Inventor · disambiguated record
Sacha Holland
Also filed as: HOLLAND SACHA · HOLLAND SACHA J
90 granted patents·11 pending applications·2,391 citations·filing 1997–2021
99Inventor score
Files withRIGEL PHARMACEUTICALS INC74SINGH RAJINDER12GOFF DANE7DING PINGYU2MOUNT SINAI HOSPITAL CORP2
Top patents by PatentIndex Score
101 records- 0199US8853397B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2013·Granted Oct 7, 2014·45 cites·7 claims
- 0299US8835430B22,4-pyrimidinediamine compounds and their usesSINGH RAJINDER·Filed 2013·Granted Sep 16, 2014·48 cites·16 claims
- 0399US8822685B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2013·Granted Sep 2, 2014·43 cites·17 claims
- 0499US7820819B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2006·Granted Oct 26, 2010·87 cites·17 claims
- 0599US7655797B2Intermediates for making 2,4-pyrimidinediamine compoundsRIGEL PHARMACEUTICALS INC·Filed 2008·Granted Feb 2, 2010·81 cites·21 claims
- 0699US7642351B22,4-Pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2006·Granted Jan 5, 2010·105 cites·14 claims
- 0799US7589200B25-Fluoro-4N-phenyl-4-pyrimidineamine compoundsRIGEL PHARMACEUTICALS INC·Filed 2004·Granted Sep 15, 2009·102 cites·18 claims
- 0899US7557210B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2003·Granted Jul 7, 2009·190 cites·16 claims
- 0999US7550460B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2007·Granted Jun 23, 2009·95 cites·18 claims
- 1099US7498435B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2006·Granted Mar 3, 2009·93 cites·21 claims
- 1199US7485724B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2006·Granted Feb 3, 2009·119 cites·20 claims
- 1299US7435814B22,4-Pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2005·Granted Oct 14, 2008·94 cites·11 claims
- 1399US7332484B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2005·Granted Feb 19, 2008·146 cites·4 claims
- 1499US7329672B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2005·Granted Feb 12, 2008·130 cites·19 claims
- 1599US7329671B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2005·Granted Feb 12, 2008·147 cites·19 claims
- 1699US7060827B2Intermediates useful for making 2,4-pyrimidinediamine compoundsRIGEL PHARMACEUTICALS INC·Filed 2004·Granted Jun 13, 2006·255 cites·11 claims
- 1798US8389557B2Triazole derivatives useful as Axl inhibitorsSINGH RAJINDER·Filed 2010·Granted Mar 5, 2013·73 cites·6 claims
- 1896US9913842B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2016·Granted Mar 13, 2018·8 cites·28 claims
- 1996US7709482B2Polycyclic heteroaryl substituted triazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2007·Granted May 4, 2010·34 cites·62 claims
- 2095US9133133B22,4-pyridinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2014·Granted Sep 15, 2015·10 cites·14 claims
- 2195US9018204B12,4-pyrimidinediamine compounds and their usesSINGH RAJINDER·Filed 2015·Granted Apr 28, 2015·8 cites·10 claims
- 2294US9162989B22,4-Pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2015·Granted Oct 20, 2015·7 cites·9 claims
- 2394US8097630B2Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitorsSINGH RAJINDER·Filed 2007·Granted Jan 17, 2012·32 cites·10 claims
- 2494US7879856B2Diaminothiazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2007·Granted Feb 1, 2011·25 cites·22 claims
- 2593US9586908B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2015·Granted Mar 7, 2017·5 cites·10 claims
- 2693US9540334B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2015·Granted Jan 10, 2017·5 cites·18 claims
- 2793US9499493B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2015·Granted Nov 22, 2016·5 cites·17 claims
- 2893US9040550B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2014·Granted May 26, 2015·7 cites·16 claims
- 2993US8012965B2Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2007·Granted Sep 6, 2011·21 cites·6 claims
- 3093US7884119B2Triazole derivatives useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2006·Granted Feb 8, 2011·23 cites·36 claims
- 3193US7872000B2Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2007·Granted Jan 18, 2011·27 cites·53 claims
- 3292US9416112B22,4-pyrimidinediamine compounds and their usesSINGH RAJINDER·Filed 2014·Granted Aug 16, 2016·6 cites·20 claims
- 3392US8658669B2Bridged bicyclic heteroaryl substituted triazoles useful as Axl inhibitorsSINGH RAJINDER·Filed 2012·Granted Feb 25, 2014·15 cites·6 claims
- 3492US8431594B2Bridged bicyclic heteroaryl substituted triazoles useful as AXL inhibitorsSINGH RAJINDER·Filed 2009·Granted Apr 30, 2013·13 cites·3 claims
- 3592US8168636B2Polycyclic heteroaryl substituted triazoles useful as Axl inhibitorsGOFF DANE·Filed 2011·Granted May 1, 2012·13 cites·9 claims
- 3691US10314840B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2017·Granted Jun 11, 2019·3 cites·23 claims
- 3791US8563559B2Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitorsSINGH RAJINDER·Filed 2011·Granted Oct 22, 2013·16 cites·10 claims
- 3890US10369148B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2016·Granted Aug 6, 2019·3 cites·23 claims
- 3990US8741898B2Polycyclic heteroaryl substituted triazoles useful as Axl inhibitorsGOFF DANE·Filed 2012·Granted Jun 3, 2014·11 cites·15 claims
- 4090US8492373B2Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as Axl inhibitorsGOFF DANE·Filed 2010·Granted Jul 23, 2013·12 cites·4 claims
- 4190US8349838B2Polycyclic heteroaryl substituted triazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2009·Granted Jan 8, 2013·12 cites·38 claims
- 4290US7935693B2Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2007·Granted May 3, 2011·15 cites·63 claims
- 4389US8618331B2Polycyclic heteroaryl substituted triazoles useful as axl inhibitorsGOFF DANE·Filed 2010·Granted Dec 31, 2013·9 cites·23 claims
- 4489US8609650B2Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as Axl inhibitorsGOFF DANE·Filed 2011·Granted Dec 17, 2013·11 cites·12 claims
- 4588US11110082B2Tyrosine kinase inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2019·Granted Sep 7, 2021·2 cites·28 claims
- 4688US9566278B2Protein kinase C inhibitors and uses thereofRIGEL PHARMACEUTICALS INC·Filed 2015·Granted Feb 14, 2017·6 cites·21 claims
- 4788US9353126B2Substituted triazoles useful as Axl inhibitorsRIGEL PHARMACEUTICALS INC·Filed 2014·Granted May 31, 2016·8 cites·3 claims
- 4888US8546433B2Axl inhibitors for use in combination therapy for preventing, treating or managing metastatic cancerHITOSHI YASUMICHI·Filed 2010·Granted Oct 1, 2013·12 cites·10 claims
- 4988US8288382B2Diaminothiazoles useful as Axl inhibitorsGOFF DANE·Filed 2010·Granted Oct 16, 2012·14 cites·27 claims
- 5087US10709703B22,4-pyrimidinediamine compounds and their usesRIGEL PHARMACEUTICALS INC·Filed 2019·Granted Jul 14, 2020·0 cites·13 claims
Showing the top 50 of 101 patent records by PatentIndex Score.
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