Inventor · disambiguated record
Bernard R. Neustadt
Also filed as: GOLD ELIJAH H · NEUSTADT BERNARD · NEUSTADT BERNARD R
77 granted patents·11 pending applications·1,883 citations·filing 1976–2014
99Inventor score
Files withSCHERING CORP69HARRIS JOEL M6NEELAMKAVIL SANTHOSH FRANCIS5NEUSTADT BERNARD R3BOYLE CRAIG D2
Top patents by PatentIndex Score
88 records- 0199US4929641AMercapto-acylamino acid antihypertensivesSCHERING CORP·Filed 1988·Granted May 29, 1990·164 cites·20 claims
- 0298US6329395B1Neuropeptide Y5 receptor antagonistsSCHERING CORP·Filed 1999·Granted Dec 11, 2001·186 cites·9 claims
- 0398US4587258AAngiotensin-converting enzyme inhibitorsSCHERING CORP·Filed 1984·Granted May 6, 1986·197 cites·30 claims
- 0497US6689765B2Piperazine derivatives useful as CCR5 antagonistsSCHERING CORP·Filed 2002·Granted Feb 10, 2004·71 cites·12 claims
- 0597US6391865B1Piperazine derivatives useful as CCR5 antagonistsSCHERING CORP·Filed 2000·Granted May 21, 2002·94 cites·19 claims
- 0695US6387930B1Piperidine derivatives useful as CCR5 antagonistsSCHERING CORP·Filed 2000·Granted May 14, 2002·76 cites·13 claims
- 0794US6630475B2Adenosine A2a receptor antagonistsSCHERING CORP·Filed 2001·Granted Oct 7, 2003·53 cites·17 claims
- 0894US4879309AMercapto-acylamino acids as antihypertensivesSCHERING CORP·Filed 1989·Granted Nov 7, 1989·43 cites·16 claims
- 0994US4818749ACarboxyalkyl dipeptides and medical use thereof in treating hypertension and congestive heart failureSCHERING CORP·Filed 1987·Granted Apr 4, 1989·73 cites·21 claims
- 1094US4808573ACarboxyalkyl dipeptides and anti-hypertensive use thereofSCHERING CORP·Filed 1987·Granted Feb 28, 1989·71 cites·14 claims
- 1193US4093742AAnti-hypertensive polyhaloisopropyl-substituted arylureasSCHERING CORP·Filed 1976·Granted Jun 6, 1978·20 cites·20 claims
- 1292US5208236AN-(acylaminomethyl)glutaryl amino acids and useSCHERING CORP·Filed 1992·Granted May 4, 1993·38 cites·11 claims
- 1391US5393755APolycyclic guanine derivativesSCHERING CORP·Filed 1991·Granted Feb 28, 1995·117 cites·13 claims
- 1491US4230635ASubstituted 4'-polyhaloisopropylsulfonanilidesSCHERING CORP·Filed 1978·Granted Oct 28, 1980·22 cites·18 claims
- 1590US4199597AOmega-(4-polyfluoro-2-hydroxy-2-propyl)-2,3,6-substituted-phenoxy and phenylthio)alkanoic acids and compounds related theretoSCHERING CORP·Filed 1979·Granted Apr 22, 1980·22 cites·15 claims
- 1687US6897217B22-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonistsSCHERING CORP·Filed 2004·Granted May 24, 2005·25 cites·21 claims
- 1785US6602885B2Piperidine derivatives useful as CCR5 antagonistsSCHERING CORP·Filed 2001·Granted Aug 5, 2003·21 cites·17 claims
- 1885US4470972A7-Carboxyalkylaminoacyl-1,4-dithia-7-azaspiro[4.4]-nonane-8-carboxylic acidsSCHERING CORP·Filed 1982·Granted Sep 11, 1984·46 cites·29 claims
- 1985US4058612A6-(Polyhaloisopropyl)quinazoline-2,4-dionesSCHERING CORP·Filed 1976·Granted Nov 15, 1977·12 cites·12 claims
- 2083US8815876B2Bicyclic heterocycle derivatives and methods of use thereofNEELAMKAVIL SANTHOSH FRANCIS·Filed 2009·Granted Aug 26, 2014·7 cites·16 claims
- 2183US5061710AMercapto-acylamino acid antihypertensivesSCHERING CORP·Filed 1987·Granted Oct 29, 1991·34 cites·4 claims
- 2282US6875772B2[1,2,4]-Triazole bicyclic adeonsine A2a receptor antagonistsSCHERING CORP·Filed 2002·Granted Apr 5, 2005·16 cites·11 claims
- 2382US4379166AArylmethoxy-, arylmethylthio-, heteroarylmethoxy-, and heteroarylmethylthio-alkylaminoalcoholsSCHERING CORP·Filed 1981·Granted Apr 5, 1983·16 cites·14 claims
- 2482US4267193AN-substituted-4-(polyfluoro-2-hydroxy-2-propyl)anilines and compounds related theretoSCHERING CORP·Filed 1979·Granted May 12, 1981·13 cites·7 claims
- 2581US5298492ADiamino acid derivatives as antihypertensivesSCHERING CORP·Filed 1992·Granted Mar 29, 1994·45 cites·11 claims
- 2681US4831157APreparation of angiotensin-converting enzyme inhibitorsSCHERING CORP·Filed 1988·Granted May 16, 1989·24 cites·1 claims
- 2780US7368449B22-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonistsSCHERING CORP·Filed 2005·Granted May 6, 2008·4 cites·16 claims
- 2879US7041666B2Adenosine A2a receptor antagonistsSCHERING CORP·Filed 2002·Granted May 9, 2006·13 cites·8 claims
- 2978US7465740B22-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonistsSCHERING CORP·Filed 2006·Granted Dec 16, 2008·3 cites·17 claims
- 3078US7384944B2Piperazine derivatives useful as CCR5 antagonistsSCHERING CORP·Filed 2003·Granted Jun 10, 2008·6 cites·18 claims
- 3178US6204282B1Benzimidazole compounds that are vitronectin receptor antagonistsSCHERING CORP·Filed 1999·Granted Mar 20, 2001·22 cites·22 claims
- 3277US8435994B2Substituted [1,2,4]triazolo[4,3-alpha]quinoxalines as adenosine A2a receptor antagonistsHARRIS JOEL M·Filed 2010·Granted May 7, 2013·3 cites·2 claims
- 3377US5075302AMercaptoacyl aminolactam endopeptidase inhibitorsSCHERING CORP·Filed 1990·Granted Dec 24, 1991·37 cites·10 claims
- 3476US8318751B2Pyrimidinone derivatives and methods of use thereofBOYLE CRAIG D·Filed 2008·Granted Nov 27, 2012·3 cites·42 claims
- 3574US7709492B2Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonistsSCHERING CORP·Filed 2005·Granted May 4, 2010·2 cites·20 claims
- 3674US7078408B2[1,2,4]-Triazole bicyclic adenosine A2a receptor antagonistsSCHERING CORP·Filed 2004·Granted Jul 18, 2006·6 cites·9 claims
- 3774US6897216B2Adenosine A2a receptor antagonistsSCHERING CORP·Filed 2003·Granted May 24, 2005·5 cites·6 claims
- 3874US6228985B1Derivatives of aminobenzoic and aminobiphenylcarboxylic acids useful as anti-cancer agentsSCHERING CORP·Filed 1998·Granted May 8, 2001·19 cites·9 claims
- 3972USRE44205EAdenosine A2a receptor antagonistsNEUSTADT BERNARD R·Filed 2012·Granted May 7, 2013·2 cites·21 claims
- 4072US7741318B2Pyrazolo [1,5-A]pyrimidine adenosine A2a receptor antagonistsSCHERING CORP·Filed 2005·Granted Jun 22, 2010·2 cites·20 claims
- 4172US7067655B2Adenosine A2a receptor antagonistsSCHERING CORP·Filed 2004·Granted Jun 27, 2006·4 cites·3 claims
- 4272US4103018A2-[4-(Polyhalo-2-hydroxy-2-propyl)anilino]-2-oxazolin-4-ones and thiazolin-4-ones corresponding theretoSCHERING CORP·Filed 1976·Granted Jul 25, 1978·8 cites·10 claims
- 4371US9440952B2Compounds inhibiting leucine-rich repeat kinase enzyme activityMERCK SHARP & DOHME·Filed 2014·Granted Sep 13, 2016·1 cites·19 claims
- 4471US8822480B2Bicyclic heterocycle derivatives and use thereof as GPR119 modulatorsNEELAMKAVIL SANTHOSH FRANCIS·Filed 2009·Granted Sep 2, 2014·1 cites·19 claims
- 4571US8415353B2Amino-quinoxaline and amino-quinoline compounds for use as adenosine A2a receptor antagonistsHARRIS JOEL M·Filed 2009·Granted Apr 9, 2013·1 cites·7 claims
- 4671US5232920AN-(mercaptoalkyl)amidesSCHERING CORP·Filed 1990·Granted Aug 3, 1993·24 cites·8 claims
- 4769US4304790A2-(Alkylthio, alkylsulfinyl or alkylsulfonyl)-4-[2-anilinoalkylamino)-1-hydroxyethyl]phenols and derivatives thereofSCHERING CORP·Filed 1979·Granted Dec 8, 1981·5 cites·13 claims
- 4869US4081547APara-polyfluoroisopropyl-anilino-2-oxazoline compounds, pharmaceutical compositions and method of treating hypertensionSCHERING CORP·Filed 1976·Granted Mar 28, 1978·4 cites·18 claims
- 4968US4511569ATricyclic lactams and derivatives useful in increasing cardiac contractilitySCHERING CORP·Filed 1982·Granted Apr 16, 1985·10 cites·19 claims
- 5067US4801609AMercapto-acylamino acid antihypertensivesSCHERING CORP·Filed 1987·Granted Jan 31, 1989·33 cites·17 claims
Showing the top 50 of 88 patent records by PatentIndex Score.
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