565430AAzaaspartic acid analogs as interleukin-1β converting enzyme inhibitorsSTERLING WINTHROP INC·Filed 1994·Granted Oct 15, 1996·41 cites·9 claims
- 3080US7906646B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2009·Granted Mar 15, 2011·2 cites·4 claims
- 3179US7576207B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2007·Granted Aug 18, 2009·3 cites·62 claims
- 3278US7381721B2Substituted piperidine compoundsADOLOR CORP·Filed 2003·Granted Jun 3, 2008·9 cites·37 claims
- 3378US7091354B2Processes for the preparation of peripheral opioid antagonist compounds and intermediates theretoADOLOR CORP·Filed 2004·Granted Aug 15, 2006·7 cites·11 claims
- 3478US6747031B2N-heterocyclic derivatives as NOS inhibitorsBERLEX LAB·Filed 2002·Granted Jun 8, 2004·6 cites·10 claims
- 3577US8071611B2Spirocyclic heterocyclic derivatives and methods of their useDOLLE ROLAND E·Filed 2010·Granted Dec 6, 2011·2 cites·16 claims
- 3676US5639745AFused-bicyclic lactams as interleukin-1β converting enzyme inhibitorsSANOFI SA·Filed 1995·Granted Jun 17, 1997·37 cites·33 claims
- 3776US5585486APeptidic ketones as interleukin-1β-converting enzyme inhibitorsSTERLING WINTHROP INC·Filed 1995·Granted Dec 17, 1996·36 cites·2 claims
- 3876US2009233959A1Beloxepin and analogs for the treatment of painADOLOR CORP·Filed 2009·Application pending·0 cites
- 3974US8022060B2Spirocyclic heterocyclic derivatives and methods of their useADOLOR CORP·Filed 2009·Granted Sep 20, 2011·1 cites·206 claims
- 4073US6670473B2N-heterocyclic derivatives as NOS inhibitorsBERLEX LAB·Filed 2002·Granted Dec 30, 2003·3 cites·8 claims
- 4172US6162800AN-(pyrimidinyl)-aspartic acid analogs as interleukin-1β converting enzyme inhibitorsVERTEX PHARMA·Filed 1997·Granted Dec 19, 2000·25 cites·7 claims
- 4272US2025145652A1Inorganic salts of nicotinamide mononucleotide as anti-aging agentsLIFE BIOSCIENCES INC·Filed 2024·Application pending·0 cites
- 4372US2024207212A1Methods and compositions for treating inflammationUNIV MASSACHUSETTS·Filed 2023·Application pending·0 cites
- 4471US10654883B2Inorganic salts of nicotinic acid mononucleotide as anti-aging agentsJumpstart Fertility Pty Ltd·Filed 2019·Granted May 19, 2020·1 cites·6 claims
- 4571US8895560B2Opioid antagonistsADOLOR CORP·Filed 2014·Granted Nov 25, 2014·0 cites·6 claims
- 4671US5734054AHydroxy-amino acid amidesPHARMACOPEIA INC·Filed 1996·Granted Mar 31, 1998·29 cites·7 claims
- 4770US6900213B2Bisaryl derivatives having FSH modulatory activityPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted May 31, 2005·5 cites·13 claims
- 4870US6841674B2N-heterocyclic derivatives as NOS inhibitorsBERLEX LAB·Filed 2002·Granted Jan 11, 2005·2 cites·6 claims
- 4970US5843905APeptidic phosphinyloxymethyl ketones as interleukin-1β-converting enzyme inhibitorsVERTEX PHARMA·Filed 1996·Granted Dec 1, 1998·15 cites·8 claims
- 5069US6407080B2N-(pyrimidinyl)-aspartic acid analogs as interleukin-1β converting enzyme inhibitorsVERTEX PHARMA·Filed 2000·Granted Jun 18, 2002·3 cites·5 claims
Showing the top 50 of 120 patent records by PatentIndex Score.
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