Inventor · disambiguated record
Kamil Paruch
Also filed as: PARUCH KAMIL
50 granted patents·9 pending applications·434 citations·filing 2002–2023
98Inventor score
Files withSCHERING CORP38PHARMACOPEIA DRUG DISCOVERY6UNIV MASARYKOVA6GUZI TIMOTHY J5ALVAREZ CARMEN S1
Top patents by PatentIndex Score
59 records- 0194US6919341B2Imidazopyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2003·Granted Jul 19, 2005·65 cites·17 claims
- 0292US7605155B2Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Oct 20, 2009·28 cites·14 claims
- 0392US7601724B2Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Oct 13, 2009·22 cites·3 claims
- 0491US7119200B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2004·Granted Oct 10, 2006·45 cites·13 claims
- 0590US8586576B2Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitorsGUZI TIMOTHY J·Filed 2007·Granted Nov 19, 2013·15 cites·15 claims
- 0690US7196092B2N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2005·Granted Mar 27, 2007·15 cites·9 claims
- 0790US7196078B2Trisubstituted and tetrasubstituted pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORPOARTION·Filed 2005·Granted Mar 27, 2007·26 cites·29 claims
- 0889US7038045B2Pyrazolotriazines as kinase inhibitorsSCHERING CORP·Filed 2005·Granted May 2, 2006·10 cites·22 claims
- 0988US8580782B2Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitorsGUZI TIMOTHY J·Filed 2007·Granted Nov 12, 2013·14 cites·20 claims
- 1088US8211854B2Methods for inhibiting protein kinasesGUZI TIMOTHY J·Filed 2010·Granted Jul 3, 2012·12 cites·2 claims
- 1188US7205308B2Trisubstituted 7-aminopyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2005·Granted Apr 17, 2007·12 cites·14 claims
- 1288US7161003B1Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jan 9, 2007·32 cites·31 claims
- 1387US7642266B2Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Jan 5, 2010·11 cites·21 claims
- 1487US7563798B2Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Jul 21, 2009·11 cites·3 claims
- 1586US7576085B2Imidazopyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2005·Granted Aug 18, 2009·10 cites·15 claims
- 1685US8673924B2Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitorsGUZI TIMOTHY J·Filed 2007·Granted Mar 18, 2014·11 cites·25 claims
- 1785US7776865B2Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Aug 17, 2010·9 cites·37 claims
- 1885US7645762B2Substituted pyrazolo[1,5-a] pyrimidines as protein kinase inhibitorsSCHERING CORP·Filed 2006·Granted Jan 12, 2010·8 cites·31 claims
- 1984US7468372B2Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Dec 23, 2008·7 cites·13 claims
- 2082US7078525B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jul 18, 2006·15 cites·27 claims
- 2180US8603998B2Modulators of cell cycle checkpoints and their use in combination with checkpoint kinase inhibitorsGUZI TIMOTHY J·Filed 2008·Granted Dec 10, 2013·5 cites·7 claims
- 2280US7700773B24-cyano, 4-amino, and 4-aminomethyl derivatives of pyrazolo[1,5-a]pyridines, pyrazolo[1,5-c]pyrimidines and 2H-indazole compounds and 5-cyano, 5-amino, and 5-aminomethyl derivatives of imidazo[1,2-a]pyridines, and imidazo[1,5-a]pyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Apr 20, 2010·3 cites·20 claims
- 2380US7138396B217 β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2005·Granted Nov 21, 2006·3 cites·12 claims
- 2478US7452902B2Imidazopyridines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2005·Granted Nov 18, 2008·2 cites·3 claims
- 2578US6992080B2Imidazopyridines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2003·Granted Jan 31, 2006·7 cites·16 claims
- 2677US7309705B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Dec 18, 2007·2 cites·2 claims
- 2777US7084271B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Aug 1, 2006·9 cites·28 claims
- 2875US7557104B2Imidazopyrazines as protein kinase inhibitorsSCHERING CORP·Filed 2007·Granted Jul 7, 2009·2 cites·39 claims
- 2975US7186740B2Imidazopyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2003·Granted Mar 6, 2007·7 cites·18 claims
- 3074US7432268B217β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2005·Granted Oct 7, 2008·1 cites·16 claims
- 3174US7166602B2Pyrazolotriazines as kinase inhibitorsSCHERING CORP·Filed 2006·Granted Jan 23, 2007·1 cites·4 claims
- 3273US7476681B217β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2006·Granted Jan 13, 2009·1 cites·10 claims
- 3372US7514442B2Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Apr 7, 2009·1 cites·12 claims
- 3472US7067661B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jun 27, 2006·5 cites·21 claims
- 3569US6903102B217β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2002·Granted Jun 7, 2005·3 cites·29 claims
- 3667US7074924B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jul 11, 2006·2 cites·28 claims
- 3765US6969718B217-β hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2002·Granted Nov 29, 2005·2 cites·18 claims
- 3859US7511049B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2007·Granted Mar 31, 2009·0 cites·10 claims
- 3959US7354921B2Pyrazolotriazines as kinase inhibitorsSCHERING CORP·Filed 2006·Granted Apr 8, 2008·0 cites·5 claims
- 4057US7807683B2N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Oct 5, 2010·0 cites·11 claims
- 4157US2025352550A1Substituted furopyridines for therapeutic useUNIV MASARYKOVA·Filed 2023·Application pending·0 cites
- 4255US7432265B2Imidazopyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2005·Granted Oct 7, 2008·0 cites·7 claims
- 4355US2007155751A1Novel imidazopyrazines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2007·Application pending·0 cites
- 4453US7470695B2N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitorsSCHERING CORP·Filed 2006·Granted Dec 30, 2008·0 cites·12 claims
- 4553US7074795B217β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseasesSCHERING CORP·Filed 2003·Granted Jul 11, 2006·0 cites·21 claims
- 4653US2007082900A1Methods for inhibiting protein kinasesSCHERING CORP·Filed 2006·Application pending·0 cites
- 4752US2007054925A1Novel pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA INC·Filed 2006·Application pending·0 cites
- 4849US2012029204A1Synthesis of substituted-3-aminopyrazolesALVAREZ CARMEN S·Filed 2008·Application pending·0 cites
- 4949US2010143384A1NOVEL 4-CYANO, 4-AMINO, AND 4-AMINOMETHYL DERIVATIVES OF PYRAZOLO[1,5-a]PYRIDINES, PYRAZOLO[1,5-c]PYRIMIDINES AND 2H-INDAZOLE COMPOUNDS AND 5-CYANO, 5-AMINO, AND 5-AMINOMETHYL DERIVATIVES OF IMIDAZO[1,2-a]PYRIDINES, AND IMIDAZO[1,5-a]PYRAZINES AS CYCLIN DEPENDENT KINASE INHIBITORSMALLAMS ALAN K·Filed 2010·Application pending·0 cites
- 5049US2010137326A1NOVEL 4-CYANO, 4-AMINO, AND 4-AMINOMETHYL DERIVATIVES OF PYRAZOLO[1,5-a]PYRIDINES, PYRAZOLO[1,5-c]PYRIMIDINES AND 2H-INDAZOLE COMPOUNDS AND 5-CYANO, 5-AMINO, AND 5-AMINOMETHYL DERIVATIVES OF IMIDAZO[1,2-a]PYRIDINES, AND IMIDAZO[1,5-a]PYRAZINES AS CYCLIN DEPENDENT KINASE INHIBITORSSCHERING CORP·Filed 2010·Application pending·0 cites
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