Inventor · disambiguated record
Henricus Jacobus Maria Gijsen
Also filed as: GIJSEN HENRICUS J M · GIJSEN HENRICUS JACOBUS MARIA
39 granted patents·11 pending applications·121 citations·filing 1999–2018
96Inventor score
Files withJANSSEN PHARMACEUTICA NV28GIJSEN HENRICUS JACOBUS MARIA7TRABANCO-SUÁREZ ANDRÉS AVELINO2BERTHELOT DIDIER JEAN-CALUDE1BOSMANS JEAN-PAUL RENE MARIE ANDRE1
Top patents by PatentIndex Score
50 records- 0194US9453002B2Substituted imidazoles as N-type calcium channel blockersJANSSEN PHARMACEUTICA NV·Filed 2013·Granted Sep 27, 2016·18 cites·24 claims
- 0284US6544997B14-(aminomethyl)-piperidine benzamides for treating gastrointestinal disordersJANSSEN PHARMACEUTICA NV·Filed 1999·Granted Apr 8, 2003·60 cites·9 claims
- 0381US8546440B2Substituted bicyclic imidazole derivatives as gamma secretase modulatorsGIJSEN HENRICUS JACOBUS MARIA·Filed 2009·Granted Oct 1, 2013·5 cites·13 claims
- 0478US9284303B2Benzimidazole cannabinoid agonists bearing a substituted heterocyclic groupJANSSEN PHARMACEUTICA NV·Filed 2013·Granted Mar 15, 2016·4 cites·7 claims
- 0576US8461145B2Dibenzoazepine and dibenzooxazepine TRPA1 agonistsGIJSEN HENRICUS JACOBUS MARIA·Filed 2008·Granted Jun 11, 2013·3 cites·11 claims
- 0675US8614201B2Heterocyclic amides as modulators of TRPA1BERTHELOT DIDIER JEAN-CALUDE·Filed 2010·Granted Dec 24, 2013·6 cites·17 claims
- 0774US9751886B24-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)JANSSEN PHARMACEUTICA NV·Filed 2014·Granted Sep 5, 2017·2 cites·13 claims
- 0873US9974775B2Substituted imidazoles as N-type calcium channel blockersJANSSEN PHARMACEUTICA NV·Filed 2016·Granted May 22, 2018·1 cites·16 claims
- 0973US7652040B2Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT4-antagonistsJANSSEN PHARMACEUTICA NV·Filed 2004·Granted Jan 26, 2010·5 cites·10 claims
- 1070US9828350B25,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (BACE)JANSSEN PHARMACEUTICA NV·Filed 2016·Granted Nov 28, 2017·1 cites·4 claims
- 1170US8772504B2Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulatorsGIJSEN HENRICUS JACOBUS MARIA·Filed 2010·Granted Jul 8, 2014·2 cites·12 claims
- 1269US9834559B24-Amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase (BACE)JANSSEN PHARMACEUTICA NV·Filed 2014·Granted Dec 5, 2017·1 cites·10 claims
- 1369US7205410B24-(aminomethyl)-piperidine benzamides for treating gastrointestinal disordersJANSSEN PHARMACEUTICA NV·Filed 2003·Granted Apr 17, 2007·4 cites·1 claims
- 1468US9115143B2Substituted indole derivatives as gamma secretase modulatorsMINNE GARRETT BERLOND·Filed 2012·Granted Aug 25, 2015·3 cites·14 claims
- 1567US9181245B2Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's diseaseJANSSEN PHARMACEUTICALS INC·Filed 2013·Granted Nov 10, 2015·1 cites·14 claims
- 1667US8946266B2Substituted triazole and imidazole derivatives as gamma secretase modulatorsWU TONGFEI·Filed 2010·Granted Feb 3, 2015·2 cites·14 claims
- 1765US10653673B2Substituted imidazoles as N-type calcium channel blockersJANSSEN PHARMACEUTICA NV·Filed 2018·Granted May 19, 2020·0 cites·16 claims
- 1865US7635706B25HT4-antagonistic 4-(aminomethyl)-piperidine benzamidesJANSSEN PHARMACEUTICA NV·Filed 2004·Granted Dec 22, 2009·2 cites·8 claims
- 1964US10106524B22,3,4,5-tetrahydropyridin-6-amine and 3,4-dihydro-2H-pyrrol-5-amine compound inhibitors of beta-secretaseJANSSEN PHARMACEUTICA NV·Filed 2015·Granted Oct 23, 2018·1 cites·16 claims
- 2061US8334304B2Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT4-antagonistsBOSMANS JEAN-PAUL RENE MARIE ANDRE·Filed 2009·Granted Dec 18, 2012·0 cites·8 claims
- 2152US8524757B2Benzimidazole cannabinoid agonists bearing a substituted heterocyclic groupGIJSEN HENRICUS JACOBUS MARIA·Filed 2007·Granted Sep 3, 2013·0 cites·11 claims
- 2252US2015094311A1Novel substituted bicyclic heterocyclic compounds as gamma secretase modulatorsCELLZOME LTD·Filed 2014·Application pending·0 cites
- 2351US2011124666A13,4-dihydropyrimidine trpa1 antagonistsJANSSEN PHARMACEUTICA NV A CORP·Filed 2009·Application pending·0 cites
- 2449US8193369B2Benzimidazole cannabinoid agonistsGIJSEN HENRICUS JACOBUS MARIA·Filed 2008·Granted Jun 5, 2012·0 cites·8 claims
- 2548US10562897B2Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulatorsJANSSEN PHARMACEUTICA NV·Filed 2018·Granted Feb 18, 2020·0 cites·11 claims
- 2647US7732464B2Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT4-antagonistsJANSSEN PHARMACEUTICA NV·Filed 2004·Granted Jun 8, 2010·0 cites·10 claims
- 2747US7638535B24-(aminomethyl)-piperidine benzamides as 5HT4-antagonistsJANSSEN PHARMACEUTICA NV·Filed 2004·Granted Dec 29, 2009·0 cites·9 claims
- 2847US7498347B2Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT4 antagonistsJANSSEN PHARMACEUTICA NV·Filed 2004·Granted Mar 3, 2009·0 cites·9 claims
- 2946US2010273831A1Fluoro alkyl substituted benzimidazole cannabinoid agonistsGIJSEN HENRICUS JACOBUS MARIA·Filed 2008·Application pending·0 cites
- 3045US9580433B24-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)JANSSEN PHARMACEUTICA NV·Filed 2014·Granted Feb 28, 2017·0 cites·15 claims
- 3144US10112943B2Substituted imidazoles as gamma secretase modulatorsJANSSEN PHARMACEUTICA NV·Filed 2013·Granted Oct 30, 2018·0 cites·14 claims
- 3243US8946426B2Substituted bicyclic heterocyclic compounds as gamma secretase modulatorsGIJSEN HENRICUS JACOBUS MARIA·Filed 2010·Granted Feb 3, 2015·0 cites·9 claims
- 3342US10246454B2Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulatorsJANSSEN PHARMACEUTICA NV·Filed 2014·Granted Apr 2, 2019·0 cites·11 claims
- 3442US9079886B2Substituted triazole derivatives as gamma secretase modulatorsVAN BRANDT SVEN FRANCISCUS ANNA·Filed 2011·Granted Jul 14, 2015·0 cites·12 claims
- 3542US2014343048A16-difluoromethyl-5,6-dihydro-2h-[1,4]oxazin-3-amine derivativesJanssen Pharmacetuica NV·Filed 2012·Application pending·0 cites
- 3642US2021284659A1Inhibitors of beta secretaseJANSSEN PHARMACEUTICA NV·Filed 2018·Application pending·0 cites
- 3742US2014364428A15-(3-aminophenyl)-5-alkyl-5,6-dihydro-2h-[1,4]oxazin-3-amine derivativesJANSSEN PHARMACEUTICA NV·Filed 2012·Application pending·0 cites
- 3841US11053248B2[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitorsJANSSEN PHARMACEUTICA NV·Filed 2017·Granted Jul 6, 2021·0 cites·9 claims
- 3941US10947239B2[1,2,4]triazolo[1,5-a]pyrimidin-7-yl compoundJANSSEN PHARMACEUTICA NV·Filed 2016·Granted Mar 16, 2021·0 cites·11 claims
- 4041US9145399B2Substituted bicyclic triazole derivatives as gamma secretase modulatorsDE CLEYN MICHEL ANNA JOZEF·Filed 2011·Granted Sep 29, 2015·0 cites·4 claims
- 4141US2019389882A1Inhibitors of beta secretaseJANSSEN PHARMACEUTICA NV·Filed 2018·Application pending·0 cites
- 4241US2013109683A15,6-dihydro-2h-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (bace)TRABANCO-SUAREZ ANDRES AVELINO·Filed 2011·Application pending·0 cites
- 4341US2020010482A1Inhibitors of beta secretaseJANSSEN PHARMACEUTICA NV·Filed 2018·Application pending·0 cites
- 4440US11319321B2[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitorsJANSSEN PHARMACEUTICA NV·Filed 2017·Granted May 3, 2022·0 cites·6 claims
- 4540US2006216749A1Chimeric gaba receptorSMANS KARINE ALFONSINE A·Filed 2004·Application pending·0 cites
- 4639US2018334447A12,3,4,5-tetrahydropyridin-6-amine derivativesJANSSEN PHARMACEUTICA NV·Filed 2016·Application pending·0 cites
- 4736US10947242B2[1,2,4]triazolo[1,5and#8208;A]pyrimidine compounds as PDE2 inhibitorsJANSSEN PHARMACEUTICA NV·Filed 2017·Granted Mar 16, 2021·0 cites·13 claims
- 4836US9346811B26,7-dihydro-pyrazolo[1,5-a]pyrazin-4-ylamine derivatives useful as inhibitors of beta-secretase (BACE)TRABANCO-SUÁREZ ANDRÉS AVELINO·Filed 2012·Granted May 24, 2016·0 cites·12 claims
- 4935US9840507B25,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine derivatives useful as inhibitors of beta-secretase (BACE)TRABANCO-SUÁREZ ANDRÉS AVELINO·Filed 2011·Granted Dec 12, 2017·0 cites·7 claims
- 5027US8835482B2Substituted indazole and aza-indazole derivatives as gamma secretase modulatorsBischoff François Paul·Filed 2010·Granted Sep 16, 2014·0 cites·10 claims
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